PaperScalable and Sustainable DMF-Free Solid-Phase Synthesis of Liraglutide by 1-Tert-Butyl-3-Ethylcarbodiimide-Mediated Couplings and Catch-and-Release Acylation and Purification Strategies
Pacini, Lorenzo, Muthyala, Manoj Kumar, Zitterbart, Robert, Marder, Oleg, Rovero, Paolo, Papini, Anna Maria · 2025 · International Journal of Peptide Research and Therapeutics · DOI
Full title: Scalable and Sustainable DMF-Free Solid-Phase Synthesis of Liraglutide by 1-Tert-Butyl-3-Ethylcarbodiimide-Mediated Couplings and Catch-and-Release Acylation and Purification Strategies
Authors: Pacini, Lorenzo, Muthyala, Manoj Kumar, Zitterbart, Robert, Marder, Oleg, Rovero, Paolo, Papini, Anna Maria
Year: 2025
Venue: International Journal of Peptide Research and Therapeutics
PaperStereoselective synthesis of Gly-Gly-type (E)-methylalkene and (Z)-chloroalkene dipeptide isosteres and their application to 14-mer RGG peptidomimetics.
Full title: Stereoselective synthesis of Gly-Gly-type (E)-methylalkene and (Z)-chloroalkene dipeptide isosteres and their application to 14-mer RGG peptidomimetics.
PaperSolid-Phase Peptide Synthesis Using a Four-Dimensional (Safety-Catch) Protecting Group Scheme.
Noki, Sikabwe, Brasil, Edikarlos, Zhang, Haixiang, Bruckdorfer, Thomas, de la Torre, Beatriz G, Albericio, Fernando · 2022 · The Journal of organic chemistry · DOI
Full title: Solid-Phase Peptide Synthesis Using a Four-Dimensional (Safety-Catch) Protecting Group Scheme.
Authors: Noki, Sikabwe, Brasil, Edikarlos, Zhang, Haixiang, Bruckdorfer, Thomas, de la Torre, Beatriz G, Albericio, Fernando
PaperPerfluorophenyl Derivatives as Unsymmetrical Linkers for Solid Phase Conjugation.
Alapour, Saba, Sharma, Anamika, de la Torre, Beatriz G, Ramjugernath, Deresh, Koorbanally, Neil A, Albericio, Fernando · 2018 · Frontiers in chemistry · DOI
Full title: Perfluorophenyl Derivatives as Unsymmetrical Linkers for Solid Phase Conjugation.
Authors: Alapour, Saba, Sharma, Anamika, de la Torre, Beatriz G, Ramjugernath, Deresh, Koorbanally, Neil A, Albericio, Fernando
PaperSolid Phase Synthesis of an Insect Pyrokinin Analog Incorporating an Imidazoline Ring as Isosteric Replacement of a <em>trans</em> Peptide Bond
Kaczmarek, Krzysztof; Pacholczyk‐Sienicka, Barbara; Albrecht, Łukasz et al. · 2021 · Molecules · DOI
Full title: Solid Phase Synthesis of an Insect Pyrokinin Analog Incorporating an Imidazoline Ring as Isosteric Replacement of a <em>trans</em> Peptide Bond
Authors: Kaczmarek, Krzysztof; Pacholczyk‐Sienicka, Barbara; Albrecht, Łukasz; Zabrocki, Janusz; Nachman, Ronald J.
PaperDevelopment of synthetic strategies towards libraries of heterocyclic and bicyclic inhibitors of Cdc25A & development of solid phase synthesis of cyclic peptides
Luo, Hao · 2015 · Institutional Repository of Leibniz Universität Hannover (Leibniz Universität Hannover) · DOI
Full title: Development of synthetic strategies towards libraries of heterocyclic and bicyclic inhibitors of Cdc25A & development of solid phase synthesis of cyclic peptides
Authors: Luo, Hao
Year: 2015
Venue: Institutional Repository of Leibniz Universität Hannover (Leibniz Universität Hannover)
PaperSelf-Assembly of a Novel Pentapeptide into Hydrogelated Dendritic Architecture: Synthesis, Properties, Molecular Docking and Prospective Applications
Jitaru, Stefania-Claudia; Enache, Andra-Cristina; Cojocaru, Corneliu et al. · 2024 · Gels · DOI
Full title: Self-Assembly of a Novel Pentapeptide into Hydrogelated Dendritic Architecture: Synthesis, Properties, Molecular Docking and Prospective Applications
Authors: Jitaru, Stefania-Claudia; Enache, Andra-Cristina; Cojocaru, Corneliu; Drochioiu, Gabi; Petre, Brîndușa Alina; Grădinaru, Vasile Robert
PaperCover Feature: Upscaled Synthesis of α‐ and β‐Peptides in a Continuous‐Flow Reactor Using Propylene Carbonate as an Eco‐Friendly Solvent (Chem. Methods 8/2025)
Varró, Nikolett, Huszka, Beáta Mándityné, Erdei, Eszter, Mándoki, András, Mándity, István M. · 2025 · Chemistry - Methods · DOI
Full title: Cover Feature: Upscaled Synthesis of α‐ and β‐Peptides in a Continuous‐Flow Reactor Using Propylene Carbonate as an Eco‐Friendly Solvent (Chem. Methods 8/2025)
Authors: Varró, Nikolett, Huszka, Beáta Mándityné, Erdei, Eszter, Mándoki, András, Mándity, István M.
PaperAssessing the correlation of microscopy-based and volumetry-based measurements for resin swelling in a range of potential greener solvents for SPPS.
Magtaan, Jordan Kevin; Devocelle, Marc; Kelleher, Fintan · 2020 · Journal of peptide science : an official publication of the European Peptide Society · DOI
Full title: Assessing the correlation of microscopy-based and volumetry-based measurements for resin swelling in a range of potential greener solvents for SPPS.
Authors: Magtaan, Jordan Kevin; Devocelle, Marc; Kelleher, Fintan
Year: 2020
Venue: Journal of peptide science : an official publication of the European Peptide Society
PaperN-Butylpyrrolidinone is an equally good solvent as N,N-dimethylformamide for microwave assisted solid phase peptide synthesis.
Öhlander, Andrea; Lüdtke, Carsten; Sahakjan, Artur et al. · 2024 · Journal of peptide science : an official publication of the European Peptide Society · DOI
Full title: N-Butylpyrrolidinone is an equally good solvent as N,N-dimethylformamide for microwave assisted solid phase peptide synthesis.
Authors: Öhlander, Andrea; Lüdtke, Carsten; Sahakjan, Artur; Johnsson, Richard E
Year: 2024
Venue: Journal of peptide science : an official publication of the European Peptide Society
PaperOptimization of peptide synthesis time and sustainability using novel eco-friendly binary solvent systems with induction heating on an automated peptide synthesizer.
Pacini, Lorenzo; Muthyala, Manoj; Aguiar, Luisa et al. · 2024 · Journal of peptide science : an official publication of the European Peptide Society · DOI
Full title: Optimization of peptide synthesis time and sustainability using novel eco-friendly binary solvent systems with induction heating on an automated peptide synthesizer.
Authors: Pacini, Lorenzo; Muthyala, Manoj; Aguiar, Luisa; Zitterbart, Robert; Rovero, Paolo; Papini, Anna Maria
Year: 2024
Venue: Journal of peptide science : an official publication of the European Peptide Society
Paper2-Methyltetrahydrofuran and cyclopentyl methyl ether for green solid-phase peptide synthesis.
Jad, Yahya E, Acosta, Gerardo A, Khattab, Sherine N, de la Torre, Beatriz G, Govender, Thavendran, Kruger, Hendrik G, El-Faham, Ayman, Albericio, Fernando · 2016 · Amino acids · DOI
Full title: 2-Methyltetrahydrofuran and cyclopentyl methyl ether for green solid-phase peptide synthesis.
Authors: Jad, Yahya E, Acosta, Gerardo A, Khattab, Sherine N, de la Torre, Beatriz G, Govender, Thavendran, Kruger, Hendrik G, El-Faham, Ayman, Albericio, Fernando
PaperEfficient oxidation of N-protected tryptophan and tryptophanyl-dipeptides by in situ generated dimethyldioxirane provides hexahydropyrroloindoline-containing synthons suitable for peptide synthesis and subsequent tryptathionylation.
Blanc, Antoine, Xia, Fan, Todorovic, Mihajlo, Perrin, David M · 2017 · Amino acids · DOI
Full title: Efficient oxidation of N-protected tryptophan and tryptophanyl-dipeptides by in situ generated dimethyldioxirane provides hexahydropyrroloindoline-containing synthons suitable for peptide synthesis and subsequent tryptathionylation.
Authors: Blanc, Antoine, Xia, Fan, Todorovic, Mihajlo, Perrin, David M
PaperEnvironmentally Friendly SPPS II: Scope of Green Fmoc Removal Protocol Using NaOH and Its Application for Synthesis of Commercial Drug Triptorelin.
Přibylka, Adam; Krchňák, Viktor; Schütznerová, Eva · 2020 · The Journal of organic chemistry · DOI
Full title: Environmentally Friendly SPPS II: Scope of Green Fmoc Removal Protocol Using NaOH and Its Application for Synthesis of Commercial Drug Triptorelin.
Authors: Přibylka, Adam; Krchňák, Viktor; Schütznerová, Eva
PaperCombining Real-Time Monitoring Using Raman Spectroscopy, Rotating-Bed Reactors, and Green Solvents to Improve Sustainability in Solid-Phase Peptide Synthesis
Full title: Combining Real-Time Monitoring Using Raman Spectroscopy, Rotating-Bed Reactors, and Green Solvents to Improve Sustainability in Solid-Phase Peptide Synthesis
PaperBulk Mixing in a Milligram-Scale Solid Phase Batch Reactor
Pinzón-López, Sebastián, Ebert, Dominik, Reuber, Emelie E., Kraume, Matthias, Seeberger, Peter H., Danglad‐Flores, José · 2025 · Organic Process Research & Development · DOI
Full title: Bulk Mixing in a Milligram-Scale Solid Phase Batch Reactor
Authors: Pinzón-López, Sebastián, Ebert, Dominik, Reuber, Emelie E., Kraume, Matthias, Seeberger, Peter H., Danglad‐Flores, José
PaperOptimized SPPS Process for Octreotide: Using Green Solvent GVL to Reduce Hazardous DMF and Ether Consumption
KULKARNI, C. L., Dhote, Mohan, Mathur, Abhishek, Pandit, Ravindra, Dudhade, Rahul, Suryawanshi, Yogeshwar, Parameswaran, Sreejith · 2025 · Organic Process Research & Development · DOI
Full title: Optimized SPPS Process for Octreotide: Using Green Solvent GVL to Reduce Hazardous DMF and Ether Consumption
PaperGreen Solid-Phase Peptide Synthesis 2. 2-Methyltetrahydrofuran and Ethyl Acetate for Solid-Phase Peptide Synthesis under Green Conditions
Jad, Yahya E., Acosta, Gerardo, Govender, Thavendran, Kruger, Hendrik G., El‐Faham, Ayman, Torre, Beatriz G. de la, Alberício, Fernando · 2016 · ACS Sustainable Chemistry & Engineering · DOI
Full title: Green Solid-Phase Peptide Synthesis 2. 2-Methyltetrahydrofuran and Ethyl Acetate for Solid-Phase Peptide Synthesis under Green Conditions
Authors: Jad, Yahya E., Acosta, Gerardo, Govender, Thavendran, Kruger, Hendrik G., El‐Faham, Ayman, Torre, Beatriz G. de la, Alberício, Fernando
PaperThe application of anisole in greener solid-phase peptide synthesis protocols – Compatibility with green bases in Fmoc removal and new green binary mixture for coupling
Přibylka, Adam, Pastorek, Milan, Grepl, Martin, Schütznerová, Eva · 2021 · Tetrahedron · DOI
Full title: The application of anisole in greener solid-phase peptide synthesis protocols – Compatibility with green bases in Fmoc removal and new green binary mixture for coupling
Authors: Přibylka, Adam, Pastorek, Milan, Grepl, Martin, Schütznerová, Eva
PaperAdvancing Sustainable Peptide Synthesis by Solvent Quality Control: Understanding and Mitigating Hydroperoxide in 1-Butyl-2-pyrrolidinone (NBP)
Pawlas, Jan, El‐Dine, Tharwat Mohy, Bargen, Katharina von, Bargen, Christoph von, Nilsson, Johan, Ludemann‐Hombourger, Olivier, Rasmussen, Jon H. · 2024 · Organic Process Research & Development · DOI
Full title: Advancing Sustainable Peptide Synthesis by Solvent Quality Control: Understanding and Mitigating Hydroperoxide in 1-Butyl-2-pyrrolidinone (NBP)
Authors: Pawlas, Jan, El‐Dine, Tharwat Mohy, Bargen, Katharina von, Bargen, Christoph von, Nilsson, Johan, Ludemann‐Hombourger, Olivier, Rasmussen, Jon H.
