PaperGreen Solid-Phase Peptide Synthesis (GSPPS) 3. Green Solvents for Fmoc Removal in Peptide Chemistry
Jad, Yahya E., Govender, Thavendran, Kruger, Hendrik G., El‐Faham, Ayman, Torre, Beatriz G. de la, Alberício, Fernando · 2017 · Organic Process Research & Development · DOI
Full title: Green Solid-Phase Peptide Synthesis (GSPPS) 3. Green Solvents for Fmoc Removal in Peptide Chemistry
Authors: Jad, Yahya E., Govender, Thavendran, Kruger, Hendrik G., El‐Faham, Ayman, Torre, Beatriz G. de la, Alberício, Fernando
PaperTwo-step hard acid deprotection/cleavage procedure for solid phase peptide synthesis.
Nomizu, M, Inagaki, Y, Yamashita, T, Ohkubo, A, Otaka, A, Fujii, N, Roller, P P, Yajima, H · 1991 · International journal of peptide and protein research · DOI
Full title: Two-step hard acid deprotection/cleavage procedure for solid phase peptide synthesis.
Authors: Nomizu, M, Inagaki, Y, Yamashita, T, Ohkubo, A, Otaka, A, Fujii, N, Roller, P P, Yajima, H
Year: 1991
Venue: International journal of peptide and protein research
PaperTailoring ultraresins based on the cross-linking of polyethylene imines. Comparative investigation of the chemical composition, the swelling, the mobility, the chemical accessibility, and the performance in solid-phase synthesis of very high loaded resins.
Barth, Michael, Rademann, Jörg · 2004 · Journal of combinatorial chemistry · DOI
Full title: Tailoring ultraresins based on the cross-linking of polyethylene imines. Comparative investigation of the chemical composition, the swelling, the mobility, the chemical accessibility, and the performance in solid-phase synthesis of very high loaded resins.
PaperDeprotection of Nin-formyl tryptophan using 1,2-ethanedithiol in liquid hydrogen fluoride. Deformylation upon HF treatment of Merrifield peptidyl-resins.
Matsueda, G R · 1982 · International journal of peptide and protein research
Full title: Deprotection of Nin-formyl tryptophan using 1,2-ethanedithiol in liquid hydrogen fluoride. Deformylation upon HF treatment of Merrifield peptidyl-resins.
Authors: Matsueda, G R
Year: 1982
Venue: International journal of peptide and protein research
PaperInfluence of resin cross-linking on solid-phase chemistry.
Rana, S, White, P, Bradley, M · 2001 · Journal of combinatorial chemistry · DOI
Full title: Influence of resin cross-linking on solid-phase chemistry.
PaperPhysical properties of poly(ethylene glycol) (PEG)-based resins for combinatorial solid phase organic chemistry: a comparison of PEG-cross-linked and PEG-grafted resins.
Grøtli, M, Gotfredsen, C H, Rademann, J, Buchardt, J, Clark, A J, Duus, J O, Meldal, M · 2000 · Journal of combinatorial chemistry · DOI
Full title: Physical properties of poly(ethylene glycol) (PEG)-based resins for combinatorial solid phase organic chemistry: a comparison of PEG-cross-linked and PEG-grafted resins.
Authors: Grøtli, M, Gotfredsen, C H, Rademann, J, Buchardt, J, Clark, A J, Duus, J O, Meldal, M
PaperSolid-phase synthesis of difficult peptide sequences at elevated temperatures: a critical comparison of microwave and conventional heating technologies.
Bacsa, Bernadett, Horváti, Kata, Bõsze, Szilvia, Andreae, Fritz, Kappe, C Oliver · 2008 · The Journal of organic chemistry · DOI
Full title: Solid-phase synthesis of difficult peptide sequences at elevated temperatures: a critical comparison of microwave and conventional heating technologies.
Authors: Bacsa, Bernadett, Horváti, Kata, Bõsze, Szilvia, Andreae, Fritz, Kappe, C Oliver
PaperEfficient macrocyclization for cyclicpeptide using solid-phase reaction.
Kim, Joonghup, Hong, Il-Khee, Kim, Hyo-Jeong, Jeong, Hyeh-Jean, Choi, Moon-Jeong, Yoon, Chang-No, Jeong, Jin-Hyun · 2002 · Archives of pharmacal research · DOI
Full title: Efficient macrocyclization for cyclicpeptide using solid-phase reaction.
Authors: Kim, Joonghup, Hong, Il-Khee, Kim, Hyo-Jeong, Jeong, Hyeh-Jean, Choi, Moon-Jeong, Yoon, Chang-No, Jeong, Jin-Hyun
PaperLarge-pore polydimethylacrylamide resin for solid-phase peptide synthesis: applications in Fmoc chemistry.
Sparrow, J T, Knieb-Cordonier, N G, Obeyseskere, N U, McMurray, J S · 1996 · Peptide research
Full title: Large-pore polydimethylacrylamide resin for solid-phase peptide synthesis: applications in Fmoc chemistry.
Authors: Sparrow, J T, Knieb-Cordonier, N G, Obeyseskere, N U, McMurray, J S
Year: 1996
Venue: Peptide research
PaperSolid-phase synthesis of neurokinin A antagonists. Comparison of the Boc and Fmoc methods.
Rovero, P, Quartara, L, Fabbri, G · 1991 · International journal of peptide and protein research
Full title: Solid-phase synthesis of neurokinin A antagonists. Comparison of the Boc and Fmoc methods.
Authors: Rovero, P, Quartara, L, Fabbri, G
Year: 1991
Venue: International journal of peptide and protein research
PaperSUBPOL: a novel SUcrose-Based Polymer support for solid-phase peptide synthesis and affinity chromatography applications.
Poschalko, Alexander, Rohr, Thomas, Gruber, Heinrich, Bianco, Alberto, Guichard, Gilles, Briand, Jean-Paul, Weber, Viktoria, Falkenhagen, Dieter · 2003 · Journal of the American Chemical Society · DOI
Full title: SUBPOL: a novel SUcrose-Based Polymer support for solid-phase peptide synthesis and affinity chromatography applications.
PaperSyntheses of four peptides from the immunodominant region of hepatitis C viral pathogens using PS-TTEGDA support for the investigation of HCV infection in human blood.
Kumar, K S, Rajasekharan Pillai, V N, Das, M R · 2000 · The journal of peptide research : official journal of the American Peptide Society · DOI
Full title: Syntheses of four peptides from the immunodominant region of hepatitis C viral pathogens using PS-TTEGDA support for the investigation of HCV infection in human blood.
Authors: Kumar, K S, Rajasekharan Pillai, V N, Das, M R
Year: 2000
Venue: The journal of peptide research : official journal of the American Peptide Society
PaperUnexpected hydrolytic instability of N-acylated amino acid amides and peptides.
Samaritoni, J Geno, Copes, Alexus T, Crews, DeMarcus K, Glos, Courtney, Thompson, Andre L, Wilson, Corydon, O'Donnell, Martin J, Scott, William L · 2014 · The Journal of organic chemistry · DOI
Full title: Unexpected hydrolytic instability of N-acylated amino acid amides and peptides.
Authors: Samaritoni, J Geno, Copes, Alexus T, Crews, DeMarcus K, Glos, Courtney, Thompson, Andre L, Wilson, Corydon, O'Donnell, Martin J, Scott, William L
PaperSPED-(styrene-polyethyleneglycol diacrylate-9-decen-1-ol): a novel resin for solid phase peptide synthesis; synthesis and characterization of biologically potent endothelin classes of peptides.
Siyad, Mohammedhaneefa A, Kumar, Gopalakrishnapillai S V · 2012 · Combinatorial chemistry & high throughput screening · DOI
Full title: SPED-(styrene-polyethyleneglycol diacrylate-9-decen-1-ol): a novel resin for solid phase peptide synthesis; synthesis and characterization of biologically potent endothelin classes of peptides.
Authors: Siyad, Mohammedhaneefa A, Kumar, Gopalakrishnapillai S V
Year: 2012
Venue: Combinatorial chemistry & high throughput screening
Nkwanyana, Nonsikelelo, Kumar, Ashish, Chakraborty, Amit, Potvin, Steeves, Thibaut-Koumba, Georges, Nardone, Brunello, Beland, Francois, Sharma, Anamika, de la Torre, Beatriz G, Albericio, Fernando · 2025 · Journal of peptide science : an official publication of the European Peptide Society · DOI
Full title: Silica-Assisted Solid-Phase Peptide Synthesis (SiPPS).
Authors: Nkwanyana, Nonsikelelo, Kumar, Ashish, Chakraborty, Amit, Potvin, Steeves, Thibaut-Koumba, Georges, Nardone, Brunello, Beland, Francois, Sharma, Anamika, de la Torre, Beatriz G, Albericio, Fernando
Year: 2025
Venue: Journal of peptide science : an official publication of the European Peptide Society
PaperSynthesis and comparative properties of two amide-generating resin linkers for use in solid phase peptide synthesis.