Full title: Green Solvent Mixtures for Solid-Phase Peptide Synthesis: A Dimethylformamide-Free Highly Efficient Synthesis of Pharmaceutical-Grade Peptides
PaperReplacing DMF in solid-phase peptide synthesis: varying the composition of green binary solvent mixtures as a tool to mitigate common side-reactions
S. Jadhav; Vincent Martin; P. H. G. Egelund et al. · 2021 · Green Chemistry · DOI
Full title: Replacing DMF in solid-phase peptide synthesis: varying the composition of green binary solvent mixtures as a tool to mitigate common side-reactions
Authors: S. Jadhav; Vincent Martin; P. H. G. Egelund; Henrik Johansson Castro; Tobias Krüger; Franziska Richner; Sebastian Thordal Le Quement; F. Albericio; Frank Dettner; Carolin Lechner; Ralph Schönleber; D. Pedersen
PaperTriethyl phosphate (TEP) – dimethylsulfoxide (DMSO), as a green solvent mixture for solid-phase peptide synthesis (SPPS)
Sikabwe Noki, Luana Lastella, Simona Serban, Alessandra Basso, Gyorgy Orosz, Beatriz G de la Torre, F. Albericio · 2024 · Green Chemistry Letters and Reviews · DOI
Full title: Triethyl phosphate (TEP) – dimethylsulfoxide (DMSO), as a green solvent mixture for solid-phase peptide synthesis (SPPS)
Authors: Sikabwe Noki, Luana Lastella, Simona Serban, Alessandra Basso, Gyorgy Orosz, Beatriz G de la Torre, F. Albericio
PaperHarnessing polarity and viscosity to identify green binary solvent mixtures as viable alternatives to DMF in solid-phase peptide synthesis
Vincent Martin; S. Jadhav; P. H. G. Egelund et al. · 2021 · Green Chemistry · DOI
Full title: Harnessing polarity and viscosity to identify green binary solvent mixtures as viable alternatives to DMF in solid-phase peptide synthesis
Authors: Vincent Martin; S. Jadhav; P. H. G. Egelund; Raphael Liffert; Henrik Johansson Castro; Tobias Krüger; K. Haselmann; Sebastian Thordal Le Quement; F. Albericio; Frank Dettner; Carolin Lechner; Ralph Schönleber; D. Pedersen
PaperApplication of a new green protocol in solid-phase peptide synthesis: identification of a new green solvent mixture compatible with TBEC/ETT
G. Vivenzio; M. Scala; Giulia Auriemma et al. · 2024 · Green Chemistry Letters and Reviews · DOI
Full title: Application of a new green protocol in solid-phase peptide synthesis: identification of a new green solvent mixture compatible with TBEC/ETT
Authors: G. Vivenzio; M. Scala; Giulia Auriemma; Carla Sardo; P. Campiglia; M. Sala
PaperGreen solvents and Safe Reagents in SPPS taking advantage of induction heating and automation: synthesis and HPLC-free purification of difficult sequences
Pacini, L., Muthyala, Manoj Kumar, Marder, Oleg, Aguiar, Luiz Felipe Soares, Zitterbart, Robert, Rovero, Paolo, Papini, A. M. · 2024 · DOI
Full title: Green solvents and Safe Reagents in SPPS taking advantage of induction heating and automation: synthesis and HPLC-free purification of difficult sequences
Authors: Pacini, L., Muthyala, Manoj Kumar, Marder, Oleg, Aguiar, Luiz Felipe Soares, Zitterbart, Robert, Rovero, Paolo, Papini, A. M.
PaperRapid building block-economic synthesis of long, multi-<i>O</i>-GalNAcylated MUC5AC tandem repeat peptides
Arseniy, Galashov,, Ekaterina, Kazakova,, E., Stieger, Christian, R., Hackenberger, Christian P., Oliver, Seitz, · 2023 · edoc Publication server (Humboldt University of Berlin) · DOI
Full title: Rapid building block-economic synthesis of long, multi-<i>O</i>-GalNAcylated MUC5AC tandem repeat peptides
Authors: Arseniy, Galashov,, Ekaterina, Kazakova,, E., Stieger, Christian, R., Hackenberger, Christian P., Oliver, Seitz,
Year: 2023
Venue: edoc Publication server (Humboldt University of Berlin)
PaperScalable and sustainable DMF-free solid-phase synthesis of liraglutideby 1-tert-butyl-3-ethylcarbodiimide-mediated couplings and catch-and-release acylation and purification strategies
Pacini, Lorenzo, Muthyala, Manoj Kumar, Zitterbart, Robert, Marder, Oleg, Rovero, Paolo, Papini, Anna Maria · 2025 · DOI
Full title: Scalable and sustainable DMF-free solid-phase synthesis of liraglutideby 1-tert-butyl-3-ethylcarbodiimide-mediated couplings and catch-and-release acylation and purification strategies
Authors: Pacini, Lorenzo, Muthyala, Manoj Kumar, Zitterbart, Robert, Marder, Oleg, Rovero, Paolo, Papini, Anna Maria
PaperSilylated Tag-Assisted Peptide Synthesis: Continuous One-Pot Elongation for the Production of Difficult Peptides under Environmentally Friendly Conditions
Full title: Silylated Tag-Assisted Peptide Synthesis: Continuous One-Pot Elongation for the Production of Difficult Peptides under Environmentally Friendly Conditions
PaperDipropyleneglycol Dimethylether, New Green Solvent for Solid-Phase Peptide Synthesis: Further Challenges to Improve Sustainability in the Development of Therapeutic Peptides.
Vivenzio, Giovanni; Scala, Maria Carmina; Marino, Pasquale et al. · 2023 · Pharmaceutics · DOI
Full title: Dipropyleneglycol Dimethylether, New Green Solvent for Solid-Phase Peptide Synthesis: Further Challenges to Improve Sustainability in the Development of Therapeutic Peptides.
Authors: Vivenzio, Giovanni; Scala, Maria Carmina; Marino, Pasquale; Manfra, Michele; Campiglia, Pietro; Sala, Marina
PaperBypassing Osmotic Shock Dilemma in a Polystyrene Resin Using the Green Solvent Cyclopentyl methyl Ether (CPME): A Morphological Perspective.
Al Musaimi, Othman; El-Faham, Ayman; Almarhoon, Zainab et al. · 2019 · Polymers · DOI
Full title: Bypassing Osmotic Shock Dilemma in a Polystyrene Resin Using the Green Solvent Cyclopentyl methyl Ether (CPME): A Morphological Perspective.
Authors: Al Musaimi, Othman; El-Faham, Ayman; Almarhoon, Zainab; Basso, Alessandra; de la Torre, Beatriz G; Albericio, Fernando
PaperDesign and synthesis of novel prodrugs to modulate GABA receptors in cancer
Zhang, Hui · 2017 · Research Output (Edinburgh Napier University)
Full title: Design and synthesis of novel prodrugs to modulate GABA receptors in cancer
Authors: Zhang, Hui
Year: 2017
Venue: Research Output (Edinburgh Napier University)
PaperA Targeted Drug Delivery Strategy for Trypanosomiasis Towards a Diastereoselective Boronate Ester Mediated Intramolecular Diels-Alder Cycloaddition
Gordhan, Heeren M. · 2017 · TigerPrints (Clemson University)
Full title: A Targeted Drug Delivery Strategy for Trypanosomiasis Towards a Diastereoselective Boronate Ester Mediated Intramolecular Diels-Alder Cycloaddition
Authors: Gordhan, Heeren M.
Year: 2017
Venue: TigerPrints (Clemson University)
PaperDevelopment And Applications Of Thioacids In Peptide Chemistry And Exploration Of Methods Toward The Stereochemical Elucidation And Synthesis Of Virgineone
Full title: Development And Applications Of Thioacids In Peptide Chemistry And Exploration Of Methods Toward The Stereochemical Elucidation And Synthesis Of Virgineone
Authors: Sana, Kasinath
Year: 2010
Venue: DigitalCommons - WayneState (Wayne State University)
PaperTowards a Total Chemical Synthesis of Human C-C Motif Chemokine Ligand 2
Lear, Sam · 2013 · Durham e-Theses (Durham University)
Full title: Towards a Total Chemical Synthesis of Human C-C Motif Chemokine Ligand 2
Authors: Lear, Sam
Year: 2013
Venue: Durham e-Theses (Durham University)
PaperOxetane-based peptidomimetics
Beadle, Jonathan D. · 2018 · Warwick Research Archive Portal (University of Warwick)
Full title: Oxetane-based peptidomimetics
Authors: Beadle, Jonathan D.
Year: 2018
Venue: Warwick Research Archive Portal (University of Warwick)
PaperSPPS resins impact the PNA-syntheses' improvement.
Pipkorn, Rüdiger, Rawer, Stephan, Wiessler, Manfred, Waldeck, Waldemar, Koch, Mario, Schrenk, Hans Hermann, Braun, Klaus · 2013 · International journal of medical sciences · DOI
Full title: SPPS resins impact the PNA-syntheses' improvement.
Authors: Pipkorn, Rüdiger, Rawer, Stephan, Wiessler, Manfred, Waldeck, Waldemar, Koch, Mario, Schrenk, Hans Hermann, Braun, Klaus
PaperSynthesis, characterization, and biological activity of poly(arginine)-derived cancer-targeting peptides in HepG2 liver cancer cells.
Joseph, Stesha C; Blackman, Brittany A; Kelly, Megan L et al. · 2014 · Journal of peptide science : an official publication of the European Peptide Society · DOI
Full title: Synthesis, characterization, and biological activity of poly(arginine)-derived cancer-targeting peptides in HepG2 liver cancer cells.
Authors: Joseph, Stesha C; Blackman, Brittany A; Kelly, Megan L; Phillips, Mariana; Beaury, Michael W; Martinez, Ivonne; Parronchi, Christopher J; Bitsaktsis, Constantine; Blake, Allan D; Sabatino, David
Year: 2014
Venue: Journal of peptide science : an official publication of the European Peptide Society
PaperScope and Limitations of Barbituric and Thiobarbituric Amino Acid Derivatives as Protecting Groups for Solid‐Phase Peptide Synthesis: Towards a Green Protecting Group
Ramkisson, Shaveer; Al‐Rasheed, Hessa H.; Dahlous, Kholood A. et al. · 2021 · ChemistrySelect · DOI
Full title: Scope and Limitations of Barbituric and Thiobarbituric Amino Acid Derivatives as Protecting Groups for Solid‐Phase Peptide Synthesis: Towards a Green Protecting Group
Authors: Ramkisson, Shaveer; Al‐Rasheed, Hessa H.; Dahlous, Kholood A.; Torre, Beatriz G. de la; El‐Faham, Ayman; Alberício, Fernando
PaperAmine capture strategy for peptide bond formation by means of quinolinium thioester salts.
Leleu, Stéphane, Penhoat, Maël, Bouet, Alexis, Dupas, Georges, Papamicaël, Cyril, Marsais, Francis, Levacher, Vincent · 2005 · Journal of the American Chemical Society · DOI
Full title: Amine capture strategy for peptide bond formation by means of quinolinium thioester salts.
PaperE-olefin dipeptide isostere incorporation into a polypeptide backbone enables hydrogen bond perturbation: probing the requirements for Alzheimer's amyloidogenesis.
Fu, Yanwen, Bieschke, Jan, Kelly, Jeffery W · 2005 · Journal of the American Chemical Society · DOI
Full title: E-olefin dipeptide isostere incorporation into a polypeptide backbone enables hydrogen bond perturbation: probing the requirements for Alzheimer's amyloidogenesis.
Authors: Fu, Yanwen, Bieschke, Jan, Kelly, Jeffery W
PaperDevelopment of a new method for synthesis of tandem hairpin pyrrole-imidazole polyamide probes targeting human telomeres.
Kawamoto, Yusuke, Bando, Toshikazu, Kamada, Fukumi, Li, Yue, Hashiya, Kaori, Maeshima, Kazuhiro, Sugiyama, Hiroshi · 2013 · Journal of the American Chemical Society · DOI
Full title: Development of a new method for synthesis of tandem hairpin pyrrole-imidazole polyamide probes targeting human telomeres.
PaperA Versatile "Synthesis Tag" (SynTag) for the Chemical Synthesis of Aggregating Peptides and Proteins.
Bürgisser, Héloïse, Williams, Elyse T, Jeandin, Aliénor, Lescure, Robin, Premanand, Adhvitha, Wang, Songlin, Hartrampf, Nina · 2024 · Journal of the American Chemical Society · DOI
Full title: A Versatile "Synthesis Tag" (SynTag) for the Chemical Synthesis of Aggregating Peptides and Proteins.
PaperPeptidotriazoles on solid phase: [1,2,3]-triazoles by regiospecific copper(i)-catalyzed 1,3-dipolar cycloadditions of terminal alkynes to azides.
Tornøe, Christian W, Christensen, Caspar, Meldal, Morten · 2002 · The Journal of organic chemistry · DOI
Full title: Peptidotriazoles on solid phase: [1,2,3]-triazoles by regiospecific copper(i)-catalyzed 1,3-dipolar cycloadditions of terminal alkynes to azides.
Authors: Tornøe, Christian W, Christensen, Caspar, Meldal, Morten
PaperSynthesis of nucleotidylated poliovirus VPg proteins.
van der Heden van Noort, Gerbrand J, Overkleeft, Herman S, van der Marel, Gijsbert A, Filippov, Dmitri V · 2010 · The Journal of organic chemistry · DOI
Full title: Synthesis of nucleotidylated poliovirus VPg proteins.
Authors: van der Heden van Noort, Gerbrand J, Overkleeft, Herman S, van der Marel, Gijsbert A, Filippov, Dmitri V
PaperSynthetic procedure for N-Fmoc amino acyl-N-sulfanylethylaniline linker as crypto-peptide thioester precursor with application to native chemical ligation.
Sakamoto, Ken, Sato, Kohei, Shigenaga, Akira, Tsuji, Kohei, Tsuda, Shugo, Hibino, Hajime, Nishiuchi, Yuji, Otaka, Akira · 2012 · The Journal of organic chemistry · DOI
Full title: Synthetic procedure for N-Fmoc amino acyl-N-sulfanylethylaniline linker as crypto-peptide thioester precursor with application to native chemical ligation.
PaperC-Glycosyl Tyrosines. Synthesis and Incorporation into C-Glycopeptides.
Pearce, Alan J., Ramaya, Sharn, Thorn, Simon N., Bloomberg, Graham B., Walter, Daryl S., Gallagher, Timothy · 1999 · The Journal of organic chemistry · DOI
Full title: C-Glycosyl Tyrosines. Synthesis and Incorporation into C-Glycopeptides.
Authors: Pearce, Alan J., Ramaya, Sharn, Thorn, Simon N., Bloomberg, Graham B., Walter, Daryl S., Gallagher, Timothy
PaperFmoc-based synthesis of disulfide-rich cyclic peptides.
Cheneval, Olivier, Schroeder, Christina I, Durek, Thomas, Walsh, Phillip, Huang, Yen-Hua, Liras, Spiros, Price, David A, Craik, David J · 2014 · The Journal of organic chemistry · DOI
Full title: Fmoc-based synthesis of disulfide-rich cyclic peptides.
Authors: Cheneval, Olivier, Schroeder, Christina I, Durek, Thomas, Walsh, Phillip, Huang, Yen-Hua, Liras, Spiros, Price, David A, Craik, David J
PaperInhibitors of HGFA, Matriptase, and Hepsin Serine Proteases: A Nonkinase Strategy to Block Cell Signaling in Cancer.
Han, Zhenfu, Harris, Peter K W, Jones, Darin E, Chugani, Ryan, Kim, Tommy, Agarwal, Manjula, Shen, Wei, Wildman, Scott A, Janetka, James W · 2014 · ACS medicinal chemistry letters · DOI
Full title: Inhibitors of HGFA, Matriptase, and Hepsin Serine Proteases: A Nonkinase Strategy to Block Cell Signaling in Cancer.
Authors: Han, Zhenfu, Harris, Peter K W, Jones, Darin E, Chugani, Ryan, Kim, Tommy, Agarwal, Manjula, Shen, Wei, Wildman, Scott A, Janetka, James W
PaperIncorporation of pseudoproline derivatives allows the facile synthesis of human IAPP, a highly amyloidogenic and aggregation-prone polypeptide.
Abedini, Andisheh, Raleigh, Daniel P · 2005 · Organic letters · DOI
Full title: Incorporation of pseudoproline derivatives allows the facile synthesis of human IAPP, a highly amyloidogenic and aggregation-prone polypeptide.
PaperEfficient solid-phase synthesis of Vpr from HIV-1 using low quantities of uniformly 13C-, 15N-labeled amino acids for NMR structural studies.
Cornille, F, Wecker, K, Loffet, A, Genet, R, Roques, B · 1999 · The journal of peptide research : official journal of the American Peptide Society · DOI
Full title: Efficient solid-phase synthesis of Vpr from HIV-1 using low quantities of uniformly 13C-, 15N-labeled amino acids for NMR structural studies.
Authors: Cornille, F, Wecker, K, Loffet, A, Genet, R, Roques, B
Year: 1999
Venue: The journal of peptide research : official journal of the American Peptide Society
Venue: Peptide chemistry : proceedings of the ... Symposium on Peptide Chemistry
PaperPeptides as potential virus inhibitors. Synthesis and bioassay of five respiratory syncytial virus peptide analogs with antimeasles activity.
Lobl, T J, Renis, H E, Epand, R M, Maggiora, L L, Wathen, M W · 1988 · International journal of peptide and protein research
Full title: Peptides as potential virus inhibitors. Synthesis and bioassay of five respiratory syncytial virus peptide analogs with antimeasles activity.
Authors: Lobl, T J, Renis, H E, Epand, R M, Maggiora, L L, Wathen, M W
Year: 1988
Venue: International journal of peptide and protein research
PaperPseudo-prolines (psi Pro) for accessing "inaccessible" peptides.
Mutter, M, Nefzi, A, Sato, T, Sun, X, Wahl, F, Wöhr, T · 1995 · Peptide research
Full title: Pseudo-prolines (psi Pro) for accessing "inaccessible" peptides.
Authors: Mutter, M, Nefzi, A, Sato, T, Sun, X, Wahl, F, Wöhr, T
Year: 1995
Venue: Peptide research
Paper[Peptide fragment 66-77 of monocyte chemoattractant protein 1 and its retro-enantio analogue inhibits the migration of cells in vitro and in vivo].
Sidorova, M V, Molokoedov, A S, Az'muko, A A, Aref'eva, T I, Melekhov, M G, Kukhtina, N B, Krasnikova, T L, Bespalova, Zh D, Bushuev, V N · 2006 · Bioorganicheskaia khimiia
Full title: [Peptide fragment 66-77 of monocyte chemoattractant protein 1 and its retro-enantio analogue inhibits the migration of cells in vitro and in vivo].
Authors: Sidorova, M V, Molokoedov, A S, Az'muko, A A, Aref'eva, T I, Melekhov, M G, Kukhtina, N B, Krasnikova, T L, Bespalova, Zh D, Bushuev, V N
Year: 2006
Venue: Bioorganicheskaia khimiia
Paper[Solid phase peptide synthesis: interest in the valorization of molecular substances from animal venoms].
Aidi-Knani, S, Ghodhbane, H, Mourre, Ch, Benhamida, J, Jean-Marc, S, Regaya, I · 2014 · Archives de l'Institut Pasteur de Tunis
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PaperSolid-Phase Synthesis of Antitumor Peptide AP-9
O. Pingkai · 2007 · Chinese Journal of Pharmaceuticals
Full title: Solid-Phase Synthesis of Antitumor Peptide AP-9
Authors: O. Pingkai
Year: 2007
Venue: Chinese Journal of Pharmaceuticals
PaperRapid Screening and Identification of Dominant B Cell Epitopes of UreB Protein by Fluorescence Polarization Assay
Hui-fang Guo, Wen-hong Zhang, Dong-qing Wen, F. Han, Huming Zhang, Jin Luo, Xiaojun Yan · 2006 · PROGRESS IN BIOCHEMISTRY AND BIOPHYSICS
Full title: Rapid Screening and Identification of Dominant B Cell Epitopes of UreB Protein by Fluorescence Polarization Assay
Authors: Hui-fang Guo, Wen-hong Zhang, Dong-qing Wen, F. Han, Huming Zhang, Jin Luo, Xiaojun Yan
Year: 2006
Venue: PROGRESS IN BIOCHEMISTRY AND BIOPHYSICS
PaperSolid phase peptide synthesis on hydrophilic supports. Part II--Studies using Perloza beaded cellulose.
Englebretsen, D R, Harding, D R · 1992 · International journal of peptide and protein research
Full title: Solid phase peptide synthesis on hydrophilic supports. Part II--Studies using Perloza beaded cellulose.
Authors: Englebretsen, D R, Harding, D R
Year: 1992
Venue: International journal of peptide and protein research
PaperSolid-phase synthesis of bovine pancreatic trypsin inhibitor (BPTI) and two analogues. A chemical approach for evaluating the role of disulfide bridges in protein folding and stability.
Ferrer, M, Woodward, C, Barany, G · 1992 · International journal of peptide and protein research
Full title: Solid-phase synthesis of bovine pancreatic trypsin inhibitor (BPTI) and two analogues. A chemical approach for evaluating the role of disulfide bridges in protein folding and stability.
Authors: Ferrer, M, Woodward, C, Barany, G
Year: 1992
Venue: International journal of peptide and protein research
PaperStructure-activity studies with cholecystokinin: stereoisomers containing ortho-, meta- and para-tyrosine sulfate.
Stanfield, C F, Felix, A M, Danho, W · 1990 · Peptide research
Full title: Structure-activity studies with cholecystokinin: stereoisomers containing ortho-, meta- and para-tyrosine sulfate.
Authors: Stanfield, C F, Felix, A M, Danho, W
Year: 1990
Venue: Peptide research
PaperStudies towards Photochemical nanopatterning using a Caged Peptide
Belaid, Amal, Ammar, Amal Abdallah-Ben, Kellam, Barrie, Shakesheff, Kevin M. · 2015
Full title: Studies towards Photochemical nanopatterning using a Caged Peptide
Authors: Belaid, Amal, Ammar, Amal Abdallah-Ben, Kellam, Barrie, Shakesheff, Kevin M.
Year: 2015
PaperSolid-phase synthesis of a peptide-ligand affinity matrix for isolation of chymosin.
Englebretsen, D R, Harding, D R · 1993 · Peptide research
Full title: Solid-phase synthesis of a peptide-ligand affinity matrix for isolation of chymosin.
Authors: Englebretsen, D R, Harding, D R
Year: 1993
Venue: Peptide research
PaperSolid phase synthesis of cetrorelix
Xiang Guang · 2010
Full title: Solid phase synthesis of cetrorelix
Authors: Xiang Guang
Year: 2010
PaperSolid-phase synthesis of bovine pancreatic trypsin inhibitor (BPTI) and two analogues. A chemical approach for evaluating the role of disulfide bridges in protein folding and stability.
Ferrer, Marc, Woodward, Clare, Bárány, George · 1993 · PubMed
Full title: Solid-phase synthesis of bovine pancreatic trypsin inhibitor (BPTI) and two analogues. A chemical approach for evaluating the role of disulfide bridges in protein folding and stability.
Authors: Ferrer, Marc, Woodward, Clare, Bárány, George
Year: 1993
Venue: PubMed
PaperSolid Synthesis and Immunopotentiation of Thymopoietin-5
Full title: Solid Synthesis and Immunopotentiation of Thymopoietin-5
Authors: Zhang, Chunli
Year: 2003
Venue: Zhongguo shengwuzhipinxue zazhi
PaperSporopollenin. A novel, naturally occurring support for solid phase peptide synthesis.
Mackenzie, G, Shaw, G · 1980 · International journal of peptide and protein research
Full title: Sporopollenin. A novel, naturally occurring support for solid phase peptide synthesis.
Authors: Mackenzie, G, Shaw, G
Year: 1980
Venue: International journal of peptide and protein research
PaperStable isolated symmetrical anhydrides of N alpha-9-fluorenylmethyloxycarbonylamino acids in solid-phase peptide synthesis. Methionine-enkephalin synthesis as an example.
Heimer, E P, Chang, C D, Lambros, T, Meienhofer, J · 1981 · International journal of peptide and protein research
Full title: Stable isolated symmetrical anhydrides of N alpha-9-fluorenylmethyloxycarbonylamino acids in solid-phase peptide synthesis. Methionine-enkephalin synthesis as an example.
Authors: Heimer, E P, Chang, C D, Lambros, T, Meienhofer, J
Year: 1981
Venue: International journal of peptide and protein research
PaperSynthesis and folding of the circular cystine knotted cyclotide cycloviolacin O2
Aboye, Teshome Leta, Clark, Richard J., Craik, David J., Göransson, Ulf · 2008 · PubMed Central
Full title: Synthesis and folding of the circular cystine knotted cyclotide cycloviolacin O2
Authors: Aboye, Teshome Leta, Clark, Richard J., Craik, David J., Göransson, Ulf
Year: 2008
Venue: PubMed Central
PaperSynthesis and Purification of Position 4 Analogs of the Opioid Peptide JVA-4001
Hanson, Christina · 2019
Full title: Synthesis and Purification of Position 4 Analogs of the Opioid Peptide JVA-4001
Authors: Hanson, Christina
Year: 2019
PaperSynthesis and structural determination of tetrapeptide EVPK in PEVK segment of Titin
Mei, Dong · 2010 · Acta Academiae Medicinae CPAF
Full title: Synthesis and structural determination of tetrapeptide EVPK in PEVK segment of Titin
Authors: Mei, Dong
Year: 2010
Venue: Acta Academiae Medicinae CPAF
Paper[Synthesis and activities of fragments of inhibin alpha subunit].
Sun, Y, Lu, G S, Wang, D X, Zhang, J H, Cheng, Z P · 1996 · Yao xue xue bao = Acta pharmaceutica Sinica
Full title: [Synthesis and activities of fragments of inhibin alpha subunit].
Authors: Sun, Y, Lu, G S, Wang, D X, Zhang, J H, Cheng, Z P
Year: 1996
Venue: Yao xue xue bao = Acta pharmaceutica Sinica
PaperSurfactant protein B-based microemulsion as transdermal drug carrier for anti-acne agent
Ramli, Suria · 2013 · Queensland's institutional digital repository (The University of Queensland)
Full title: Surfactant protein B-based microemulsion as transdermal drug carrier for anti-acne agent
Authors: Ramli, Suria
Year: 2013
Venue: Queensland's institutional digital repository (The University of Queensland)
PaperSynthesis and Bioactivity Analysis of the Chimera Polypeptide of ω-Ctx MVIIA and HWTX-I
Tang, Hui · 2002 · Journal of Naturnal Science of Hunan Normal University
Full title: Synthesis and Bioactivity Analysis of the Chimera Polypeptide of ω-Ctx MVIIA and HWTX-I
Authors: Tang, Hui
Year: 2002
Venue: Journal of Naturnal Science of Hunan Normal University
PaperSynthesis and Biological Evaluation of Novel TLR2 Agonist-Conjugated Antigenic Peptides for use in Cancer Therapeutics
Full title: Synthesis of the Peptide-Based Phenanthridine-Nucleobase Conjugates and Study of Their Interactions With ds-DNA.
Authors: Dukši, Marko, Baretić, Domagoj, Piantanida, Ivo
Year: 2012
Venue: Acta chimica Slovenica
PaperSynthesis and screening of peptide libraries with free C-termini.
Wang, Yen-Chih, Distefano, Mark D · 2014 · Current topics in peptide & protein research
Full title: Synthesis and screening of peptide libraries with free C-termini.
Authors: Wang, Yen-Chih, Distefano, Mark D
Year: 2014
Venue: Current topics in peptide & protein research
PaperSynthesis and pharmacological characterization of endomorphin-1 analogues
Varamini, Pegah · 2012 · Queensland's institutional digital repository (The University of Queensland)
Full title: Synthesis and pharmacological characterization of endomorphin-1 analogues
Authors: Varamini, Pegah
Year: 2012
Venue: Queensland's institutional digital repository (The University of Queensland)
PaperSynthesis, biological activity and molecular modelling of the 53-54 ketomethylene analogue of HEL(52-61)
Ettouati, Laurent, Casimir, J. Richard, Raynaud, Isabelle, Biémont-Trescol, Marie-Claude, Carrupt, Pierre‐Alain, Gerlier, Denis, Rabourdin‐Combe, Chantal, Testa, Bernard, Paris, Joëlle · 1998 · HAL (Le Centre pour la Communication Scientifique Directe)
Full title: Synthesis, biological activity and molecular modelling of the 53-54 ketomethylene analogue of HEL(52-61)
Venue: HAL (Le Centre pour la Communication Scientifique Directe)
Paper[The automated "SynChrom" system for solid-phase synthesis of peptides and liquid column chromatography. I. Principles of design and structural constituents].
Baru, M B, Cherskiĭ, V V, Danilov, A V, Moshnikov, S A, Mustaeva, L G · 1995 · Bioorganicheskaia khimiia
Full title: [The automated "SynChrom" system for solid-phase synthesis of peptides and liquid column chromatography. I. Principles of design and structural constituents].
Authors: Baru, M B, Cherskiĭ, V V, Danilov, A V, Moshnikov, S A, Mustaeva, L G
Year: 1995
Venue: Bioorganicheskaia khimiia
PaperTotal synthesis of argyrin A and analogues thereof
Chen, Chou-Hsiung · 2013 · Nottingham ePrints (University of Nottingham)
Full title: Total synthesis of argyrin A and analogues thereof
Authors: Chen, Chou-Hsiung
Year: 2013
Venue: Nottingham ePrints (University of Nottingham)
PaperUse of synthetic peptides for the delivery of growth factors for tendon/ligament healing
Crispim, João F., Fernandes, Hugo, Jonkheijm, Pascal, Saris, Daniël B.F. · 2015 · TU/e Research Portal (Eindhoven University of Technology)
Full title: Use of synthetic peptides for the delivery of growth factors for tendon/ligament healing
PaperRapid, sensitive and efficient HPLC assays for HIV-1 proteinase.
Betageri, R, Hopkins, J L, Thibeault, D, Emmanuel, M J, Chow, G C, Skoog, M T, de Dreu, P, Cohen, K A · 1993 · Journal of biochemical and biophysical methods · DOI
Full title: Rapid, sensitive and efficient HPLC assays for HIV-1 proteinase.