Deng, Fang-Kun, Mandal, Kalyaneswar, Luisier, Sam, Kent, Stephen B H · 2010 · Journal of peptide science : an official publication of the European Peptide Society · DOI
Full title: Synthesis and comparative properties of two amide-generating resin linkers for use in solid phase peptide synthesis.
Authors: Deng, Fang-Kun, Mandal, Kalyaneswar, Luisier, Sam, Kent, Stephen B H
Year: 2010
Venue: Journal of peptide science : an official publication of the European Peptide Society
PaperBypassing Osmotic Shock Dilemma in a Polystyrene Resin Using the Green Solvent Cyclopentyl methyl Ether (CPME): A Morphological Perspective.
Al Musaimi, Othman, El-Faham, Ayman, Almarhoon, Zainab, Basso, Alessandra, de la Torre, Beatriz G, Albericio, Fernando · 2019 · Polymers · DOI
Full title: Bypassing Osmotic Shock Dilemma in a Polystyrene Resin Using the Green Solvent Cyclopentyl methyl Ether (CPME): A Morphological Perspective.
Authors: Al Musaimi, Othman, El-Faham, Ayman, Almarhoon, Zainab, Basso, Alessandra, de la Torre, Beatriz G, Albericio, Fernando
PaperPalladium(0)-catalyzed coupling-cyclization reaction of polymer-supported aryl iodides with 1,2-allenyl carboxylic acids. Solid-phase parallel synthesis of butenolides.
Ma, Shengming, Duan, Dehui, Wang, Yizhong · 2002 · Journal of combinatorial chemistry · DOI
Full title: Palladium(0)-catalyzed coupling-cyclization reaction of polymer-supported aryl iodides with 1,2-allenyl carboxylic acids. Solid-phase parallel synthesis of butenolides.
PaperOptimized aminolysis conditions for cleavage of N-protected hydrophobic peptides from solid-phase resins.
Greathouse, D V, Goforth, R L, Crawford, T, Van Der Wel, P C, Killian, J A · 2001 · The journal of peptide research : official journal of the American Peptide Society · DOI
Full title: Optimized aminolysis conditions for cleavage of N-protected hydrophobic peptides from solid-phase resins.
Authors: Greathouse, D V, Goforth, R L, Crawford, T, Van Der Wel, P C, Killian, J A
Year: 2001
Venue: The journal of peptide research : official journal of the American Peptide Society
PaperOptimization of peptide synthesis time and sustainability using novel eco-friendly binary solvent systems with induction heating on an automated peptide synthesizer.
Pacini, Lorenzo, Muthyala, Manoj, Aguiar, Luisa, Zitterbart, Robert, Rovero, Paolo, Papini, Anna Maria · 2024 · Journal of peptide science : an official publication of the European Peptide Society · DOI
Full title: Optimization of peptide synthesis time and sustainability using novel eco-friendly binary solvent systems with induction heating on an automated peptide synthesizer.
Authors: Pacini, Lorenzo, Muthyala, Manoj, Aguiar, Luisa, Zitterbart, Robert, Rovero, Paolo, Papini, Anna Maria
Year: 2024
Venue: Journal of peptide science : an official publication of the European Peptide Society
PaperA modified Arg-Asp-Val (RDV) peptide derived during the synthesis of Arg-Glu-Asp-Val (REDV), a tetrapeptide derived from an alternatively spliced site in fibronectin, inhibits the binding of fibrinogen, fibronectin, von Willebrand factor and vitronectin to activated platelets.
Chen, C S, Papayannopoulos, I A, Timmons, S, Chou, S H, Thiagarajan, P · 1991 · Biochimica et biophysica acta · DOI
Full title: A modified Arg-Asp-Val (RDV) peptide derived during the synthesis of Arg-Glu-Asp-Val (REDV), a tetrapeptide derived from an alternatively spliced site in fibronectin, inhibits the binding of fibrinogen, fibronectin, von Willebrand factor and vitronectin to activated platelets.
Authors: Chen, C S, Papayannopoulos, I A, Timmons, S, Chou, S H, Thiagarajan, P
PaperSynthesis of protected secretin 16-27 on a Merrifield resin. Examination of ammonolysis conditions for preparing carboxamide terminal protected peptides suitable for fragment condensation.
Wright, D E, Agarwal, N S, Hruby, V J · 1980 · International journal of peptide and protein research
Full title: Synthesis of protected secretin 16-27 on a Merrifield resin. Examination of ammonolysis conditions for preparing carboxamide terminal protected peptides suitable for fragment condensation.
Authors: Wright, D E, Agarwal, N S, Hruby, V J
Year: 1980
Venue: International journal of peptide and protein research
PaperResin Swelling in Mixed Solvents Analysed using Hansen Solubility Parameter Space.
Ran, Yanrui, Byrne, Fergal, Ingram, Ian D V, North, Michael · 2019 · Chemistry (Weinheim an der Bergstrasse, Germany) · DOI
Full title: Resin Swelling in Mixed Solvents Analysed using Hansen Solubility Parameter Space.
Authors: Ran, Yanrui, Byrne, Fergal, Ingram, Ian D V, North, Michael
Year: 2019
Venue: Chemistry (Weinheim an der Bergstrasse, Germany)
PaperSyntheses, characterization and application of cross-linked polystyrene-ethyleneglycol acrylate resin (CLPSER) as a novel polymer support for polypeptide syntheses.
Leena, S, Kumar, K S · 2001 · The journal of peptide research : official journal of the American Peptide Society · DOI
Full title: Syntheses, characterization and application of cross-linked polystyrene-ethyleneglycol acrylate resin (CLPSER) as a novel polymer support for polypeptide syntheses.
Authors: Leena, S, Kumar, K S
Year: 2001
Venue: The journal of peptide research : official journal of the American Peptide Society
PaperChemistry of alpha-hydroxymethylserine: problems and solutions.
Stasiak, Marcin, Słomczyńska, Urszula, Olma, Aleksandra, Leplawy, Mirosław T · 2008 · Journal of peptide science : an official publication of the European Peptide Society · DOI
Full title: Chemistry of alpha-hydroxymethylserine: problems and solutions.
Authors: Stasiak, Marcin, Słomczyńska, Urszula, Olma, Aleksandra, Leplawy, Mirosław T
Year: 2008
Venue: Journal of peptide science : an official publication of the European Peptide Society
PaperSynthesis of the protected tridecapeptide (56-68) of the VH domain of mouse myeloma immunoglobulin M603 and its reattachment to resin supports.
Voss, C, Dimarchi, R, Whitney, D B, Tjoeng, F S, Merrifield, R B, Tam, J P · 1983 · International journal of peptide and protein research · DOI
Full title: Synthesis of the protected tridecapeptide (56-68) of the VH domain of mouse myeloma immunoglobulin M603 and its reattachment to resin supports.
Authors: Voss, C, Dimarchi, R, Whitney, D B, Tjoeng, F S, Merrifield, R B, Tam, J P
Year: 1983
Venue: International journal of peptide and protein research
PaperMechanistic Study of Diketopiperazine Formation during Solid-Phase Peptide Synthesis of Tirzepatide.
Wang, Jingyao, Berglund, Mark R, Braden, Timothy, Embry, Matthew C, Johnson, Martin D, Groskreutz, Stephen R, Sayyed, Fareed Bhasha, Tsukanov, Sergey Vladimirovich, White, Timothy D, Jalan, Ankur, Seibert, Kevin D, Kopach, Michael E · 2022 · ACS omega · DOI
Full title: Mechanistic Study of Diketopiperazine Formation during Solid-Phase Peptide Synthesis of Tirzepatide.
Authors: Wang, Jingyao, Berglund, Mark R, Braden, Timothy, Embry, Matthew C, Johnson, Martin D, Groskreutz, Stephen R, Sayyed, Fareed Bhasha, Tsukanov, Sergey Vladimirovich, White, Timothy D, Jalan, Ankur, Seibert, Kevin D, Kopach, Michael E
PaperSynthetic Evaluation of Standard and Microwave-Assisted Solid Phase Peptide Synthesis of a Long Chimeric Peptide Derived from Four Plasmodium falciparum Proteins.
Varela, Yahson F, Vanegas Murcia, Magnolia, Patarroyo, Manuel Elkin · 2018 · Molecules (Basel, Switzerland) · DOI
Full title: Synthetic Evaluation of Standard and Microwave-Assisted Solid Phase Peptide Synthesis of a Long Chimeric Peptide Derived from Four Plasmodium falciparum Proteins.
Authors: Varela, Yahson F, Vanegas Murcia, Magnolia, Patarroyo, Manuel Elkin
PaperExpanding the scope of sustainable peptide synthesis through post-linear synthesis reactions.
Malone, Michael A, De Francisco Craparotta, Matilde, Arnott, Kirsty I M, Jamieson, Andrew G, Wade, Nicola · 2026 · Organic & biomolecular chemistry · DOI
Full title: Expanding the scope of sustainable peptide synthesis through post-linear synthesis reactions.