Authors: Betageri, R, Hopkins, J L, Thibeault, D, Emmanuel, M J, Chow, G C, Skoog, M T, de Dreu, P, Cohen, K A
Year: 1993
Venue: Journal of biochemical and biophysical methods
PaperRecent advances in solid-phase peptide synthesis and preparation of antibodies to synthetic peptides.
Plaue, S, Muller, S, Briand, J P, Van Regenmortel, M H · 1990 · Biologicals : journal of the International Association of Biological Standardization · DOI
Full title: Recent advances in solid-phase peptide synthesis and preparation of antibodies to synthetic peptides.
Authors: Plaue, S, Muller, S, Briand, J P, Van Regenmortel, M H
Year: 1990
Venue: Biologicals : journal of the International Association of Biological Standardization
PaperSynthesis, biological evaluation and preclinical study of a novel 99mTc-peptide: A targeting probe of amyloid-β plaques as a possible diagnostic agent for Alzheimer's disease.
Full title: Synthesis, biological evaluation and preclinical study of a novel 99mTc-peptide: A targeting probe of amyloid-β plaques as a possible diagnostic agent for Alzheimer's disease.
PaperCost-effective synthesis of a chromogenic substrate for SARS-CoV-2 Mpro and development of a miniaturized high-throughput inhibition assay.
Spinelli, Roque, Humpola, Maria Veronica, Sanchis, Ivan, Siano, Alvaro S · 2025 · Methods in enzymology · DOI
Full title: Cost-effective synthesis of a chromogenic substrate for SARS-CoV-2 Mpro and development of a miniaturized high-throughput inhibition assay.
Authors: Spinelli, Roque, Humpola, Maria Veronica, Sanchis, Ivan, Siano, Alvaro S
PaperDevelopment of caged non-hydrolyzable phosphoamino acids and application to photo-control of binding affinity of phosphopeptide mimetic to phosphopeptide-recognizing protein.
Full title: Development of caged non-hydrolyzable phosphoamino acids and application to photo-control of binding affinity of phosphopeptide mimetic to phosphopeptide-recognizing protein.
PaperGeneration of a glycosylated asparagine residue through chemoselective acylation of a glycosylhydrazide.
Rykaczewski, Katie A, Sabourin, Kate E, Goo, Paul J, Griggs, Lydia H, Jain, Saumya, Reed, Paxton A M, Langenhan, Joseph M · 2020 · Carbohydrate research · DOI
Full title: Generation of a glycosylated asparagine residue through chemoselective acylation of a glycosylhydrazide.
Authors: Rykaczewski, Katie A, Sabourin, Kate E, Goo, Paul J, Griggs, Lydia H, Jain, Saumya, Reed, Paxton A M, Langenhan, Joseph M
PaperPeptide-based targeted cancer therapeutics: design, synthesis and biological evaluation.
Iwan Iwanov, Arianna Rossi, M. Montesi, I. Doytchinova, A. Sargsyan, G. Momekov, S. Panseri, E. Naydenova · 2022 · European Journal of Pharmaceutical Sciences · DOI
Full title: Peptide-based targeted cancer therapeutics: design, synthesis and biological evaluation.
Authors: Iwan Iwanov, Arianna Rossi, M. Montesi, I. Doytchinova, A. Sargsyan, G. Momekov, S. Panseri, E. Naydenova
Year: 2022
Venue: European Journal of Pharmaceutical Sciences
PaperCyclic N-locked indolicidin analogues with antimicrobial activity: Effect of ring size and fatty acid acylation
Lone, Abdullah, Nielsen, Josefine Eilsø, Thulstrup, Peter W., Lund, Reidar, Hansen, Per Brinch, Jenssen, Håvard · 2022 · European Journal of Medicinal Chemistry Reports · DOI
Full title: Cyclic N-locked indolicidin analogues with antimicrobial activity: Effect of ring size and fatty acid acylation
Authors: Lone, Abdullah, Nielsen, Josefine Eilsø, Thulstrup, Peter W., Lund, Reidar, Hansen, Per Brinch, Jenssen, Håvard
Year: 2022
Venue: European Journal of Medicinal Chemistry Reports
PaperPeptide-derivatized biodegradable nanoparticles able to cross the blood-brain barrier.
Costantino, Luca, Gandolfi, Francesca, Tosi, Giovanni, Rivasi, Francesco, Vandelli, Maria Angela, Forni, Flavio · 2005 · Journal of controlled release : official journal of the Controlled Release Society · DOI
Full title: Peptide-derivatized biodegradable nanoparticles able to cross the blood-brain barrier.
PaperSynthesis, radiolabeling and biological evaluation of a neutral tripeptide and its derivatives for potential nuclear medicine applications.
Chandra, Susmita, De, Kakali, Ganguly, Santanu, Sarkar, Bharat, Misra, Mridula · 2009 · Peptides · DOI
Full title: Synthesis, radiolabeling and biological evaluation of a neutral tripeptide and its derivatives for potential nuclear medicine applications.
PaperDevelopment and validation of a reversed-phase high-performance liquid chromatographic method for quantification of peptide dendrimers in human skin permeation experiments.
Mutalik, S, Hewavitharana, A K, Shaw, P N, Anissimov, Y G, Roberts, M S, Parekh, H S · 2009 · Journal of chromatography. B, Analytical technologies in the biomedical and life sciences · DOI
Full title: Development and validation of a reversed-phase high-performance liquid chromatographic method for quantification of peptide dendrimers in human skin permeation experiments.
Authors: Mutalik, S, Hewavitharana, A K, Shaw, P N, Anissimov, Y G, Roberts, M S, Parekh, H S
Year: 2009
Venue: Journal of chromatography. B, Analytical technologies in the biomedical and life sciences
PaperSynthesis, biophysical, and biological studies of wild-type and mutant psalmopeotoxins--anti-malarial cysteine knot peptides from Psalmopoeus cambridgei.
Full title: Synthesis, biophysical, and biological studies of wild-type and mutant psalmopeotoxins--anti-malarial cysteine knot peptides from Psalmopoeus cambridgei.
PaperA highly sensitive and selective fluorescent "on-off-on" peptide-based probe for sequential detection of Hg2+ and S2- ions: Applications in living cells and zebrafish imaging.
Miao Zhou, Maoyue Zheng, Weiliang Deng, Na Kong, Jinglan Hu, Peng Wang, Xiupei Yang · 2024 · Spectrochimica Acta Part A - Molecular and Biomolecular Spectroscopy · DOI
Full title: A highly sensitive and selective fluorescent "on-off-on" peptide-based probe for sequential detection of Hg2+ and S2- ions: Applications in living cells and zebrafish imaging.
Authors: Miao Zhou, Maoyue Zheng, Weiliang Deng, Na Kong, Jinglan Hu, Peng Wang, Xiupei Yang
Year: 2024
Venue: Spectrochimica Acta Part A - Molecular and Biomolecular Spectroscopy
PaperSolid-phase peptide synthesis of analogues of the N-terminus A-ring fragment of the lantibiotic nisin: Replacements for the dehydroalanine (Dha) residue at position 5 and the first incorporation of a thioamide residue
Kim Manzor, Keith ó Proinsias, F. Kelleher · 2017 · DOI
Full title: Solid-phase peptide synthesis of analogues of the N-terminus A-ring fragment of the lantibiotic nisin: Replacements for the dehydroalanine (Dha) residue at position 5 and the first incorporation of a thioamide residue
Authors: Kim Manzor, Keith ó Proinsias, F. Kelleher
PaperPreparation of Peptide Thioesters using Fmoc-Solid-Phase Peptide Synthesis and its Application to the Construction of a Template-Assembled Synthetic Protein (TASP)
Full title: Preparation of Peptide Thioesters using Fmoc-Solid-Phase Peptide Synthesis and its Application to the Construction of a Template-Assembled Synthetic Protein (TASP)
PaperSynthesis and biological evaluation of enantiopure thionitrites: the solid-phase synthesis and nitrosation of D-glutathione as a molecular probe.
Cavero, M, Hobbs, A, Madge, D, Motherwell, W B, Selwood, D, Potier, P · 2000 · Bioorganic & medicinal chemistry letters · DOI
Full title: Synthesis and biological evaluation of enantiopure thionitrites: the solid-phase synthesis and nitrosation of D-glutathione as a molecular probe.
Authors: Cavero, M, Hobbs, A, Madge, D, Motherwell, W B, Selwood, D, Potier, P
PaperA new class of compounds, peptide derivatives of adenosine 5'-carboxylic acid, includes inhibitors of ATP receptor-mediated responses.
Uri, A, Järlebark, L, von Kügelgen, I, Schönberg, T, Undén, A, Heilbronn, E · 1994 · Bioorganic & medicinal chemistry · DOI
Full title: A new class of compounds, peptide derivatives of adenosine 5'-carboxylic acid, includes inhibitors of ATP receptor-mediated responses.
Authors: Uri, A, Järlebark, L, von Kügelgen, I, Schönberg, T, Undén, A, Heilbronn, E
Full title: A Custom-Engineered Water-Soluble Peptide-Based Macrocyclic Polynuclear Gd3+-Chelated Paramagnetic Multimodal Contrast Agent for Mitochondria-Targeted Fluorescence Imaging Integrated with MRI.
PaperDeprotection and cleavage of peptides bound to Merrifield resin by stable dimethyl ether-poly(hydrogen fluoride) (DMEPHF) complex. a new and convenient reagent for peptide chemistry.
Török, Béla, Bucsi, Imre, Prakash, G K Surya, Olah, George A · 2002 · Chemical communications (Cambridge, England) · DOI
Full title: Deprotection and cleavage of peptides bound to Merrifield resin by stable dimethyl ether-poly(hydrogen fluoride) (DMEPHF) complex. a new and convenient reagent for peptide chemistry.
Authors: Török, Béla, Bucsi, Imre, Prakash, G K Surya, Olah, George A
Year: 2002
Venue: Chemical communications (Cambridge, England)
PaperStereoselective synthesis of alpha-monofluorinated phosphonate mimetics of naturally occurring phosphoserine and phosphothreonine, via electrophilic fluorination of lithiated bis-lactim ethers.
Ruiz, María, Ojea, Vicente, Quintela, José M, Guillín, Juan J · 2002 · Chemical communications (Cambridge, England) · DOI
Full title: Stereoselective synthesis of alpha-monofluorinated phosphonate mimetics of naturally occurring phosphoserine and phosphothreonine, via electrophilic fluorination of lithiated bis-lactim ethers.
Authors: Ruiz, María, Ojea, Vicente, Quintela, José M, Guillín, Juan J
Year: 2002
Venue: Chemical communications (Cambridge, England)
PaperA general sequence independent solid phase method for the site specific synthesis of multiple sulfated-tyrosine containing peptides.
Bunschoten, Anton, Kruijtzer, John A W, Ippel, Johannes H, de Haas, Carla J C, van Strijp, Jos A G, Kemmink, Johan, Liskamp, Rob M J · 2009 · Chemical communications (Cambridge, England) · DOI
Full title: A general sequence independent solid phase method for the site specific synthesis of multiple sulfated-tyrosine containing peptides.
Authors: Bunschoten, Anton, Kruijtzer, John A W, Ippel, Johannes H, de Haas, Carla J C, van Strijp, Jos A G, Kemmink, Johan, Liskamp, Rob M J
Year: 2009
Venue: Chemical communications (Cambridge, England)
PaperPhotorelease of tyrosine from α-carboxy-6-nitroveratryl (αCNV) derivatives.
Russell, Alexander G, Sadler, Matthew J, Laidlaw, Helen J, Gutiérrez-Loriente, Agustín, Wharton, Christopher W, Carteau, David, Bassani, Dario M, Snaith, John S · 2012 · Photochemical & photobiological sciences : Official journal of the European Photochemistry Association and the European Society for Photobiology · DOI
Full title: Photorelease of tyrosine from α-carboxy-6-nitroveratryl (αCNV) derivatives.
Authors: Russell, Alexander G, Sadler, Matthew J, Laidlaw, Helen J, Gutiérrez-Loriente, Agustín, Wharton, Christopher W, Carteau, David, Bassani, Dario M, Snaith, John S
Year: 2012
Venue: Photochemical & photobiological sciences : Official journal of the European Photochemistry Association and the European Society for Photobiology
PaperStereoselective synthesis of Arabidopsis CLAVATA3 (CLV3) glycopeptide, unique protein post-translational modifications of secreted peptide hormone in plant.
Full title: Stereoselective synthesis of Arabidopsis CLAVATA3 (CLV3) glycopeptide, unique protein post-translational modifications of secreted peptide hormone in plant.
PaperDirected self-assembly of peptide-diketopyrrolopyrrole conjugates - a platform for bio-organic thin film preparation.
Aakanksha Rani, I. Kavianinia, P. Hume, Luis M. De Leon-Rodriguez, Shinji Kihara, David E. Williams, D. McGillivray, N. Plank, J. Gerrard, J. Hodgkiss, M. Brimble · 2020 · Soft Matter · DOI
Full title: Directed self-assembly of peptide-diketopyrrolopyrrole conjugates - a platform for bio-organic thin film preparation.
Authors: Aakanksha Rani, I. Kavianinia, P. Hume, Luis M. De Leon-Rodriguez, Shinji Kihara, David E. Williams, D. McGillivray, N. Plank, J. Gerrard, J. Hodgkiss, M. Brimble
PaperOptimized solid phase-assisted synthesis of dendrons applicable as scaffolds for radiolabeled bioactive multivalent compounds intended for molecular imaging.
Fischer, Gabriel, Wängler, Björn, Wängler, Carmen · 2014 · Molecules (Basel, Switzerland) · DOI
Full title: Optimized solid phase-assisted synthesis of dendrons applicable as scaffolds for radiolabeled bioactive multivalent compounds intended for molecular imaging.
Authors: Fischer, Gabriel, Wängler, Björn, Wängler, Carmen
PaperUnlocking the Potential of the Antimicrobial Peptide Gomesin: From Discovery and Structure-Activity Relationships to Therapeutic Applications.
Liu, Xiaorong, Henriques, Sónia T, Craik, David J, Chan, Lai Yue · 2023 · International journal of molecular sciences · DOI
Full title: Unlocking the Potential of the Antimicrobial Peptide Gomesin: From Discovery and Structure-Activity Relationships to Therapeutic Applications.
Authors: Liu, Xiaorong, Henriques, Sónia T, Craik, David J, Chan, Lai Yue
Year: 2023
Venue: International journal of molecular sciences
PaperSynthesis, Antimalarial Activity and Molecular Dynamics Studies of Pipecolisporin: A Novel Cyclic Hexapeptide with Potent Therapeutic Potential
Kurniaty, Nety; Fakih, Taufik Muhammad; Maharani, Rani et al. · 2025 · Molecules · DOI
Full title: Synthesis, Antimalarial Activity and Molecular Dynamics Studies of Pipecolisporin: A Novel Cyclic Hexapeptide with Potent Therapeutic Potential
PaperChallenges in the Characterization and Purification of (Peptide)n-Calix[4]Resorcinarene Conjugates Synthesized via Thiol-Maleimide Reaction Using Liquid Chromatography
Niño‐Ramírez, Victor Alfonso; Maldonado, Mauricio; Cuero-Amu, Kelin Johana et al. · 2025 · Processes · DOI
Full title: Challenges in the Characterization and Purification of (Peptide)n-Calix[4]Resorcinarene Conjugates Synthesized via Thiol-Maleimide Reaction Using Liquid Chromatography
Authors: Niño‐Ramírez, Victor Alfonso; Maldonado, Mauricio; Cuero-Amu, Kelin Johana; García‐Castañeda, Javier Eduardo; Rivera‐Monroy, Zuly Jenny
PaperDevelopment of a Polyclonal Antibody for the Immunoanalysis of Ochratoxin A (OTA) by Employing a Specially Designed Synthetic OTA Derivative as the Immunizing Hapten.
Full title: Development of a Polyclonal Antibody for the Immunoanalysis of Ochratoxin A (OTA) by Employing a Specially Designed Synthetic OTA Derivative as the Immunizing Hapten.
PaperSolid phase synthesis, radiolabeling and biological evaluation of a (99m) Tc-labeled α(V)β(3) tripeptide (RGD) conjugated to DOTA as a tumor imaging agent.
Full title: Solid phase synthesis, radiolabeling and biological evaluation of a (99m) Tc-labeled α(V)β(3) tripeptide (RGD) conjugated to DOTA as a tumor imaging agent.
Paper[Synthetic conformational antigen, simulating the extracellular part of M2-muscarinic receptor and its reactivity with sera from patients with idiopathic arrhythmias].
Pal'keeva, M E, Sidorova, M V, Molokoedov, A S, Az'muko, A A, Bespalova, Zh D, Sharf, T V, Mamochkina, E N, Efremov, E E, Rogova, M M, Mironova, N A, Zykov, K A, Golitsyn, S P · 2013 · Bioorganicheskaia khimiia · DOI
Full title: [Synthetic conformational antigen, simulating the extracellular part of M2-muscarinic receptor and its reactivity with sera from patients with idiopathic arrhythmias].
Authors: Pal'keeva, M E, Sidorova, M V, Molokoedov, A S, Az'muko, A A, Bespalova, Zh D, Sharf, T V, Mamochkina, E N, Efremov, E E, Rogova, M M, Mironova, N A, Zykov, K A, Golitsyn, S P
Full title: AGEing Peptides: Synthesis and Analysis of Peptides Site-Specifically Modified by Advanced Glycation Endproducts
Authors: Kamalov, Meder
Year: 2015
Venue: ResearchSPAce (Bath Spa University)
Paper[Application of multiple antigen peptide immunomagnetic beads in single-epitope antibody preparation].
Xu, Xiao-jie, Zhang, Wen-hong, Kang, Lei, Han, Feng-chan, Yan, Zhen, Yan, Xiao-jun · 2007 · Xi bao yu fen zi mian yi xue za zhi = Chinese journal of cellular and molecular immunology
Full title: [Application of multiple antigen peptide immunomagnetic beads in single-epitope antibody preparation].
PaperAn investigation into the key structural role of glycosylated lysine residues in the collagenous domain of adiponectin, a potential therapeutic for type II diabetes
Full title: An investigation into the key structural role of glycosylated lysine residues in the collagenous domain of adiponectin, a potential therapeutic for type II diabetes
Authors: KR, Lutteroth,
Year: 2017
Venue: ResearchSPAce (Bath Spa University)
PaperA swellographic approach to monitoring continuous-flow solid-phase peptide synthesis.
Rodionov, I L; Baru, M B; Ivanov, V T · 1992 · Peptide research
Full title: A swellographic approach to monitoring continuous-flow solid-phase peptide synthesis.
Authors: Rodionov, I L; Baru, M B; Ivanov, V T
Year: 1992
Venue: Peptide research
PaperConformational studies on beta-amyloid protein carboxy-terminal region (residues 34-42): strategic use of amide backbone protection as a structural probe.
Quibell, M, Johnson, T, Turnell, W G · 1994 · Biomedical peptides, proteins & nucleic acids : structure, synthesis & biological activity
Full title: Conformational studies on beta-amyloid protein carboxy-terminal region (residues 34-42): strategic use of amide backbone protection as a structural probe.
PaperAdvances in automatic, manual and microwave-assisted solid-phase peptide synthesis.
Sabatino, Giuseppina, Papini, Anna M · 2008 · Current opinion in drug discovery & development
Full title: Advances in automatic, manual and microwave-assisted solid-phase peptide synthesis.
Authors: Sabatino, Giuseppina, Papini, Anna M
Year: 2008
Venue: Current opinion in drug discovery & development
PaperCleavage of λDNA by Seryl-histidine Planted Peptide Dendrimer
Zhao Yu · 2006 · Gaodeng xuexiao huaxue xuebao
Full title: Cleavage of λDNA by Seryl-histidine Planted Peptide Dendrimer
Authors: Zhao Yu
Year: 2006
Venue: Gaodeng xuexiao huaxue xuebao
PaperCLipPA Lipidation in the Synthesis of a New Generation of Polymyxin Analogues
Mao, Yubing · 2019
Full title: CLipPA Lipidation in the Synthesis of a New Generation of Polymyxin Analogues
Authors: Mao, Yubing
Year: 2019
PaperDesign of Peptides to Interfere with the RANK-TRAF6 Pathway: an Integrated Approach
Pereira, Mafalda Inês Apolinário · 2018 · Portuguese National Funding Agency for Science, Research and Technology (RCAAP Project by FCT)
Full title: Design of Peptides to Interfere with the RANK-TRAF6 Pathway: an Integrated Approach
Authors: Pereira, Mafalda Inês Apolinário
Year: 2018
Venue: Portuguese National Funding Agency for Science, Research and Technology (RCAAP Project by FCT)
Paper[Directed and spontaneous disulfide bond closure using hydrogen peroxide in the synthesis of endothelins-1 and -3].
Kudriavtseva, E V, Sidorova, M V, Molokoedov, A S, Ovchinnikov, M V, Bespalova, Zh D · 1999 · Bioorganicheskaia khimiia
Full title: [Directed and spontaneous disulfide bond closure using hydrogen peroxide in the synthesis of endothelins-1 and -3].
Authors: Kudriavtseva, E V, Sidorova, M V, Molokoedov, A S, Ovchinnikov, M V, Bespalova, Zh D
Year: 1999
Venue: Bioorganicheskaia khimiia
PaperEnhancement of Oral Drug Absorption - Effect of Lipid and Glycoside Conjugation on the Enzymatic Stability and Intestinal Permeability of IM862
Bergeon, Julie A., Chan, Yiu‐Ngok, Tóth, Ildikó V. · 2007 · Queensland's institutional digital repository (The University of Queensland)
Full title: Enhancement of Oral Drug Absorption - Effect of Lipid and Glycoside Conjugation on the Enzymatic Stability and Intestinal Permeability of IM862
Authors: Bergeon, Julie A., Chan, Yiu‐Ngok, Tóth, Ildikó V.
Year: 2007
Venue: Queensland's institutional digital repository (The University of Queensland)
PaperConvergent solid-phase peptide synthesis IX: application to the synthesis of peptides with repetitive sequences.
Celma, C, Albericio, F, Pedroso, E, Giralt, E · 1992 · Peptide research
Full title: Convergent solid-phase peptide synthesis IX: application to the synthesis of peptides with repetitive sequences.
Authors: Celma, C, Albericio, F, Pedroso, E, Giralt, E
Year: 1992
Venue: Peptide research
PaperSynthesis of Mannosylated Lipopeptides with Receptor Targeting Properties.
Sedaghat, Bita, Stephenson, Rachel J, Giddam, Ashwini Kumar, Eskandari, Sharareh, Apte, Simon H, Pattinson, David J, Doolan, Denise L, Toth, Istvan · 2016 · Bioconjugate chemistry · DOI
Full title: Synthesis of Mannosylated Lipopeptides with Receptor Targeting Properties.
PaperUsing Chemical Synthesis to Probe Structure-Activity Relationships of the Glycoactive Bacteriocin Glycocin F.
Bisset, Sean W, Yang, Sung-Hyun, Amso, Zaid, Harris, Paul W R, Patchett, Mark L, Brimble, Margaret A, Norris, Gillian E · 2018 · ACS chemical biology · DOI
Full title: Using Chemical Synthesis to Probe Structure-Activity Relationships of the Glycoactive Bacteriocin Glycocin F.
Authors: Bisset, Sean W, Yang, Sung-Hyun, Amso, Zaid, Harris, Paul W R, Patchett, Mark L, Brimble, Margaret A, Norris, Gillian E
PaperEnantioselective Synthesis and Application of Small and Environmentally Sensitive Fluorescent Amino Acids for Probing Biological Interactions.
Noden, Michael, Taylor, Scott D · 2021 · The Journal of organic chemistry · DOI
Full title: Enantioselective Synthesis and Application of Small and Environmentally Sensitive Fluorescent Amino Acids for Probing Biological Interactions.
PaperMimicking of Arginine by Functionalized N(ω)-Carbamoylated Arginine As a New Broadly Applicable Approach to Labeled Bioactive Peptides: High Affinity Angiotensin, Neuropeptide Y, Neuropeptide FF, and Neurotensin Receptor Ligands As Examples.
Keller, Max, Kuhn, Kilian K, Einsiedel, Jürgen, Hübner, Harald, Biselli, Sabrina, Mollereau, Catherine, Wifling, David, Svobodová, Jaroslava, Bernhardt, Günther, Cabrele, Chiara, Vanderheyden, Patrick M L, Gmeiner, Peter, Buschauer, Armin · 2016 · Journal of medicinal chemistry · DOI
Full title: Mimicking of Arginine by Functionalized N(ω)-Carbamoylated Arginine As a New Broadly Applicable Approach to Labeled Bioactive Peptides: High Affinity Angiotensin, Neuropeptide Y, Neuropeptide FF, and Neurotensin Receptor Ligands As Examples.
Northrup, Justin D, Wiener, Jesse A, Hurley, Matthew F D, Hou, Chun-Feng David, Keller, Taylor M, Baxter, Richard H G, Zdilla, Michael J, Voelz, Vincent A, Schafmeister, Christian E · 2021 · The Journal of organic chemistry · DOI
Full title: Metal-Binding Q-Proline Macrocycles.
Authors: Northrup, Justin D, Wiener, Jesse A, Hurley, Matthew F D, Hou, Chun-Feng David, Keller, Taylor M, Baxter, Richard H G, Zdilla, Michael J, Voelz, Vincent A, Schafmeister, Christian E
PaperProcess Development of a Macrocyclic Peptide Inhibitor of PD-L1.
Subha Mukherjee, Amanda J. Rogers, Gardner Creech, Chao Hang, Antonio Ramirez, Michael Dummeldinger, Shawn Brueggemeier, C. Mapelli, Serge Zaretsky, Masano Huang, R. Black, Michael Peddicord, N. Cunière, J. Kempson, J. Pawluczyk, Martin P Allen, R. Parsons, Chris Sfouggatakis · 2024 · Journal of Organic Chemistry · DOI
Full title: Process Development of a Macrocyclic Peptide Inhibitor of PD-L1.
Authors: Subha Mukherjee, Amanda J. Rogers, Gardner Creech, Chao Hang, Antonio Ramirez, Michael Dummeldinger, Shawn Brueggemeier, C. Mapelli, Serge Zaretsky, Masano Huang, R. Black, Michael Peddicord, N. Cunière, J. Kempson, J. Pawluczyk, Martin P Allen, R. Parsons, Chris Sfouggatakis
PaperAdvancing Sustainable Synthesis of Cyclic Peptides by Integrating Aqueous Fmoc/t-Bu Solid-Phase Peptide Synthesis with Disulfide Bond Formation and TFA/PFAS-Free Resin Cleavage.
Pawlas, Jan, Qvist, Thilda, Haugaard-Kedström, Linda M · 2025 · The Journal of organic chemistry · DOI
Full title: Advancing Sustainable Synthesis of Cyclic Peptides by Integrating Aqueous Fmoc/t-Bu Solid-Phase Peptide Synthesis with Disulfide Bond Formation and TFA/PFAS-Free Resin Cleavage.
Authors: Pawlas, Jan, Qvist, Thilda, Haugaard-Kedström, Linda M
Paperα-Azido Acids in Solid-Phase Peptide Synthesis: Compatibility with Fmoc Chemistry and an Alternative Approach to the Solid Phase Synthesis of Daptomycin Analogs.
Lohani, Chuda Raj, Rasera, Benjamin, Scott, Bradley, Palmer, Michael, Taylor, Scott D · 2016 · The Journal of organic chemistry · DOI
Full title: α-Azido Acids in Solid-Phase Peptide Synthesis: Compatibility with Fmoc Chemistry and an Alternative Approach to the Solid Phase Synthesis of Daptomycin Analogs.
Authors: Lohani, Chuda Raj, Rasera, Benjamin, Scott, Bradley, Palmer, Michael, Taylor, Scott D
PaperSynthesis and SAR Analysis of Lipovelutibols B and D and Their Lipid Analogues.
Cameron, Alan J, Davison, Emma K, An, Chalice, Stubbing, Louise A, Dunbar, P Rod, Harris, Paul W R, Brimble, Margaret A · 2020 · The Journal of organic chemistry · DOI
Full title: Synthesis and SAR Analysis of Lipovelutibols B and D and Their Lipid Analogues.
Authors: Cameron, Alan J, Davison, Emma K, An, Chalice, Stubbing, Louise A, Dunbar, P Rod, Harris, Paul W R, Brimble, Margaret A
PaperMultiple Synthetic Routes to the Mini-Protein Omomyc and Coiled-Coil Domain Truncations.