Authors: Malone, Michael A, De Francisco Craparotta, Matilde, Arnott, Kirsty I M, Jamieson, Andrew G, Wade, Nicola
PaperComparative evaluation of four trityl-type amidomethyl polystyrene resins in Fmoc solid phase peptide synthesis.
Zikos, Christos, Livaniou, Evangelia, Leondiadis, Leondios, Ferderigos, Nikolas, Ithakissios, Dionyssis S, Evangelatos, Gregory P · 2003 · Journal of peptide science : an official publication of the European Peptide Society · DOI
Full title: Comparative evaluation of four trityl-type amidomethyl polystyrene resins in Fmoc solid phase peptide synthesis.
PaperSuccessful synthesis of a glial-specific blood-brain barrier shuttle peptide following a fragment condensation approach on a solid-phase resin.
Al Musaimi, Othman, Morse, Sophie V, Lombardi, Lucia, Serban, Simona, Basso, Alessandra, Williams, Daryl R · 2023 · Journal of peptide science : an official publication of the European Peptide Society · DOI
Full title: Successful synthesis of a glial-specific blood-brain barrier shuttle peptide following a fragment condensation approach on a solid-phase resin.
Authors: Al Musaimi, Othman, Morse, Sophie V, Lombardi, Lucia, Serban, Simona, Basso, Alessandra, Williams, Daryl R
Year: 2023
Venue: Journal of peptide science : an official publication of the European Peptide Society
PaperPreparation of tri(ethylene glycol) grafted core-shell type polymer support for solid-phase peptide synthesis.
Kim, Jaehi, Kim, Seojung, Shin, Dong-Sik, Lee, Yoon-Sik · 2018 · Journal of peptide science : an official publication of the European Peptide Society · DOI
Full title: Preparation of tri(ethylene glycol) grafted core-shell type polymer support for solid-phase peptide synthesis.
Authors: Kim, Jaehi, Kim, Seojung, Shin, Dong-Sik, Lee, Yoon-Sik
Year: 2018
Venue: Journal of peptide science : an official publication of the European Peptide Society
PaperSolid-Phase Synthesis of Oligopeptides Containing Sterically Hindered Amino Acids on Nonswellable Resin Using 3-Nitro-1,2,4-triazol-1-yl-tris(pyrrolidin-1-yl)phosphonium Hexafluorophosphate (PyNTP) as the Condensing Reagent.
Full title: Solid-Phase Synthesis of Oligopeptides Containing Sterically Hindered Amino Acids on Nonswellable Resin Using 3-Nitro-1,2,4-triazol-1-yl-tris(pyrrolidin-1-yl)phosphonium Hexafluorophosphate (PyNTP) as the Condensing Reagent.
PaperHigh-yield, solid-phase synthesis of humanin, an Alzheimer's disease associated, novel 24-mer peptide which contains a difficult sequence.
Evangelou, Alexandra, Zikos, Christos, Livaniou, Evangelia, Evangelatos, Gregory P · 2004 · Journal of peptide science : an official publication of the European Peptide Society · DOI
Full title: High-yield, solid-phase synthesis of humanin, an Alzheimer's disease associated, novel 24-mer peptide which contains a difficult sequence.
Authors: Evangelou, Alexandra, Zikos, Christos, Livaniou, Evangelia, Evangelatos, Gregory P
Year: 2004
Venue: Journal of peptide science : an official publication of the European Peptide Society
PaperSolid-phase synthesis of cyclic analogues related to the hypoglycaemic peptide hGH(6-13): comparison of two i-->i + 4 lactam cyclization procedures.
Cavallaro, V, Thompson, P E, Hearn, M T · 2001 · Journal of peptide science : an official publication of the European Peptide Society · DOI
Full title: Solid-phase synthesis of cyclic analogues related to the hypoglycaemic peptide hGH(6-13): comparison of two i-->i + 4 lactam cyclization procedures.
Authors: Cavallaro, V, Thompson, P E, Hearn, M T
Year: 2001
Venue: Journal of peptide science : an official publication of the European Peptide Society
PaperApplication of arylsulphonyl side-chain protected arginines in solid-phase peptide synthesis based on 9-fluorenylmethoxycarbonyl amino protecting strategy.
Fischer, P M, Retson, K V, Tyler, M I, Howden, M E · 1992 · International journal of peptide and protein research · DOI
Full title: Application of arylsulphonyl side-chain protected arginines in solid-phase peptide synthesis based on 9-fluorenylmethoxycarbonyl amino protecting strategy.
Authors: Fischer, P M, Retson, K V, Tyler, M I, Howden, M E
Year: 1992
Venue: International journal of peptide and protein research
PaperN-Butylpyrrolidinone is an equally good solvent as N,N-dimethylformamide for microwave assisted solid phase peptide synthesis.
Öhlander, Andrea, Lüdtke, Carsten, Sahakjan, Artur, Johnsson, Richard E · 2024 · Journal of peptide science : an official publication of the European Peptide Society · DOI
Full title: N-Butylpyrrolidinone is an equally good solvent as N,N-dimethylformamide for microwave assisted solid phase peptide synthesis.
Authors: Öhlander, Andrea, Lüdtke, Carsten, Sahakjan, Artur, Johnsson, Richard E
Year: 2024
Venue: Journal of peptide science : an official publication of the European Peptide Society
PaperSynthesis of N-tert.-butoxycarbonyl-( alpha-phenyl)aminomethylphenoxyacetic acid for use as a handle in solid-phase synthesis of peptide alpha-carboxamides.
Gaehde, S A, Matsueda, G R · 1981 · International journal of peptide and protein research · DOI
Full title: Synthesis of N-tert.-butoxycarbonyl-( alpha-phenyl)aminomethylphenoxyacetic acid for use as a handle in solid-phase synthesis of peptide alpha-carboxamides.
Authors: Gaehde, S A, Matsueda, G R
Year: 1981
Venue: International journal of peptide and protein research
PaperSynthesis of [1-8-NαC]-zanriorb A1, alanine-containing analogues, and their cytotoxic and anti-inflammatory activity.
Nadeem-Ul-Haque, Muhammad, Bashir, Anila, Karim, Humira, Khan, Sadiq Noor, Shah, Zafar Ali, Jabeen, Almas, Qayyum, Shaista, Ganesan, A, Choudhary, M Iqbal, Shaheen, Farzana · 2022 · Journal of peptide science : an official publication of the European Peptide Society · DOI
Full title: Synthesis of [1-8-NαC]-zanriorb A1, alanine-containing analogues, and their cytotoxic and anti-inflammatory activity.
Authors: Nadeem-Ul-Haque, Muhammad, Bashir, Anila, Karim, Humira, Khan, Sadiq Noor, Shah, Zafar Ali, Jabeen, Almas, Qayyum, Shaista, Ganesan, A, Choudhary, M Iqbal, Shaheen, Farzana
Year: 2022
Venue: Journal of peptide science : an official publication of the European Peptide Society
PaperImproved loading and cleavage methods for solid-phase synthesis using chlorotrityl resins: synthesis and testing of a library of 144 discrete chemicals as potential farnesyltransferase inhibitors.
Park, Jewn Giew, Langenwalter, Kevin J, Weinbaum, Carolyn A, Casey, Patrick J, Pang, Yuan-Ping · 2004 · Journal of combinatorial chemistry · DOI
Full title: Improved loading and cleavage methods for solid-phase synthesis using chlorotrityl resins: synthesis and testing of a library of 144 discrete chemicals as potential farnesyltransferase inhibitors.
Authors: Park, Jewn Giew, Langenwalter, Kevin J, Weinbaum, Carolyn A, Casey, Patrick J, Pang, Yuan-Ping
PaperConformational studies on beta-amyloid protein carboxy-terminal region (residues 34-42): strategic use of amide backbone protection as a structural probe.
Quibell, M, Johnson, T, Turnell, W G · 1994 · Biomedical peptides, proteins & nucleic acids : structure, synthesis & biological activity
Full title: Conformational studies on beta-amyloid protein carboxy-terminal region (residues 34-42): strategic use of amide backbone protection as a structural probe.
PaperSynthesis and high performance liquid chromatography/electrospray mass spectrometry single-bead decoding of split-pool structural libraries of polyamines supported on polystyrene and polystyrene/ethylene glycol resins.
Manku, Sukhdev, Wang, Fan, Hall, Dennis G · 2003 · Journal of combinatorial chemistry · DOI
Full title: Synthesis and high performance liquid chromatography/electrospray mass spectrometry single-bead decoding of split-pool structural libraries of polyamines supported on polystyrene and polystyrene/ethylene glycol resins.
Authors: Manku, Sukhdev, Wang, Fan, Hall, Dennis G
PaperToward a Green SPPS: The Use of an Innovative Mesoporous pDVB Support for Environmentally Friendly Solvents.
Lastella, Luana, Zecca, Marco, Centomo, Paolo, Jeřábek, Karel, Formaggio, Fernando, Guryanov, Ivan, Ricci, Antonio, Biondi, Barbara · 2025 · Journal of peptide science : an official publication of the European Peptide Society · DOI
Full title: Toward a Green SPPS: The Use of an Innovative Mesoporous pDVB Support for Environmentally Friendly Solvents.
PaperRegioselective formation of the three disulfide bonds of a 35-residue insect peptide.
Kellenberger, C, Hietter, H, Luu, B · 1995 · Peptide research
Full title: Regioselective formation of the three disulfide bonds of a 35-residue insect peptide.
Authors: Kellenberger, C, Hietter, H, Luu, B
Year: 1995
Venue: Peptide research
PaperBrønsted Acid-Lewis Acid (BA-LA) Induced Final Deprotection/Peptide Resin Cleavage in Fmoc/t-Bu Solid-Phase Peptide Synthesis: HCl/FeCl3 and AcOH/FeCl3 as Viable PFAS-Free Alternatives for TFA.
Pawlas, Jan, André, Christophe, Rasmussen, Jon H, Ludemann-Hombourger, Olivier · 2024 · Organic letters · DOI
Full title: Brønsted Acid-Lewis Acid (BA-LA) Induced Final Deprotection/Peptide Resin Cleavage in Fmoc/t-Bu Solid-Phase Peptide Synthesis: HCl/FeCl3 and AcOH/FeCl3 as Viable PFAS-Free Alternatives for TFA.
Authors: Pawlas, Jan, André, Christophe, Rasmussen, Jon H, Ludemann-Hombourger, Olivier
PaperSynthesis of insulin-like growth factor I using N-methyl pyrrolidinone as the coupling solvent and trifluoromethane sulphonic acid cleavage from the resin.
Bagley, C J, Otteson, K M, May, B L, McCurdy, S N, Pierce, L, Ballard, F J, Wallace, J C · 1990 · International journal of peptide and protein research · DOI
Full title: Synthesis of insulin-like growth factor I using N-methyl pyrrolidinone as the coupling solvent and trifluoromethane sulphonic acid cleavage from the resin.
Authors: Bagley, C J, Otteson, K M, May, B L, McCurdy, S N, Pierce, L, Ballard, F J, Wallace, J C
Year: 1990
Venue: International journal of peptide and protein research
Full title: Quantitative and Nondestructive Colorimetric Amine Detection Method for the Solid-Phase Peptide Synthesis as an Alternative to the Kaiser Test.
PaperThe Significance of Oligomer C-Terminus Design in Solid-Phase Synthesis of Peptide Nucleic Acid Tetramers With the Incorporation of γ-S-Monomer Units Based on L-Glu.
Esenina, Anna A, Prohorov, Ivan A, Severov, Viacheslav V, Smirnov, Igor P, Luzyanin, Timofey A, Kirillova, Yulia G · 2025 · Journal of peptide science : an official publication of the European Peptide Society · DOI
Full title: The Significance of Oligomer C-Terminus Design in Solid-Phase Synthesis of Peptide Nucleic Acid Tetramers With the Incorporation of γ-S-Monomer Units Based on L-Glu.
Authors: Esenina, Anna A, Prohorov, Ivan A, Severov, Viacheslav V, Smirnov, Igor P, Luzyanin, Timofey A, Kirillova, Yulia G
Year: 2025
Venue: Journal of peptide science : an official publication of the European Peptide Society
PaperMicrowave-assisted TFA cleavage of peptides from Merrifield resin.
Kluczyk, Alicja, Rudowska, Magdalena, Stefanowicz, Piotr, Szewczuk, Zbigniew · 2010 · Journal of peptide science : an official publication of the European Peptide Society · DOI
Full title: Microwave-assisted TFA cleavage of peptides from Merrifield resin.
Authors: Kluczyk, Alicja, Rudowska, Magdalena, Stefanowicz, Piotr, Szewczuk, Zbigniew
Year: 2010
Venue: Journal of peptide science : an official publication of the European Peptide Society
PaperEnantioselective synthesis of (2R, 3S)- and (2S, 3R)-4,4,4-trifluoro-N-Fmoc-O-tert-butyl-threonine and their racemization-free incorporation into oligopeptides via solid-phase synthesis.
Xiao, Nu, Jiang, Zhong-Xing, Yu, Y Bruce · 2007 · Biopolymers · DOI
Full title: Enantioselective synthesis of (2R, 3S)- and (2S, 3R)-4,4,4-trifluoro-N-Fmoc-O-tert-butyl-threonine and their racemization-free incorporation into oligopeptides via solid-phase synthesis.
PaperInvestigation of the automated solid-phase synthesis of a 38mer peptide with difficult sequence pattern under different synthesis strategies.
Winkler, Dirk F H, Tian, Kerry · 2015 · Amino acids · DOI
Full title: Investigation of the automated solid-phase synthesis of a 38mer peptide with difficult sequence pattern under different synthesis strategies.
PaperPeptide engineering - controlling the folding of disulfide-rich peptides
Muttenthaler, Markus · 2009 · Queensland's institutional digital repository (The University of Queensland)
Full title: Peptide engineering - controlling the folding of disulfide-rich peptides
Authors: Muttenthaler, Markus
Year: 2009
Venue: Queensland's institutional digital repository (The University of Queensland)
PaperSynthesis, characterization, and evaluation of PS-PPDC resin: a novel flexible cross-linked polymeric support for solid-phase organic synthesis.
Siyad, M A, Vinod Kumar, G S · 2012 · Biopolymers · DOI
Full title: Synthesis, characterization, and evaluation of PS-PPDC resin: a novel flexible cross-linked polymeric support for solid-phase organic synthesis.
PaperCombining a polar resin and a pseudo-proline to optimize the solid-phase synthesis of a 'difficult sequence'.
Cremer, Gaëlle-Anne, Tariq, Hanane, Delmas, Agnes F · 2006 · Journal of peptide science : an official publication of the European Peptide Society · DOI
Full title: Combining a polar resin and a pseudo-proline to optimize the solid-phase synthesis of a 'difficult sequence'.
Authors: Cremer, Gaëlle-Anne, Tariq, Hanane, Delmas, Agnes F
Year: 2006
Venue: Journal of peptide science : an official publication of the European Peptide Society
PaperDevelopment of a Single-Chain Peptide Agonist of the Relaxin-3 Receptor Using Hydrocarbon Stapling.
Hojo, Keiko, Hossain, Mohammed Akhter, Tailhades, Julien, Shabanpoor, Fazel, Wong, Lilian L L, Ong-Pålsson, Emma E K, Kastman, Hanna E, Ma, Sherie, Gundlach, Andrew L, Rosengren, K Johan, Wade, John D, Bathgate, Ross A D · 2016 · Journal of medicinal chemistry · DOI
Full title: Development of a Single-Chain Peptide Agonist of the Relaxin-3 Receptor Using Hydrocarbon Stapling.
Authors: Hojo, Keiko, Hossain, Mohammed Akhter, Tailhades, Julien, Shabanpoor, Fazel, Wong, Lilian L L, Ong-Pålsson, Emma E K, Kastman, Hanna E, Ma, Sherie, Gundlach, Andrew L, Rosengren, K Johan, Wade, John D, Bathgate, Ross A D
PaperSynbeads Porous-Rigid Methacrylic Support: Application to Solid Phase Peptide Synthesis and Characterization of the Polymeric Matrix by FTIR Microspectroscopy and High Resolution Magic Angle Spinning NMR
Full title: Synbeads Porous-Rigid Methacrylic Support: Application to Solid Phase Peptide Synthesis and Characterization of the Polymeric Matrix by FTIR Microspectroscopy and High Resolution Magic Angle Spinning NMR
Paper[The synthesis of immunomodulating peptide alloferon, the active component of the antiviral drug allokine-alpha].
Sidorova, M V, Molokoedov, A S, Kudriavtseva, E V, Baldin, M I, Frid, D A, Ovchinnikov, M V, Bespalova, Zh D, Bushuev, V N · 2006 · Bioorganicheskaia khimiia
Full title: [The synthesis of immunomodulating peptide alloferon, the active component of the antiviral drug allokine-alpha].
Authors: Sidorova, M V, Molokoedov, A S, Kudriavtseva, E V, Baldin, M I, Frid, D A, Ovchinnikov, M V, Bespalova, Zh D, Bushuev, V N
Year: 2006
Venue: Bioorganicheskaia khimiia
PaperStudy of the effect of the peptide loading and solvent system in SPPS by HRMAS-NMR.
Valente, Ana P, Almeida, Fábio C L, Nakaie, Clovis R, Schreier, Shirley, Crusca, Edson, Cilli, Eduardo M · 2005 · Journal of peptide science : an official publication of the European Peptide Society · DOI
Full title: Study of the effect of the peptide loading and solvent system in SPPS by HRMAS-NMR.
Authors: Valente, Ana P, Almeida, Fábio C L, Nakaie, Clovis R, Schreier, Shirley, Crusca, Edson, Cilli, Eduardo M
Year: 2005
Venue: Journal of peptide science : an official publication of the European Peptide Society
PaperSolid-phase synthesis of a nucleopeptide from the linking site of adenovirus-2 nucleoprotein, -Ser(p5'CATCAT)-Gly-Asp-. Convergent versus stepwise strategy.