Brown, Zachary Z, Mapelli, Claudio, Farasat, Iman, Shoultz, Alycia V, Johnson, Scott A, Orvieto, Federica, Santoprete, Alessia, Bianchi, Elisabetta, McCracken, Amy Bittner, Chen, Kuanchang, Zhu, Xiaohong, Demma, Mark J, Lacey, Brian M, Canada, Keith A, Garbaccio, Robert M, O'Neil, Jennifer, Walji, Abbas · 2020 · The Journal of organic chemistry · DOI
Full title: Multiple Synthetic Routes to the Mini-Protein Omomyc and Coiled-Coil Domain Truncations.
Authors: Brown, Zachary Z, Mapelli, Claudio, Farasat, Iman, Shoultz, Alycia V, Johnson, Scott A, Orvieto, Federica, Santoprete, Alessia, Bianchi, Elisabetta, McCracken, Amy Bittner, Chen, Kuanchang, Zhu, Xiaohong, Demma, Mark J, Lacey, Brian M, Canada, Keith A, Garbaccio, Robert M, O'Neil, Jennifer, Walji, Abbas
PaperSynthesis of the Antifungal and Antiviral Cyclic Lipodepsipeptides Verlamelins A and B.
Palpal-Latoc, Dennise, Hauk, Bernhard N, Rajchakit, Urawadee, Lin, Yongqi, Yang, Sung-Hyun, Stubbing, Louise A, Li, Freda F, Cameron, Alan J, Brimble, Margaret A · 2026 · The Journal of organic chemistry · DOI
Full title: Synthesis of the Antifungal and Antiviral Cyclic Lipodepsipeptides Verlamelins A and B.
Authors: Palpal-Latoc, Dennise, Hauk, Bernhard N, Rajchakit, Urawadee, Lin, Yongqi, Yang, Sung-Hyun, Stubbing, Louise A, Li, Freda F, Cameron, Alan J, Brimble, Margaret A
PaperSynthetic Peptides in Doping Control: A Powerful Tool for an Analytical Challenge
Néstor Alejandro Gómez-Guerrero, Nicolás Mateo González-López, Juan Diego Zapata-Velásquez, Jorge Ariel Martínez-Ramírez, Z. Rivera-Monroy, J. García‐Castañeda · 2022 · ACS Omega · DOI
Full title: Synthetic Peptides in Doping Control: A Powerful Tool for an Analytical Challenge
Authors: Néstor Alejandro Gómez-Guerrero, Nicolás Mateo González-López, Juan Diego Zapata-Velásquez, Jorge Ariel Martínez-Ramírez, Z. Rivera-Monroy, J. García‐Castañeda
PaperDevelopment of High-Functionality and -Quality Lipids with RGD Peptide Ligands: Application for PEGylated Liposomes and Analysis of Intratumoral Distribution in a Murine Colon Cancer Model.
Tadaharu Suga, Naoya Kato, Masayori Hagimori, Yuki Fuchigami, N. Kuroda, Yukinobu Kodama, H. Sasaki, S. Kawakami · 2018 · Molecular Pharmaceutics · DOI
Full title: Development of High-Functionality and -Quality Lipids with RGD Peptide Ligands: Application for PEGylated Liposomes and Analysis of Intratumoral Distribution in a Murine Colon Cancer Model.
Authors: Tadaharu Suga, Naoya Kato, Masayori Hagimori, Yuki Fuchigami, N. Kuroda, Yukinobu Kodama, H. Sasaki, S. Kawakami
PaperHybrid Cyclic-Linear Cell-Penetrating Peptides Containing Alternative Positively Charged and Hydrophobic Residues as Molecular Transporters.
Khayyatnejad Shoushtari, Sorour, Zoghebi, Khalid, Sajid, Muhammad Imran, Tiwari, Rakesh Kumar, Parang, Keykavous · 2021 · Molecular pharmaceutics · DOI
Full title: Hybrid Cyclic-Linear Cell-Penetrating Peptides Containing Alternative Positively Charged and Hydrophobic Residues as Molecular Transporters.
PaperSynthesis of O-Sulfated Human Syndecan-1-like Glyco-polypeptides by Incorporating Peptide Ligation and O-Sulfated Glycopeptide Cassette Strategies.
Full title: Synthesis of O-Sulfated Human Syndecan-1-like Glyco-polypeptides by Incorporating Peptide Ligation and O-Sulfated Glycopeptide Cassette Strategies.
PaperBrønsted Acid-Lewis Acid (BA-LA) Induced Final Deprotection/Peptide Resin Cleavage in Fmoc/t-Bu Solid-Phase Peptide Synthesis: HCl/FeCl3 and AcOH/FeCl3 as Viable PFAS-Free Alternatives for TFA.
Pawlas, Jan, André, Christophe, Rasmussen, Jon H, Ludemann-Hombourger, Olivier · 2024 · Organic letters · DOI
Full title: Brønsted Acid-Lewis Acid (BA-LA) Induced Final Deprotection/Peptide Resin Cleavage in Fmoc/t-Bu Solid-Phase Peptide Synthesis: HCl/FeCl3 and AcOH/FeCl3 as Viable PFAS-Free Alternatives for TFA.
Authors: Pawlas, Jan, André, Christophe, Rasmussen, Jon H, Ludemann-Hombourger, Olivier
Giltrap, Andrew M, Dowman, Luke J, Nagalingam, Gayathri, Ochoa, Jessica L, Linington, Roger G, Britton, Warwick J, Payne, Richard J · 2016 · Organic letters · DOI
Full title: Total Synthesis of Teixobactin.
Authors: Giltrap, Andrew M, Dowman, Luke J, Nagalingam, Gayathri, Ochoa, Jessica L, Linington, Roger G, Britton, Warwick J, Payne, Richard J
PaperAn Entirely Solid Phase Peptide Synthesis-Based Strategy for Synthesis of Gelatinase Biosynthesis-Activating Pheromone (GBAP) Analogue Libraries: Investigating the Structure-Activity Relationships of the Enterococcus faecalis Quorum Sensing Signal.
McBrayer, Dominic N, Gantman, Brooke K, Cameron, Crissey D, Tal-Gan, Yftah · 2017 · Organic letters · DOI
Full title: An Entirely Solid Phase Peptide Synthesis-Based Strategy for Synthesis of Gelatinase Biosynthesis-Activating Pheromone (GBAP) Analogue Libraries: Investigating the Structure-Activity Relationships of the Enterococcus faecalis Quorum Sensing Signal.
PaperInteraction of alpha-dansylated peptide inhibitors with porcine pepsin: detection of complex formation by fluorescence energy transfer and chromatography and evidence for a two-step binding scheme.
Dunn, B M, Pham, C, Raney, L, Abayasekara, D, Gillespie, W, Hsu, A · 1981 · Biochemistry · DOI
Full title: Interaction of alpha-dansylated peptide inhibitors with porcine pepsin: detection of complex formation by fluorescence energy transfer and chromatography and evidence for a two-step binding scheme.
Authors: Dunn, B M, Pham, C, Raney, L, Abayasekara, D, Gillespie, W, Hsu, A
PaperAza-amino acid scanning of secondary structure suited for solid-phase peptide synthesis with fmoc chemistry and aza-amino acids with heteroatomic side chains.
D. Boeglin, W. Lubell · 2005 · Journal of combinatorial chemistry · DOI
Full title: Aza-amino acid scanning of secondary structure suited for solid-phase peptide synthesis with fmoc chemistry and aza-amino acids with heteroatomic side chains.
PaperLabeling of the neuropeptide enkephalin with functionalized tris(pyrazolyl)borate complexes: solid-phase synthesis and characterization of p-[Enk-OH]COC6H4TpPtMe3 and p-[Enk-OH]COC6H4TpMeRe(CO)3.
Kuchta, Matthew C, Gross, Annika, Pinto, Antonio, Metzler-Nolte, Nils · 2007 · Inorganic chemistry · DOI
Full title: Labeling of the neuropeptide enkephalin with functionalized tris(pyrazolyl)borate complexes: solid-phase synthesis and characterization of p-[Enk-OH]COC6H4TpPtMe3 and p-[Enk-OH]COC6H4TpMeRe(CO)3.
Authors: Kuchta, Matthew C, Gross, Annika, Pinto, Antonio, Metzler-Nolte, Nils
PaperChemical synthesis of a glycoprotein having an intact human complex-type sialyloligosaccharide under the Boc and Fmoc synthetic strategies.
Yamamoto, Naoki, Tanabe, Yasutaka, Okamoto, Ryo, Dawson, Philip E, Kajihara, Yasuhiro · 2008 · Journal of the American Chemical Society · DOI
Full title: Chemical synthesis of a glycoprotein having an intact human complex-type sialyloligosaccharide under the Boc and Fmoc synthetic strategies.
Authors: Yamamoto, Naoki, Tanabe, Yasutaka, Okamoto, Ryo, Dawson, Philip E, Kajihara, Yasuhiro
PaperA novel Tc-99m and fluorescence-labeled arginine-arginine-leucine-containing peptide as a multimodal tumor imaging agent in a murine tumor model.
Kim, Myoung Hyoun, Kim, Seul-Gi, Kim, Dae-Weung · 2018 · Journal of labelled compounds & radiopharmaceuticals · DOI
Full title: A novel Tc-99m and fluorescence-labeled arginine-arginine-leucine-containing peptide as a multimodal tumor imaging agent in a murine tumor model.
Authors: Kim, Myoung Hyoun, Kim, Seul-Gi, Kim, Dae-Weung
Year: 2018
Venue: Journal of labelled compounds & radiopharmaceuticals
PaperSynthesis and evaluation of Tc-99m and fluorescence-labeled elastin-derived peptide, VAPG for multimodal tumor imaging in murine tumor model.
Kim, Myoung Hyoun, Kim, Chang Guhn, Kim, Seul-Gi, Kim, Dae-Weung · 2017 · Journal of labelled compounds & radiopharmaceuticals · DOI
Full title: Synthesis and evaluation of Tc-99m and fluorescence-labeled elastin-derived peptide, VAPG for multimodal tumor imaging in murine tumor model.
Authors: Kim, Myoung Hyoun, Kim, Chang Guhn, Kim, Seul-Gi, Kim, Dae-Weung
Year: 2017
Venue: Journal of labelled compounds & radiopharmaceuticals
PaperDual-labeled prostate-specific membrane antigen (PSMA)-targeting agent for preoperative molecular imaging and fluorescence-guided surgery for prostate cancer.
Kim, Myoung Hyoun, Kim, Seul-Gi, Kim, Dae-Weung · 2021 · Journal of labelled compounds & radiopharmaceuticals · DOI
Full title: Dual-labeled prostate-specific membrane antigen (PSMA)-targeting agent for preoperative molecular imaging and fluorescence-guided surgery for prostate cancer.
Authors: Kim, Myoung Hyoun, Kim, Seul-Gi, Kim, Dae-Weung
Year: 2021
Venue: Journal of labelled compounds & radiopharmaceuticals
PaperBioactive mesoglobules of poly(di(ethylene glycol) monomethyl ether methacrylate)–peptide conjugate
Roza Trzcinska, D. Szweda, S. Rangelov, P. Suder, J. Silberring, A. Dworak, B. Trzebicka · 2012 · Journal of Polymer Science Part A Polymer Chemistry · DOI
Full title: Bioactive mesoglobules of poly(di(ethylene glycol) monomethyl ether methacrylate)–peptide conjugate
Authors: Roza Trzcinska, D. Szweda, S. Rangelov, P. Suder, J. Silberring, A. Dworak, B. Trzebicka
Year: 2012
Venue: Journal of Polymer Science Part A Polymer Chemistry
PaperConformational studies of [Abu(3, 11)]-SFTI-1, an analogue of the trypsin inhibitor isolated from sunflower seeds.
Brzozowski, Krzysztof, Majewski, Radosław, Jaśkiewicz, Anna, Legowska, Anna, Klaudel, Lidia, Rodziewicz-Motowidło, Sylwia, Rolka, Krzysztof · 2008 · Journal of peptide science : an official publication of the European Peptide Society · DOI
Full title: Conformational studies of [Abu(3, 11)]-SFTI-1, an analogue of the trypsin inhibitor isolated from sunflower seeds.
PaperPreclinical evaluation of a bispecific low-molecular heterodimer targeting both PSMA and GRPR for improved PET imaging and therapy of prostate cancer.
Eder, Matthias, Schäfer, Martin, Bauder-Wüst, Ulrike, Haberkorn, Uwe, Eisenhut, Michael, Kopka, Klaus · 2014 · The Prostate · DOI
Full title: Preclinical evaluation of a bispecific low-molecular heterodimer targeting both PSMA and GRPR for improved PET imaging and therapy of prostate cancer.
PaperSolid-phase peptide synthesis using acetonitrile as a solvent in combination with PEG-based resins.
Acosta, Gerardo A; del Fresno, Montserrat; Paradis-Bas, Marta et al. · 2009 · Journal of peptide science : an official publication of the European Peptide Society · DOI
Full title: Solid-phase peptide synthesis using acetonitrile as a solvent in combination with PEG-based resins.
Authors: Acosta, Gerardo A; del Fresno, Montserrat; Paradis-Bas, Marta; Rigau-DeLlobet, Maria; Côté, Simon; Royo, Miriam; Albericio, Fernando
Year: 2009
Venue: Journal of peptide science : an official publication of the European Peptide Society
PaperPreparation of truncated orf virus entry fusion complex proteins by chemical synthesis.
Yeung, Ho, Harris, Paul W R, Squire, Christopher J, Baker, Edward N, Brimble, Margaret A · 2014 · Journal of peptide science : an official publication of the European Peptide Society · DOI
Full title: Preparation of truncated orf virus entry fusion complex proteins by chemical synthesis.
Authors: Yeung, Ho, Harris, Paul W R, Squire, Christopher J, Baker, Edward N, Brimble, Margaret A
Year: 2014
Venue: Journal of peptide science : an official publication of the European Peptide Society
PaperSynthesis of peptide thioesters via an N-S acyl shift reaction under mild acidic conditions on an N-4,5-dimethoxy-2-mercaptobenzyl auxiliary group.
Nakamura, Ken'ichiroh, Kanao, Tomoki, Uesugi, Tomoya, Hara, Toshiaki, Sato, Takeshi, Kawakami, Toru, Aimoto, Saburo · 2009 · Journal of peptide science : an official publication of the European Peptide Society · DOI
Full title: Synthesis of peptide thioesters via an N-S acyl shift reaction under mild acidic conditions on an N-4,5-dimethoxy-2-mercaptobenzyl auxiliary group.
PaperChemical synthesis of La1 isolated from the venom of the scorpion Liocheles australasiae and determination of its disulfide bonding pattern.