Robles, J, Pedroso, E, Grandas, A · 1995 · Nucleic acids research · DOI
Full title: Solid-phase synthesis of a nucleopeptide from the linking site of adenovirus-2 nucleoprotein, -Ser(p5'CATCAT)-Gly-Asp-. Convergent versus stepwise strategy.
PaperImproving the performance of an acid-labile 4-hydroxymethyl phenoxyacetic acid (HMP) linker on resin and SynPhase grafted solid-supports.
Bui, C T, Ercole, F, Pham, Y, Campbell, R, Rasoul, F A, Maeji, N J, Ede, N J · 2000 · Journal of peptide science : an official publication of the European Peptide Society · DOI
Full title: Improving the performance of an acid-labile 4-hydroxymethyl phenoxyacetic acid (HMP) linker on resin and SynPhase grafted solid-supports.
Authors: Bui, C T, Ercole, F, Pham, Y, Campbell, R, Rasoul, F A, Maeji, N J, Ede, N J
Year: 2000
Venue: Journal of peptide science : an official publication of the European Peptide Society
PaperSolid phase synthesis of the protected 43-55 tridecapeptide of the heavy chain of myeloma immunoglobin M603, employing cyclohexyl ester protection for glutamic acid.
Dimarchi, R D, Tam, J P, Merrifield, R B · 1982 · International journal of peptide and protein research · DOI
Full title: Solid phase synthesis of the protected 43-55 tridecapeptide of the heavy chain of myeloma immunoglobin M603, employing cyclohexyl ester protection for glutamic acid.
Authors: Dimarchi, R D, Tam, J P, Merrifield, R B
Year: 1982
Venue: International journal of peptide and protein research
PaperPeptide synthesis in water IV. Preparation of N-ethanesulfonylethoxycarbonyl (Esc) amino acids and their application to solid phase peptide synthesis.
Full title: Peptide synthesis in water IV. Preparation of N-ethanesulfonylethoxycarbonyl (Esc) amino acids and their application to solid phase peptide synthesis.
PaperProtected peptide disulfides by oxidative detachment from a support.
Rietman, B H, Smulders, R H, Eggen, I F, van Vliet, A, van de Werken, G, Tesser, G I · 1994 · International journal of peptide and protein research · DOI
Full title: Protected peptide disulfides by oxidative detachment from a support.
Authors: Rietman, B H, Smulders, R H, Eggen, I F, van Vliet, A, van de Werken, G, Tesser, G I
Year: 1994
Venue: International journal of peptide and protein research
PaperConformational origin of a difficult coupling in a human growth hormone releasing factor analog.
Deber, C M, Lutek, M K, Heimer, E P, Felix, A M · 1989 · Peptide research
Full title: Conformational origin of a difficult coupling in a human growth hormone releasing factor analog.
Authors: Deber, C M, Lutek, M K, Heimer, E P, Felix, A M
Year: 1989
Venue: Peptide research
PaperSolid-phase synthesis and on-resin cyclization of a disulfide bond peptide and lactam analogues corresponding to the major antigenic site of HIV gp41 protein.
Limal, D, Briand, J P, Dalbon, P, Jolivet, M · 1998 · The journal of peptide research : official journal of the American Peptide Society · DOI
Full title: Solid-phase synthesis and on-resin cyclization of a disulfide bond peptide and lactam analogues corresponding to the major antigenic site of HIV gp41 protein.
Authors: Limal, D, Briand, J P, Dalbon, P, Jolivet, M
Year: 1998
Venue: The journal of peptide research : official journal of the American Peptide Society
PaperPeptide synthesis beyond DMF: THF and ACN as excellent and friendlier alternatives.
Jad, Yahya E, Acosta, Gerardo A, Khattab, Sherine N, de la Torre, Beatriz G, Govender, Thavendran, Kruger, Hendrik G, El-Faham, Ayman, Albericio, Fernando · 2015 · Organic & biomolecular chemistry · DOI
Full title: Peptide synthesis beyond DMF: THF and ACN as excellent and friendlier alternatives.
Authors: Jad, Yahya E, Acosta, Gerardo A, Khattab, Sherine N, de la Torre, Beatriz G, Govender, Thavendran, Kruger, Hendrik G, El-Faham, Ayman, Albericio, Fernando
PaperEvaluation of the trifluoromethanosulfonic acid/trifluoroacetic acid/thioanisole cleavage procedure for application in solid-phase peptide synthesis.
Jubilut, G N, Cilli, E M, Tominaga, M, Miranda, A, Okada, Y, Nakaie, C R · 2001 · Chemical & pharmaceutical bulletin · DOI
Full title: Evaluation of the trifluoromethanosulfonic acid/trifluoroacetic acid/thioanisole cleavage procedure for application in solid-phase peptide synthesis.
Authors: Jubilut, G N, Cilli, E M, Tominaga, M, Miranda, A, Okada, Y, Nakaie, C R
PaperSolid-phase synthesis of cionin, a protochordate-derived octapeptide related to the gastrin/cholecystokinin family of peptides, and its mono-tyrosine-sulfate-containing derivatives.
Kitagawa, K, Futaki, S, Yagami, T, Sumi, S, Inoue, K · 1994 · International journal of peptide and protein research · DOI
Full title: Solid-phase synthesis of cionin, a protochordate-derived octapeptide related to the gastrin/cholecystokinin family of peptides, and its mono-tyrosine-sulfate-containing derivatives.
Pantarotto, Davide, Bianco, Alberto, Pellarini, Federica, Tossi, Alessandro, Giangaspero, Anna, Zelezetsky, Igor, Briand, Jean-Paul, Prato, Maurizio · 2002 · Journal of the American Chemical Society · DOI
Full title: Solid-phase synthesis of fullerene-peptides.
PaperA backbone amide protecting group for overcoming difficult sequences and suppressing aspartimide formation.
Abdel-Aal, Abu-Baker M, Papageorgiou, George, Raz, Richard, Quibell, Martin, Burlina, Fabienne, Offer, John · 2016 · Journal of peptide science : an official publication of the European Peptide Society · DOI
Full title: A backbone amide protecting group for overcoming difficult sequences and suppressing aspartimide formation.
Authors: Abdel-Aal, Abu-Baker M, Papageorgiou, George, Raz, Richard, Quibell, Martin, Burlina, Fabienne, Offer, John
Year: 2016
Venue: Journal of peptide science : an official publication of the European Peptide Society
Paper[Side reactions in peptide synthesis. V. O-sulfonation of serine and threonine during removal of pmc- and mtr-protecting groups from arginine residues in fmoc-solid phase synthesis].
Jaeger, E, Remmer, H A, Jung, G, Metzger, J, Oberthür, W, Rücknagel, K P, Schäfer, W, Sonnenbichler, J, Zetl, I · 1993 · Biological chemistry Hoppe-Seyler
Full title: [Side reactions in peptide synthesis. V. O-sulfonation of serine and threonine during removal of pmc- and mtr-protecting groups from arginine residues in fmoc-solid phase synthesis].
Authors: Jaeger, E, Remmer, H A, Jung, G, Metzger, J, Oberthür, W, Rücknagel, K P, Schäfer, W, Sonnenbichler, J, Zetl, I
Year: 1993
Venue: Biological chemistry Hoppe-Seyler
PaperSolid phase synthesis of porcine LH-releasing hormone with hydrogen chloride in formic acid as the deblocking reagent.
Yonezawa, H, Takahashi, N, Ohno, M, Izumiya, N · 1978 · International journal of peptide and protein research · DOI
Full title: Solid phase synthesis of porcine LH-releasing hormone with hydrogen chloride in formic acid as the deblocking reagent.
Authors: Yonezawa, H, Takahashi, N, Ohno, M, Izumiya, N
Year: 1978
Venue: International journal of peptide and protein research
Paper2-Methyltetrahydrofuran and cyclopentyl methyl ether for green solid-phase peptide synthesis.
Jad, Yahya E, Acosta, Gerardo A, Khattab, Sherine N, de la Torre, Beatriz G, Govender, Thavendran, Kruger, Hendrik G, El-Faham, Ayman, Albericio, Fernando · 2016 · Amino acids · DOI
Full title: 2-Methyltetrahydrofuran and cyclopentyl methyl ether for green solid-phase peptide synthesis.
Authors: Jad, Yahya E, Acosta, Gerardo A, Khattab, Sherine N, de la Torre, Beatriz G, Govender, Thavendran, Kruger, Hendrik G, El-Faham, Ayman, Albericio, Fernando
PaperNew t-butyl based aspartate protecting groups preventing aspartimide formation in Fmoc SPPS.
Behrendt, Raymond, Huber, Simon, Martí, Roger, White, Peter · 2015 · Journal of peptide science : an official publication of the European Peptide Society · DOI
Full title: New t-butyl based aspartate protecting groups preventing aspartimide formation in Fmoc SPPS.