Nagao, Junya, Miyashita, Masahiro, Nakagawa, Yoshiaki, Miyagawa, Hisashi · 2015 · Journal of peptide science : an official publication of the European Peptide Society · DOI
Full title: Chemical synthesis of La1 isolated from the venom of the scorpion Liocheles australasiae and determination of its disulfide bonding pattern.
PaperFacile preparation of the N-acetyl-glucosaminylated asparagine derivative with TFA-sensitive protecting groups useful for solid-phase glycopeptide synthesis.
Katayama, Hidekazu · 2015 · Journal of peptide science : an official publication of the European Peptide Society · DOI
Full title: Facile preparation of the N-acetyl-glucosaminylated asparagine derivative with TFA-sensitive protecting groups useful for solid-phase glycopeptide synthesis.
Authors: Katayama, Hidekazu
Year: 2015
Venue: Journal of peptide science : an official publication of the European Peptide Society
PaperTidbits for the synthesis of bis(2-sulfanylethyl)amido (SEA) polystyrene resin, SEA peptides and peptide thioesters.
Ollivier, Nathalie, Raibaut, Laurent, Blanpain, Annick, Desmet, Rémi, Dheur, Julien, Mhidia, Reda, Boll, Emmanuelle, Drobecq, Hervé, Pira, Silvain L, Melnyk, Oleg · 2014 · Journal of peptide science : an official publication of the European Peptide Society · DOI
Full title: Tidbits for the synthesis of bis(2-sulfanylethyl)amido (SEA) polystyrene resin, SEA peptides and peptide thioesters.
PaperFluorescently labeled adrenomedullin allows real-time monitoring of adrenomedullin receptor trafficking in living cells.
Schönauer, Ria, Kaiser, Anette, Holze, Cathleen, Babilon, Stefanie, Köbberling, Johannes, Riedl, Bernd, Beck-Sickinger, Annette G · 2015 · Journal of peptide science : an official publication of the European Peptide Society · DOI
Full title: Fluorescently labeled adrenomedullin allows real-time monitoring of adrenomedullin receptor trafficking in living cells.
PaperFullerene-based inhibitors of HIV-1 protease.
Strom, T Amanda, Durdagi, Serdar, Ersoz, Suha Salih, Salmas, Ramin Ekhteiari, Supuran, Claudiu T, Barron, Andrew R · 2015 · Journal of peptide science : an official publication of the European Peptide Society · DOI
Full title: Fullerene-based inhibitors of HIV-1 protease.
Authors: Strom, T Amanda, Durdagi, Serdar, Ersoz, Suha Salih, Salmas, Ramin Ekhteiari, Supuran, Claudiu T, Barron, Andrew R
Year: 2015
Venue: Journal of peptide science : an official publication of the European Peptide Society
García-Pindado, Júlia, Royo, Soledad, Teixidó, Meritxell, Giralt, Ernest · 2017 · Journal of peptide science : an official publication of the European Peptide Society · DOI
Full title: Bike peptides: a ride through the membrane.
Authors: García-Pindado, Júlia, Royo, Soledad, Teixidó, Meritxell, Giralt, Ernest
Year: 2017
Venue: Journal of peptide science : an official publication of the European Peptide Society
PaperAn efficient solid-phase synthesis of peptidyl-N-acetylguanidines for use in native chemical ligation.
Okamoto, Ryo, Isoe, Madoka, Izumi, Masayuki, Kajihara, Yasuhiro · 2016 · Journal of peptide science : an official publication of the European Peptide Society · DOI
Full title: An efficient solid-phase synthesis of peptidyl-N-acetylguanidines for use in native chemical ligation.
PaperA comparative study of synthetic and semisynthetic approaches for ligating the epidermal growth factor to a bivalent scaffold.
Gell, Anna Lena, Groysbeck, Nadja, Becker, Christian F W, Conibear, Anne C · 2017 · Journal of peptide science : an official publication of the European Peptide Society · DOI
Full title: A comparative study of synthetic and semisynthetic approaches for ligating the epidermal growth factor to a bivalent scaffold.
Authors: Gell, Anna Lena, Groysbeck, Nadja, Becker, Christian F W, Conibear, Anne C
Year: 2017
Venue: Journal of peptide science : an official publication of the European Peptide Society
PaperSolid-Phase synthesis of a dendritic peptide related to a retinoblastoma protein fragment utilizing a combined boc- and fmoc-chemistry approach.
Cavallaro, V, Thompson, P, Hearn, M · 2001 · Journal of peptide science : an official publication of the European Peptide Society · DOI
Full title: Solid-Phase synthesis of a dendritic peptide related to a retinoblastoma protein fragment utilizing a combined boc- and fmoc-chemistry approach.
Authors: Cavallaro, V, Thompson, P, Hearn, M
Year: 2001
Venue: Journal of peptide science : an official publication of the European Peptide Society
PaperComplete synthesis of the bicyclic ring of a mutacin analog with orthogonally protected lanthionine via solid-phase intracyclization.
Kirichenko, Kostyantyn, Hillman, Jeffrey D, Handfield, Martin, Park, Jae H · 2019 · Journal of peptide science : an official publication of the European Peptide Society · DOI
Full title: Complete synthesis of the bicyclic ring of a mutacin analog with orthogonally protected lanthionine via solid-phase intracyclization.
Authors: Kirichenko, Kostyantyn, Hillman, Jeffrey D, Handfield, Martin, Park, Jae H
Year: 2019
Venue: Journal of peptide science : an official publication of the European Peptide Society
PaperAdrenomedullin disulfide bond mimetics uncover structural requirements for AM1 receptor activation.
Fischer, Jan-Patrick, Schönauer, Ria, Els-Heindl, Sylvia, Bierer, Donald, Koebberling, Johannes, Riedl, Bernd, Beck-Sickinger, Annette G · 2019 · Journal of peptide science : an official publication of the European Peptide Society · DOI
Full title: Adrenomedullin disulfide bond mimetics uncover structural requirements for AM1 receptor activation.
PaperAntimicrobial activity and secondary structure of a novel peptide derived from ovalbumin.
Tan, Ao, Suzuki, Rio, Yokoyama, Chikako, Yano, Shigekazu, Konno, Hiroyuki · 2020 · Journal of peptide science : an official publication of the European Peptide Society · DOI
Full title: Antimicrobial activity and secondary structure of a novel peptide derived from ovalbumin.
PaperRe-evaluating the stability of COMU in different solvents.
Kumar, Ashish; Jad, Yahya E; de la Torre, Beatriz G et al. · 2017 · Journal of peptide science : an official publication of the European Peptide Society · DOI
Full title: Re-evaluating the stability of COMU in different solvents.
Authors: Kumar, Ashish; Jad, Yahya E; de la Torre, Beatriz G; El-Faham, Ayman; Albericio, Fernando
Year: 2017
Venue: Journal of peptide science : an official publication of the European Peptide Society
PaperAutomated solid-phase synthesis of metabolically stabilized triazolo-peptidomimetics.
Guarrochena, Xabier; Kaudela, Barbara; Mindt, Thomas L · 2023 · Journal of peptide science : an official publication of the European Peptide Society · DOI
Full title: Automated solid-phase synthesis of metabolically stabilized triazolo-peptidomimetics.
Authors: Guarrochena, Xabier; Kaudela, Barbara; Mindt, Thomas L
Year: 2023
Venue: Journal of peptide science : an official publication of the European Peptide Society
PaperImproved Fmoc-solid-phase peptide synthesis of an extracellular loop of CFTR for antibody selection by the phage display technology.
Ferreira, Vera F C, Correia, João D G, Farinha, Carlos M, Mendes, Filipa · 2020 · Journal of peptide science : an official publication of the European Peptide Society · DOI
Full title: Improved Fmoc-solid-phase peptide synthesis of an extracellular loop of CFTR for antibody selection by the phage display technology.
Authors: Ferreira, Vera F C, Correia, João D G, Farinha, Carlos M, Mendes, Filipa
Year: 2020
Venue: Journal of peptide science : an official publication of the European Peptide Society
PaperPreparation and characterization of two LysB29 specifically labelled fluorescent derivatives of human insulin.
Ciencialová, Alice, Záková, Lenka, Jirácek, Jiri, Barthová, Jana, Barth, Tomislav · 2004 · Journal of peptide science : an official publication of the European Peptide Society · DOI
Full title: Preparation and characterization of two LysB29 specifically labelled fluorescent derivatives of human insulin.
PaperAlpha- and beta- aspartyl peptide ester formation via aspartimide ring opening.
Stathopoulos, Panagiotis, Papas, Serafim, Kostidis, Sarantos, Tsikaris, Vassilios · 2005 · Journal of peptide science : an official publication of the European Peptide Society · DOI
Full title: Alpha- and beta- aspartyl peptide ester formation via aspartimide ring opening.
PaperSynthesis of Stylissamide B, a Pro-Rich Cyclic Heptapeptide Isolated From the Marine Sponge Stylissa caribica.
Li, Yitong, Ling, Hanyu, Teruya, Kenta, Konno, Hiroyuki · 2025 · Journal of peptide science : an official publication of the European Peptide Society · DOI
Full title: Synthesis of Stylissamide B, a Pro-Rich Cyclic Heptapeptide Isolated From the Marine Sponge Stylissa caribica.
PaperToward a Green SPPS: The Use of an Innovative Mesoporous pDVB Support for Environmentally Friendly Solvents.
Lastella, Luana, Zecca, Marco, Centomo, Paolo, Jeřábek, Karel, Formaggio, Fernando, Guryanov, Ivan, Ricci, Antonio, Biondi, Barbara · 2025 · Journal of peptide science : an official publication of the European Peptide Society · DOI
Full title: Toward a Green SPPS: The Use of an Innovative Mesoporous pDVB Support for Environmentally Friendly Solvents.
PaperSolid-phase peptide synthesis using nanoparticulate amino acids in water.
Hojo, Keiko; Ichikawa, Hideki; Maeda, Mitsuko et al. · 2007 · Journal of peptide science : an official publication of the European Peptide Society · DOI
Full title: Solid-phase peptide synthesis using nanoparticulate amino acids in water.
Nkwanyana, Nonsikelelo, Kumar, Ashish, Chakraborty, Amit, Potvin, Steeves, Thibaut-Koumba, Georges, Nardone, Brunello, Beland, Francois, Sharma, Anamika, de la Torre, Beatriz G, Albericio, Fernando · 2025 · Journal of peptide science : an official publication of the European Peptide Society · DOI
Full title: Silica-Assisted Solid-Phase Peptide Synthesis (SiPPS).
Authors: Nkwanyana, Nonsikelelo, Kumar, Ashish, Chakraborty, Amit, Potvin, Steeves, Thibaut-Koumba, Georges, Nardone, Brunello, Beland, Francois, Sharma, Anamika, de la Torre, Beatriz G, Albericio, Fernando
Year: 2025
Venue: Journal of peptide science : an official publication of the European Peptide Society
PaperSoft shell resins for solid-phase peptide synthesis.
Lee, Tae-Kyung, Choi, Jeong-Hyun, Ryoo, Sun-Jong, Lee, Yoon-Sik · 2007 · Journal of peptide science : an official publication of the European Peptide Society · DOI
Full title: Soft shell resins for solid-phase peptide synthesis.
PaperHeterotrimeric collagen peptides containing functional epitopes. Synthesis of single-stranded collagen type I peptides related to the collagenase cleavage site.
Ottl, J, Musiol, H J, Moroder, L · 1999 · Journal of peptide science : an official publication of the European Peptide Society · DOI
Full title: Heterotrimeric collagen peptides containing functional epitopes. Synthesis of single-stranded collagen type I peptides related to the collagenase cleavage site.
Authors: Ottl, J, Musiol, H J, Moroder, L
Year: 1999
Venue: Journal of peptide science : an official publication of the European Peptide Society
PaperFmoc-based solid phase chemical synthesis of 71-meric neuregulin 1-beta1, an epidermal growth factor-like domain.
Kakizawa, Taeko, Koide-Yoshida, Shizuyo, Kimura, Tooru, Uchimura, Hiromasa, Hayashi, Yoshio, Saito, Kazuki, Kiso, Yoshiaki · 2008 · Journal of peptide science : an official publication of the European Peptide Society · DOI
Full title: Fmoc-based solid phase chemical synthesis of 71-meric neuregulin 1-beta1, an epidermal growth factor-like domain.
PaperDesign, Synthesis, and Anticancer Activity of N‐1 Terminal Segment of α‐(2, 5,7‐Tri‐tert‐butylindol‐3‐yl)alanine‐Incorporated Short Peptides
Rajavenkatesh Krishnamoorthy, Meenakshi Singh, Parthiban Anaikutti, M. C. Pavar, Esthar Selvaraj, Saravanakumar Rajagopal, Rajendran Babhu Vignesh · 2024 · ChemistrySelect · DOI
Full title: Design, Synthesis, and Anticancer Activity of N‐1 Terminal Segment of α‐(2, 5,7‐Tri‐tert‐butylindol‐3‐yl)alanine‐Incorporated Short Peptides
Authors: Rajavenkatesh Krishnamoorthy, Meenakshi Singh, Parthiban Anaikutti, M. C. Pavar, Esthar Selvaraj, Saravanakumar Rajagopal, Rajendran Babhu Vignesh
PaperHigh level of aspartic acid-bond isomerization during the synthesis of an N-linked tau glycopeptide.
Hoffmann, R, Craik, D J, Bokonyi, K, Varga, I, Otvos, L · 1999 · Journal of peptide science : an official publication of the European Peptide Society · DOI
Full title: High level of aspartic acid-bond isomerization during the synthesis of an N-linked tau glycopeptide.
Authors: Hoffmann, R, Craik, D J, Bokonyi, K, Varga, I, Otvos, L
Year: 1999
Venue: Journal of peptide science : an official publication of the European Peptide Society
PaperSynthesis and activity of dimeric bradykinin antagonists containing diaminodicarboxylic acid bridge residues.
Lange, M, Cuthbertson, A S, Towart, R, Fischer, P M · 1998 · Journal of peptide science : an official publication of the European Peptide Society · DOI
Full title: Synthesis and activity of dimeric bradykinin antagonists containing diaminodicarboxylic acid bridge residues.
Authors: Lange, M, Cuthbertson, A S, Towart, R, Fischer, P M
Year: 1998
Venue: Journal of peptide science : an official publication of the European Peptide Society
PaperSynthesis of bivalent inhibitors of eucaryotic proteasomes.