Authors: Behrendt, Raymond, Huber, Simon, Martí, Roger, White, Peter
Year: 2015
Venue: Journal of peptide science : an official publication of the European Peptide Society
PaperAmino acids and peptides. XXXI. Preparation of analogs of the laminin-related peptide YIGSR and their inhibitory effect on experimental metastasis.
Maeda, M, Izuno, Y, Kawasaki, K, Kaneda, Y, Mu, Y, Tsutsumi, Y, Nakagawa, S, Mayumi, T · 1998 · Chemical & pharmaceutical bulletin · DOI
Full title: Amino acids and peptides. XXXI. Preparation of analogs of the laminin-related peptide YIGSR and their inhibitory effect on experimental metastasis.
Authors: Maeda, M, Izuno, Y, Kawasaki, K, Kaneda, Y, Mu, Y, Tsutsumi, Y, Nakagawa, S, Mayumi, T
PaperComparative investigation of the cleavage step in the synthesis of model peptide resins: implications for Nalpha-9-fluorenylmethyloxycarbonyl-solid phase peptide synthesis.
Jubilut, Guita Nicolaewsky, Cilli, Eduardo Maffud, Crusca, Edson, Silva, Elias Horacio, Okada, Yoshio, Nakaie, Clovis Ryuichi · 2007 · Chemical & pharmaceutical bulletin · DOI
Full title: Comparative investigation of the cleavage step in the synthesis of model peptide resins: implications for Nalpha-9-fluorenylmethyloxycarbonyl-solid phase peptide synthesis.
PaperSolid phase synthesis of the protected 27--42 hexadecapeptide of the heavy chain from myeloma immunoglobulin M603. Elimination of side reactions associated with glycyl-2-oxypropionyl-resin.
Tjoeng, F S, Tam, J P, Merrifield, R B · 1979 · International journal of peptide and protein research · DOI
Full title: Solid phase synthesis of the protected 27--42 hexadecapeptide of the heavy chain from myeloma immunoglobulin M603. Elimination of side reactions associated with glycyl-2-oxypropionyl-resin.
Authors: Tjoeng, F S, Tam, J P, Merrifield, R B
Year: 1979
Venue: International journal of peptide and protein research
PaperFunctionalized Spirocyclic Heterocycle Synthesis and Cytotoxicity Assay.
Gray, Amelia N, Ramirez, Breeana M, Mawugbe, Selom K, Mar, Jordan F, Wong, Yun-Lan C, Huang, Kevin S · 2021 · Journal of visualized experiments : JoVE · DOI
Full title: Functionalized Spirocyclic Heterocycle Synthesis and Cytotoxicity Assay.
Authors: Gray, Amelia N, Ramirez, Breeana M, Mawugbe, Selom K, Mar, Jordan F, Wong, Yun-Lan C, Huang, Kevin S
PaperOptimization of the solid-phase synthesis of [18F] radiolabeled peptides for positron emission tomography.
White, Jason B, Hausner, Sven H, Carpenter, Richard D, Sutcliffe, Julie L · 2012 · Applied radiation and isotopes : including data, instrumentation and methods for use in agriculture, industry and medicine · DOI
Full title: Optimization of the solid-phase synthesis of [18F] radiolabeled peptides for positron emission tomography.
Authors: White, Jason B, Hausner, Sven H, Carpenter, Richard D, Sutcliffe, Julie L
Year: 2012
Venue: Applied radiation and isotopes : including data, instrumentation and methods for use in agriculture, industry and medicine
PaperFrom the one-bead-one-compound concept to one-bead-one-reactor.
Marani, Mariela M, Paradís-Bas, Marta, Tulla-Puche, Judit, Côté, Simón, Camperi, Silvia A, Cascone, Osvaldo, Albericio, Fernando · 2007 · Journal of combinatorial chemistry · DOI
Full title: From the one-bead-one-compound concept to one-bead-one-reactor.
Authors: Marani, Mariela M, Paradís-Bas, Marta, Tulla-Puche, Judit, Côté, Simón, Camperi, Silvia A, Cascone, Osvaldo, Albericio, Fernando
PaperRegeneration of aged DMF for use in solid-phase peptide synthesis.
Magtaan, Jordan Kevin, Devocelle, Marc, Kelleher, Fintan · 2019 · Journal of peptide science : an official publication of the European Peptide Society · DOI
Full title: Regeneration of aged DMF for use in solid-phase peptide synthesis.
Authors: Magtaan, Jordan Kevin, Devocelle, Marc, Kelleher, Fintan
Year: 2019
Venue: Journal of peptide science : an official publication of the European Peptide Society
Paper2-Methoxy-4-methylsulfinylbenzyl: a backbone amide safety-catch protecting group for the synthesis and purification of difficult peptide sequences.
Paradís-Bas, Marta, Tulla-Puche, Judit, Albericio, Fernando · 2014 · Chemistry (Weinheim an der Bergstrasse, Germany) · DOI
Full title: 2-Methoxy-4-methylsulfinylbenzyl: a backbone amide safety-catch protecting group for the synthesis and purification of difficult peptide sequences.
Authors: Paradís-Bas, Marta, Tulla-Puche, Judit, Albericio, Fernando
Year: 2014
Venue: Chemistry (Weinheim an der Bergstrasse, Germany)
PaperChemMatrix(®) for complex peptides and combinatorial chemistry.
García-Ramos, Yésica, Paradís-Bas, Marta, Tulla-Puche, Judit, Albericio, Fernando · 2010 · Journal of peptide science : an official publication of the European Peptide Society · DOI
Full title: ChemMatrix(®) for complex peptides and combinatorial chemistry.
Authors: García-Ramos, Yésica, Paradís-Bas, Marta, Tulla-Puche, Judit, Albericio, Fernando
Year: 2010
Venue: Journal of peptide science : an official publication of the European Peptide Society
PaperHydrogen fluoride catalyzed migration of side chain protecting groups onto Fmoc during solid phase peptide synthesis. Characterization by CF-FAB analysis of carboxypeptidase digestions and NMR spectroscopy.
Grode, S H, Strother, D S, Runge, T A, Dobrowolski, P J · 1992 · International journal of peptide and protein research · DOI
Full title: Hydrogen fluoride catalyzed migration of side chain protecting groups onto Fmoc during solid phase peptide synthesis. Characterization by CF-FAB analysis of carboxypeptidase digestions and NMR spectroscopy.
Authors: Grode, S H, Strother, D S, Runge, T A, Dobrowolski, P J
Year: 1992
Venue: International journal of peptide and protein research
PaperSolid phase peptide synthesis of human endothelin precursor peptides using two-step hard acid deprotection/cleavage methods.
Nomizu, M, Inagaki, Y, Iwamatsu, A, Kashiwabara, T, Ohta, H, Morita, A, Nishikori, K, Otaka, A, Fujii, N, Roller, P P · 1991 · International journal of peptide and protein research · DOI
Full title: Solid phase peptide synthesis of human endothelin precursor peptides using two-step hard acid deprotection/cleavage methods.
Authors: Nomizu, M, Inagaki, Y, Iwamatsu, A, Kashiwabara, T, Ohta, H, Morita, A, Nishikori, K, Otaka, A, Fujii, N, Roller, P P
Year: 1991
Venue: International journal of peptide and protein research
PaperAutomated Fmoc-based solid-phase synthesis of peptide thioesters with self-purification effect and application in the construction of immobilized SH3 domains.
Mende, Franziska, Beisswenger, Michael, Seitz, Oliver · 2010 · Journal of the American Chemical Society · DOI
Full title: Automated Fmoc-based solid-phase synthesis of peptide thioesters with self-purification effect and application in the construction of immobilized SH3 domains.
Authors: Mende, Franziska, Beisswenger, Michael, Seitz, Oliver
PaperDeprotection of the S-trimethylacetamidomethyl (Tacm) group using silver tetrafluoroborate: application to the synthesis of porcine brain natriuretic peptide-32 (pBNP-32).
Yoshida, M, Tatsumi, T, Fujiwara, Y, Iinuma, S, Kimura, T, Akaji, K, Kiso, Y · 1990 · Chemical & pharmaceutical bulletin · DOI
Full title: Deprotection of the S-trimethylacetamidomethyl (Tacm) group using silver tetrafluoroborate: application to the synthesis of porcine brain natriuretic peptide-32 (pBNP-32).
Authors: Yoshida, M, Tatsumi, T, Fujiwara, Y, Iinuma, S, Kimura, T, Akaji, K, Kiso, Y
PaperSynthesis, 18F-labelling and radiopharmacological characterisation of the C-terminal 30mer of Clostridium perfringens enterotoxin as a potential claudin-targeting peptide.
Full title: Synthesis, 18F-labelling and radiopharmacological characterisation of the C-terminal 30mer of Clostridium perfringens enterotoxin as a potential claudin-targeting peptide.
PaperImproved Fmoc-based solid-phase synthesis of homologous peptide fragments of human and mouse prion proteins.
Grillo-Bosch, Dolors, Rabanal, Francesc, Giralt, Ernest · 2011 · Journal of peptide science : an official publication of the European Peptide Society · DOI
Full title: Improved Fmoc-based solid-phase synthesis of homologous peptide fragments of human and mouse prion proteins.
Authors: Grillo-Bosch, Dolors, Rabanal, Francesc, Giralt, Ernest
Year: 2011
Venue: Journal of peptide science : an official publication of the European Peptide Society
PaperSolid-Phase Synthesis of Difficult Purine-Rich PNAs through Selective Hmb Incorporation: Application to the Total Synthesis of Cell Penetrating Peptide-PNAs.
Tailhades, Julien, Takizawa, Hotake, Gait, Michael J, Wellings, Don A, Wade, John D, Aoki, Yoshitsugu, Shabanpoor, Fazel · 2017 · Frontiers in chemistry · DOI
Full title: Solid-Phase Synthesis of Difficult Purine-Rich PNAs through Selective Hmb Incorporation: Application to the Total Synthesis of Cell Penetrating Peptide-PNAs.
Authors: Tailhades, Julien, Takizawa, Hotake, Gait, Michael J, Wellings, Don A, Wade, John D, Aoki, Yoshitsugu, Shabanpoor, Fazel
PaperSynthesis of Abeta[1-42] and its derivatives with improved efficiency.
Zarándi, Márta, Soós, Katalin, Fülöp, Lívia, Bozsó, Zsolt, Datki, Zsolt, Tóth, Gábor K, Penke, Botond · 2007 · Journal of peptide science : an official publication of the European Peptide Society · DOI
Full title: Synthesis of Abeta[1-42] and its derivatives with improved efficiency.
PaperGreen Solid-Phase Peptide Synthesis 2. 2-Methyltetrahydrofuran and Ethyl Acetate for Solid-Phase Peptide Synthesis under Green Conditions
Jad, Yahya E., Acosta, Gerardo, Govender, Thavendran, Kruger, Hendrik G., El‐Faham, Ayman, Torre, Beatriz G. de la, Alberício, Fernando · 2016 · ACS Sustainable Chemistry & Engineering · DOI
Full title: Green Solid-Phase Peptide Synthesis 2. 2-Methyltetrahydrofuran and Ethyl Acetate for Solid-Phase Peptide Synthesis under Green Conditions
Authors: Jad, Yahya E., Acosta, Gerardo, Govender, Thavendran, Kruger, Hendrik G., El‐Faham, Ayman, Torre, Beatriz G. de la, Alberício, Fernando
PaperProblem of aspartimide formation in Fmoc-based solid-phase peptide synthesis using Dmab group to protect side chain of aspartic acid.
Ruczyński, Jarosław, Lewandowska, Brygida, Mucha, Piotr, Rekowski, Piotr · 2008 · Journal of peptide science : an official publication of the European Peptide Society · DOI
Full title: Problem of aspartimide formation in Fmoc-based solid-phase peptide synthesis using Dmab group to protect side chain of aspartic acid.
Authors: Ruczyński, Jarosław, Lewandowska, Brygida, Mucha, Piotr, Rekowski, Piotr
Year: 2008
Venue: Journal of peptide science : an official publication of the European Peptide Society
PaperHighly selective bradykinin agonists and antagonists with replacement of proline residues by N-methyl-D- and L-phenylalanine.
Reissmann, S, Schwuchow, C, Seyfarth, L, Pineda De Castro, L F, Liebmann, C, Paegelow, I, Werner, H, Stewart, J M · 1996 · Journal of medicinal chemistry · DOI
Full title: Highly selective bradykinin agonists and antagonists with replacement of proline residues by N-methyl-D- and L-phenylalanine.
Authors: Reissmann, S, Schwuchow, C, Seyfarth, L, Pineda De Castro, L F, Liebmann, C, Paegelow, I, Werner, H, Stewart, J M
PaperSynthesis, conformational studies and biological activity of N(alpha)-mono-biotinylated rat relaxin.
Mathieu, M N, Wade, J D, Catimel, B, Bond, C P, Nice, E C, Summers, R J, Otvos, L, Tregear, G W · 2001 · The journal of peptide research : official journal of the American Peptide Society · DOI
Full title: Synthesis, conformational studies and biological activity of N(alpha)-mono-biotinylated rat relaxin.
Authors: Mathieu, M N, Wade, J D, Catimel, B, Bond, C P, Nice, E C, Summers, R J, Otvos, L, Tregear, G W
Year: 2001
Venue: The journal of peptide research : official journal of the American Peptide Society
PaperSynthesis and evaluation of 2-(2-fluoro-4-hydroxymethyl-5-methoxy-phenoxy)acetic acid as a linker in solid-phase synthesis monitored by gel-phase (19)F NMR spectroscopy.
Wallner, Fredrik K, Spjut, Sara, Boström, Dan, Elofsson, Mikael · 2007 · Organic & biomolecular chemistry · DOI
Full title: Synthesis and evaluation of 2-(2-fluoro-4-hydroxymethyl-5-methoxy-phenoxy)acetic acid as a linker in solid-phase synthesis monitored by gel-phase (19)F NMR spectroscopy.
Authors: Wallner, Fredrik K, Spjut, Sara, Boström, Dan, Elofsson, Mikael
PaperSolid-phase precipitation and extraction, a new separation process applied to the isolation of synthetic peptides.
Bonner, A G, Udell, L M, Creasey, W A, Duly, S R, Laursen, R A · 2001 · The journal of peptide research : official journal of the American Peptide Society · DOI
Full title: Solid-phase precipitation and extraction, a new separation process applied to the isolation of synthetic peptides.
Authors: Bonner, A G, Udell, L M, Creasey, W A, Duly, S R, Laursen, R A
Year: 2001
Venue: The journal of peptide research : official journal of the American Peptide Society
PaperAn efficient gel-phase synthesis of peptides on a high capacity flexible crosslinked polystyrene support: comparison with Merrifield resin.
Krishna Kumar, M, Rajasekharan Pillai, V N, Mathew, Beena · 2002 · Journal of peptide science : an official publication of the European Peptide Society · DOI
Full title: An efficient gel-phase synthesis of peptides on a high capacity flexible crosslinked polystyrene support: comparison with Merrifield resin.
Authors: Krishna Kumar, M, Rajasekharan Pillai, V N, Mathew, Beena
Year: 2002
Venue: Journal of peptide science : an official publication of the European Peptide Society
PaperPeptide vaccine candidates against classical swine fever virus: T cell and neutralizing antibody responses of dendrimers displaying E2 and NS2-3 epitopes.
Monsó, Marta, Tarradas, Joan, de la Torre, Beatriz G, Sobrino, Francisco, Ganges, Llilianne, Andreu, David · 2011 · Journal of peptide science : an official publication of the European Peptide Society · DOI
Full title: Peptide vaccine candidates against classical swine fever virus: T cell and neutralizing antibody responses of dendrimers displaying E2 and NS2-3 epitopes.
Authors: Monsó, Marta, Tarradas, Joan, de la Torre, Beatriz G, Sobrino, Francisco, Ganges, Llilianne, Andreu, David
Year: 2011
Venue: Journal of peptide science : an official publication of the European Peptide Society
PaperInvestigating resins for solid phase organic synthesis: the relationship between swelling and microenvironment as probed by EPR and fluorescence spectroscopy.
Vaino, A R, Goodin, D B, Janda, K D · 2000 · Journal of combinatorial chemistry · DOI
Full title: Investigating resins for solid phase organic synthesis: the relationship between swelling and microenvironment as probed by EPR and fluorescence spectroscopy.
PaperSoft shell resins for solid-phase peptide synthesis.
Lee, Tae-Kyung, Choi, Jeong-Hyun, Ryoo, Sun-Jong, Lee, Yoon-Sik · 2007 · Journal of peptide science : an official publication of the European Peptide Society · DOI
Full title: Soft shell resins for solid-phase peptide synthesis.
PaperA convenient incorporation of conformationally constrained 5,5-dimethylproline into the ribonuclease A 89-124 sequence by condensation of synthetic peptide fragments.
Cerovský, V, Welker, E, Scheraga, H A · 2003 · The journal of peptide research : official journal of the American Peptide Society · DOI
Full title: A convenient incorporation of conformationally constrained 5,5-dimethylproline into the ribonuclease A 89-124 sequence by condensation of synthetic peptide fragments.
Authors: Cerovský, V, Welker, E, Scheraga, H A
Year: 2003
Venue: The journal of peptide research : official journal of the American Peptide Society
PaperPressure monitoring of continuous-flow solid-phase peptide synthesis.
Baru, M B, Mustaeva, L G, Vagenina, I V, Gorbunova, E Y, Cherskii, V V · 2001 · The journal of peptide research : official journal of the American Peptide Society · DOI
Full title: Pressure monitoring of continuous-flow solid-phase peptide synthesis.
Authors: Baru, M B, Mustaeva, L G, Vagenina, I V, Gorbunova, E Y, Cherskii, V V
Year: 2001
Venue: The journal of peptide research : official journal of the American Peptide Society
PaperUltrasonic-Assisted Solid-Phase Peptide Synthesis of DOTA-TATE and DOTA-linker-TATE Derivatives as a Simple and Low-Cost Method for the Facile Synthesis of Chelator-Peptide Conjugates.
Raheem, Shvan J, Schmidt, Benjamin W, Solomon, Viswas Raja, Salih, Akam K, Price, Eric W · 2021 · Bioconjugate chemistry · DOI
Full title: Ultrasonic-Assisted Solid-Phase Peptide Synthesis of DOTA-TATE and DOTA-linker-TATE Derivatives as a Simple and Low-Cost Method for the Facile Synthesis of Chelator-Peptide Conjugates.
Authors: Raheem, Shvan J, Schmidt, Benjamin W, Solomon, Viswas Raja, Salih, Akam K, Price, Eric W
PaperEvaluation of COMU as a coupling reagent for in situ neutralization Boc solid phase peptide synthesis.
Hjørringgaard, Claudia U, Brust, Andreas, Alewood, Paul F · 2012 · Journal of peptide science : an official publication of the European Peptide Society · DOI
Full title: Evaluation of COMU as a coupling reagent for in situ neutralization Boc solid phase peptide synthesis.
Authors: Hjørringgaard, Claudia U, Brust, Andreas, Alewood, Paul F
Year: 2012
Venue: Journal of peptide science : an official publication of the European Peptide Society
PaperApplication of N,N-dimethylformamide dineopentyl acetal for efficient anchoring of N alpha-9-fluorenylmethyloxycarbonylamino acids as p-alkoxybenzyl esters in solid-phase peptide synthesis.
Albericio, F, Barany, G · 1984 · International journal of peptide and protein research · DOI
Full title: Application of N,N-dimethylformamide dineopentyl acetal for efficient anchoring of N alpha-9-fluorenylmethyloxycarbonylamino acids as p-alkoxybenzyl esters in solid-phase peptide synthesis.
Authors: Albericio, F, Barany, G
Year: 1984
Venue: International journal of peptide and protein research
ThesisComparative investigation of the cleavage step in the synthesis of model peptide resins: Implications for N-alpha-9-fluorenylmethyloxycarbonyl-solid phase peptide synthesis
Jubilut, Guita Nicolaewsky; Cilli, Eduardo Maffud [UNESP]; Crusca, Edson et al. · 2014 · Theses · DOI
Full title: Comparative investigation of the cleavage step in the synthesis of model peptide resins: Implications for N-alpha-9-fluorenylmethyloxycarbonyl-solid phase peptide synthesis
ThesisSuccessful synthesis of a glial-specific blood-brain barrier shuttle peptide following a fragment condensation approach on a solid-phase resin
Al Musaimi, Othman; Morse, Sophie V; Lombardi, Lucia et al. · 2022 · Theses · DOI
Full title: Successful synthesis of a glial-specific blood-brain barrier shuttle peptide following a fragment condensation approach on a solid-phase resin
Authors: Al Musaimi, Othman; Morse, Sophie V; Lombardi, Lucia; Serban, Simona; Basso, Alessandra; Williams, Daryl R
Full title: Development of a tert-butyl thiol linker for the synthesis of peptide thioesters and thioacids for application in chemical ligation methods
ThesisSynthesis of peptides via cobalt (III) chelates of amino acid methyl esters : a thesis presented in partial fulfilment of the requirements for the degree of Master of Science in Chemistry at Massey University
Full title: Synthesis of peptides via cobalt (III) chelates of amino acid methyl esters : a thesis presented in partial fulfilment of the requirements for the degree of Master of Science in Chemistry at Massey University
Thesis'Dialyzable' Carbosilane Dendrimers as Soluble Supports in Organic Synthesis: Proof of principle, application and diafiltration performance
Full title: 'Dialyzable' Carbosilane Dendrimers as Soluble Supports in Organic Synthesis: Proof of principle, application and diafiltration performance
ThesisBypassing osmotic shock dilemma in a polystyrene resin using the green solvent cyclopentyl methyl Ether (CPME): a morphological perspective
Al Musaimi, Othman; El-Faham, Ayman; Almarhoon, Zainab et al. · 2022 · Theses · DOI
Full title: Bypassing osmotic shock dilemma in a polystyrene resin using the green solvent cyclopentyl methyl Ether (CPME): a morphological perspective
Authors: Al Musaimi, Othman; El-Faham, Ayman; Almarhoon, Zainab; Basso, Alessandra; de la Torre, Beatriz G; Albericio, Fernando
ThesisSynthesis of proteins by automated flow chemistry
Hartrampf, Nina; Saebi, Azin; Poskus, M. et al. · 2020 · Theses · DOI
Full title: Synthesis of proteins by automated flow chemistry
Authors: Hartrampf, Nina; Saebi, Azin; Poskus, M.; Gates, Zachary P; Callahan, A. J.; Cowfer, A. E.; Hanna, S.; Antilla, S.; Schissel, Carly K.; Quartararo, Anthony James; Ye, Xiyun; Mijalis, Alexander James; Simon, M. D.; Loas, Andrei Ioan; Liu, S.; Jessen, C.; Nielsen, T. E.; Pentelute, Bradley L.
ThesisSolid phase peptide synthesis on a beaded cellulose support : a thesis presented in partial fulfilment of the requirements for the degree of Doctor of Philosophy in Chemistry at Massey University
Englebretsen, Darren Ross; Englebretsen, Darren Ross · 2011 · Theses · DOI
Full title: Solid phase peptide synthesis on a beaded cellulose support : a thesis presented in partial fulfilment of the requirements for the degree of Doctor of Philosophy in Chemistry at Massey University
Authors: Englebretsen, Darren Ross; Englebretsen, Darren Ross
ThesisCorrelation between the mobility of spin-labeled peptide chains and resin solvation: An approach to optimize the synthesis of aggregating sequences
Cilli, Eduardo Maffud [UNESP]; Marchetto, Reinaldo [UNESP]; Schreier, S. et al. · 2014 · Theses · DOI
Full title: Correlation between the mobility of spin-labeled peptide chains and resin solvation: An approach to optimize the synthesis of aggregating sequences
Authors: Cilli, Eduardo Maffud [UNESP]; Marchetto, Reinaldo [UNESP]; Schreier, S.; Nakaie, C. R.
ThesisThe Optimization and Use of One-Bead One-Compound Technology to Develop Novel Protein Binders and Fluorescent Probes to Monitor Protein Interactions
Full title: The Optimization and Use of One-Bead One-Compound Technology to Develop Novel Protein Binders and Fluorescent Probes to Monitor Protein Interactions
Full title: Solvólise da ligação peptidil-resina mediada por íons metálicos divalentes: método alternativo de obter peptídeos modificados no C-terninal
Full title: Convergent Hybrid-Phase Ligation Synthetic Strategy Combined with Direct Refolding Method to Improve Synthetic Yield of Centromeric Protein A
ThesisGreening the solid-phase peptide synthesis process. 2-MeTHF for the incorporation of the first amino acid and precipitation of peptides after global deprotection
Al Musaimi, Othman; Jad, Yahya E; Kumar, Ashish et al. · 2021 · Theses · DOI
Full title: Greening the solid-phase peptide synthesis process. 2-MeTHF for the incorporation of the first amino acid and precipitation of peptides after global deprotection
Authors: Al Musaimi, Othman; Jad, Yahya E; Kumar, Ashish; El-Faham, Ayman; Collins, Jonathan M; Basso, Alessandra; de la Torre, Beatriz G; Albericio, Fernando
ThesisStudies towards the chemical synthesis of the 18 kDa antigenic protein from Mycobacterium leprae : a thesis presented in partial fulfilment of the requirements for the degree of Ph. D. in Chemistry at Massey University
Full title: Studies towards the chemical synthesis of the 18 kDa antigenic protein from Mycobacterium leprae : a thesis presented in partial fulfilment of the requirements for the degree of Ph. D. in Chemistry at Massey University
ThesisSolid-phase synthesis of difficult purine-rich PNAs through selective hmb incorporation: Application to the total synthesis of cell penetrating peptide-PNAs
Tailhades, J; Takizawa, H; Gait, MJ et al. · 2020 · Theses · DOI
Full title: Solid-phase synthesis of difficult purine-rich PNAs through selective hmb incorporation: Application to the total synthesis of cell penetrating peptide-PNAs
Authors: Tailhades, J; Takizawa, H; Gait, MJ; Wellings, DA; Wade, JD; Aoki, Y; Shabanpoor, F
ThesisAn approach to the semisynthesis of acyl carrier protein : a thesis presented in partial fulfilment of the requirements for the degree of Doctor of Philosophy in Chemistry at Massey University
Full title: An approach to the semisynthesis of acyl carrier protein : a thesis presented in partial fulfilment of the requirements for the degree of Doctor of Philosophy in Chemistry at Massey University