Loidl, G, Musiol, H J, Groll, M, Huber, R, Moroder, L · 2000 · Journal of peptide science : an official publication of the European Peptide Society · DOI
Full title: Synthesis of bivalent inhibitors of eucaryotic proteasomes.
Authors: Loidl, G, Musiol, H J, Groll, M, Huber, R, Moroder, L
Year: 2000
Venue: Journal of peptide science : an official publication of the European Peptide Society
PaperSolid-phase synthesis of caged peptides using tyrosine modified with a photocleavable protecting group: application to the synthesis of caged neuropeptide Y.
Tatsu, Y, Shigeri, Y, Sogabe, S, Yumoto, N, Yoshikawa, S · 1996 · Biochemical and biophysical research communications · DOI
Full title: Solid-phase synthesis of caged peptides using tyrosine modified with a photocleavable protecting group: application to the synthesis of caged neuropeptide Y.
Authors: Tatsu, Y, Shigeri, Y, Sogabe, S, Yumoto, N, Yoshikawa, S
Year: 1996
Venue: Biochemical and biophysical research communications
PaperDesign of Water-Soluble PEGylated Heptapeptide-Based Multifunctional Magnetic Nanovesicles for Cancer Targeted MRI Integrated With Fluorescence Imaging.
Bera, Tapas, Mondal, Aniruddha, Ghosh, Priti, Ganguly, Ipsita, Dutta, Sanjit, Afridi, Sahid, Ghara, Sucharita, Roy, Amalendu, Guha, Samit · 2025 · Small (Weinheim an der Bergstrasse, Germany) · DOI
Full title: Design of Water-Soluble PEGylated Heptapeptide-Based Multifunctional Magnetic Nanovesicles for Cancer Targeted MRI Integrated With Fluorescence Imaging.
PaperEvidence that the major degradation product of glucose-dependent insulinotropic polypeptide, GIP(3-42), is a GIP receptor antagonist in vivo.
Gault, V A, Parker, J C, Harriott, P, Flatt, P R, O'Harte, F P M · 2002 · The Journal of endocrinology · DOI
Full title: Evidence that the major degradation product of glucose-dependent insulinotropic polypeptide, GIP(3-42), is a GIP receptor antagonist in vivo.
Authors: Gault, V A, Parker, J C, Harriott, P, Flatt, P R, O'Harte, F P M
PaperLinear Peptide Analogues from Jatropha’s Orbitides Promote Migration of Human Neonatal Foreskin Fibroblasts in vitro and Collagen Deposition
S. Ramalho, M. Pinto, Renata Andricopulo, P. Sanches, E. Silveira, E. Cilli, A. Andricopulo, V. Bolzani · 2019 · Journal of the Brazilian Chemical Society · DOI
Full title: Linear Peptide Analogues from Jatropha’s Orbitides Promote Migration of Human Neonatal Foreskin Fibroblasts in vitro and Collagen Deposition
Authors: S. Ramalho, M. Pinto, Renata Andricopulo, P. Sanches, E. Silveira, E. Cilli, A. Andricopulo, V. Bolzani
PaperDesign of a New 99mTc-radiolabeled Cyclo-peptide as Promising Molecular Imaging Agent of CXCR4 Receptor: Molecular Docking, Synthesis, Radiolabeling, and Biological Evaluation.
Hassanzadeh, Leila, Erfani, Mostafa, Jokar, Safura, Shariatpanahi, Marjan · 2024 · Current radiopharmaceuticals · DOI
Full title: Design of a New 99mTc-radiolabeled Cyclo-peptide as Promising Molecular Imaging Agent of CXCR4 Receptor: Molecular Docking, Synthesis, Radiolabeling, and Biological Evaluation.
Authors: Hassanzadeh, Leila, Erfani, Mostafa, Jokar, Safura, Shariatpanahi, Marjan
PaperSPED-(styrene-polyethyleneglycol diacrylate-9-decen-1-ol): a novel resin for solid phase peptide synthesis; synthesis and characterization of biologically potent endothelin classes of peptides.
Siyad, Mohammedhaneefa A, Kumar, Gopalakrishnapillai S V · 2012 · Combinatorial chemistry & high throughput screening · DOI
Full title: SPED-(styrene-polyethyleneglycol diacrylate-9-decen-1-ol): a novel resin for solid phase peptide synthesis; synthesis and characterization of biologically potent endothelin classes of peptides.
Authors: Siyad, Mohammedhaneefa A, Kumar, Gopalakrishnapillai S V
Year: 2012
Venue: Combinatorial chemistry & high throughput screening
PaperSolid phase peptide synthesis in water VI: evaluation of water-soluble coupling reagents for solid phase peptide synthesis in aqueous media.
Hojo, Keiko, Maeda, Mitsuko, Tanakamaru, Naoko, Mochida, Kayo, Kawasaki, Koichi · 2006 · Protein and peptide letters · DOI
Full title: Solid phase peptide synthesis in water VI: evaluation of water-soluble coupling reagents for solid phase peptide synthesis in aqueous media.
PaperAn N-terminal selective thiazoline peptide macrocyclisation compatible with mRNA display and efficient SPPS
Liu, Minglong, Morewood, Richard, Yoshisada, Ryoji, Pascha, Mirte N., Hopstaken, Antonius J. P., Tarcoveanu, Eliza, Poole, David A., Haan, Cornelis A. M. de, Nitsche, Christoph, Jongkees, Seino A. K. · 2023 · DOI
Full title: An N-terminal selective thiazoline peptide macrocyclisation compatible with mRNA display and efficient SPPS
Authors: Liu, Minglong, Morewood, Richard, Yoshisada, Ryoji, Pascha, Mirte N., Hopstaken, Antonius J. P., Tarcoveanu, Eliza, Poole, David A., Haan, Cornelis A. M. de, Nitsche, Christoph, Jongkees, Seino A. K.
PaperHistidine 19 Residue Is Essential for Cell Internalization of Antifungal Peptide SmAPα1-21 Derived from the α-Core of the Silybum marianum Defensin DefSm2-D in Fusarium graminearum
Full title: Histidine 19 Residue Is Essential for Cell Internalization of Antifungal Peptide SmAPα1-21 Derived from the α-Core of the Silybum marianum Defensin DefSm2-D in Fusarium graminearum
PaperEfficient access to highly pure β-amyloid peptide by optimized solid-phase synthesis.
Choi, Ji Won; Kim, Hye Yun; Jeon, MiJin et al. · 2012 · Amyloid : the international journal of experimental and clinical investigation : the official journal of the International Society of Amyloidosis · DOI
Full title: Efficient access to highly pure β-amyloid peptide by optimized solid-phase synthesis.
Authors: Choi, Ji Won; Kim, Hye Yun; Jeon, MiJin; Kim, Dong Jin; Kim, YoungSoo
Year: 2012
Venue: Amyloid : the international journal of experimental and clinical investigation : the official journal of the International Society of Amyloidosis
PaperThe Antimicrobial Peptide Capitellacin: Chemical Synthesis of Analogues to Probe the Role of Disulphide Bridges and Their Replacement with Vinyl Sulphides.
Shepperson, Oscar A, Harris, Paul W R, Brimble, Margaret A, Cameron, Alan J · 2024 · Antibiotics (Basel, Switzerland) · DOI
Full title: The Antimicrobial Peptide Capitellacin: Chemical Synthesis of Analogues to Probe the Role of Disulphide Bridges and Their Replacement with Vinyl Sulphides.
Authors: Shepperson, Oscar A, Harris, Paul W R, Brimble, Margaret A, Cameron, Alan J
PaperSolid Phase Synthesis and TAR RNA-Binding Activity of Nucleopeptides Containing Nucleobases Linked to the Side Chains via 1,4-Linked-1,2,3-triazole
P. Mucha, Małgorzata Pieszko, Irena Bylińska, W. Wiczk, J. Ruczyński, Katarzyna Prochera, P. Rekowski · 2024 · Biomedicines · DOI
Full title: Solid Phase Synthesis and TAR RNA-Binding Activity of Nucleopeptides Containing Nucleobases Linked to the Side Chains via 1,4-Linked-1,2,3-triazole
Authors: P. Mucha, Małgorzata Pieszko, Irena Bylińska, W. Wiczk, J. Ruczyński, Katarzyna Prochera, P. Rekowski
PaperNovel Cyclic Lipopeptide Antibiotics: Effects of Acyl Chain Length and Position.
Jensen, Signe Kaustrup, Thomsen, Thomas T, Oddo, Alberto, Franzyk, Henrik, Løbner-Olesen, Anders, Hansen, Paul R · 2020 · International journal of molecular sciences · DOI
Full title: Novel Cyclic Lipopeptide Antibiotics: Effects of Acyl Chain Length and Position.
Authors: Jensen, Signe Kaustrup, Thomsen, Thomas T, Oddo, Alberto, Franzyk, Henrik, Løbner-Olesen, Anders, Hansen, Paul R
Year: 2020
Venue: International journal of molecular sciences
PaperIdentification, Synthesis, Conformation and Activity of an Insulin-like Peptide from a Sea Anemone.
Mitchell, Michela L, Hossain, Mohammed Akhter, Lin, Feng, Pinheiro-Junior, Ernesto L, Peigneur, Steve, Wai, Dorothy C C, Delaine, Carlie, Blyth, Andrew J, Forbes, Briony E, Tytgat, Jan, Wade, John D, Norton, Raymond S · 2021 · Biomolecules · DOI
Full title: Identification, Synthesis, Conformation and Activity of an Insulin-like Peptide from a Sea Anemone.
Authors: Mitchell, Michela L, Hossain, Mohammed Akhter, Lin, Feng, Pinheiro-Junior, Ernesto L, Peigneur, Steve, Wai, Dorothy C C, Delaine, Carlie, Blyth, Andrew J, Forbes, Briony E, Tytgat, Jan, Wade, John D, Norton, Raymond S
PaperDevelopment of a Novel Covalently Bonded Conjugate of Caprylic Acid Tripeptide (Isoleucine-Leucine-Aspartic Acid) for Wound-Compatible and Injectable Hydrogel to Accelerate Healing.
Baravkar, Sachin B, Lu, Yan, Masoud, Abdul-Razak, Zhao, Qi, He, Jibao, Hong, Song · 2024 · Biomolecules · DOI
Full title: Development of a Novel Covalently Bonded Conjugate of Caprylic Acid Tripeptide (Isoleucine-Leucine-Aspartic Acid) for Wound-Compatible and Injectable Hydrogel to Accelerate Healing.
PaperN-Terminally Lipidated Sialorphin Analogs—Synthesis, Molecular Modeling, In Vitro Effect on Enkephalins Degradation by NEP and Treatment of Intestinal Inflammation in Mice
Sobocińska, Małgorzata, Fichna, Jakub, Giełdoń, Artur, Skowron, Piotr M., Kamysz, Elżbieta · 2022 · International Journal of Molecular Sciences · DOI
Full title: N-Terminally Lipidated Sialorphin Analogs—Synthesis, Molecular Modeling, In Vitro Effect on Enkephalins Degradation by NEP and Treatment of Intestinal Inflammation in Mice
Authors: Sobocińska, Małgorzata, Fichna, Jakub, Giełdoń, Artur, Skowron, Piotr M., Kamysz, Elżbieta
Year: 2022
Venue: International Journal of Molecular Sciences
PaperSolid-Phase Synthesis Approaches and U-Rich RNA-Binding Activity of Homotrimer Nucleopeptide Containing Adenine Linked to L-azidohomoalanine Side Chain via 1,4-Linked-1,2,3-Triazole.
Mucha, Piotr, Pieszko, Małgorzata, Bylińska, Irena, Wiczk, Wiesław, Ruczyński, Jarosław, Rekowski, Piotr · 2025 · International journal of molecular sciences · DOI
Full title: Solid-Phase Synthesis Approaches and U-Rich RNA-Binding Activity of Homotrimer Nucleopeptide Containing Adenine Linked to L-azidohomoalanine Side Chain via 1,4-Linked-1,2,3-Triazole.
PaperTotal Linear Chemical Synthesis of LC3A and LC3B.
Huppelschoten, Yara, Buchardt, Jens, Nielsen, Thomas Eiland, van der Heden van Noort, Gerbrand J · 2023 · Methods in molecular biology (Clifton, N.J.) · DOI
Full title: Total Linear Chemical Synthesis of LC3A and LC3B.
Authors: Huppelschoten, Yara, Buchardt, Jens, Nielsen, Thomas Eiland, van der Heden van Noort, Gerbrand J
Year: 2023
Venue: Methods in molecular biology (Clifton, N.J.)
PaperImproved Handling of Peptide Segments Using Side Chain-Based "Helping Hand" Solubilizing Tools.
Jacobsen, Michael T, Spaltenstein, Paul, Giesler, Riley J, Chou, Danny Hung-Chieh, Kay, Michael S · 2022 · Methods in molecular biology (Clifton, N.J.) · DOI
Full title: Improved Handling of Peptide Segments Using Side Chain-Based "Helping Hand" Solubilizing Tools.
Authors: Jacobsen, Michael T, Spaltenstein, Paul, Giesler, Riley J, Chou, Danny Hung-Chieh, Kay, Michael S
Year: 2022
Venue: Methods in molecular biology (Clifton, N.J.)
PaperMicrowave-Assisted Synthesis of Antimicrobial Peptides.
Ramesh, Suhas, de la Torre, Beatriz G, Albericio, Fernando, Kruger, Hendrik G, Govender, Thavendran · 2017 · Methods in molecular biology (Clifton, N.J.) · DOI
Full title: Microwave-Assisted Synthesis of Antimicrobial Peptides.
Authors: Ramesh, Suhas, de la Torre, Beatriz G, Albericio, Fernando, Kruger, Hendrik G, Govender, Thavendran
Year: 2017
Venue: Methods in molecular biology (Clifton, N.J.)
PaperFacile Synthetic Access to Glycopeptide Antibiotic Precursor Peptides for the Investigation of Cytochrome P450 Action in Glycopeptide Antibiotic Biosynthesis.
Brieke, Clara, Kratzig, Veronika, Peschke, Madeleine, Cryle, Max J · 2016 · Methods in molecular biology (Clifton, N.J.) · DOI
Full title: Facile Synthetic Access to Glycopeptide Antibiotic Precursor Peptides for the Investigation of Cytochrome P450 Action in Glycopeptide Antibiotic Biosynthesis.
Authors: Brieke, Clara, Kratzig, Veronika, Peschke, Madeleine, Cryle, Max J
Year: 2016
Venue: Methods in molecular biology (Clifton, N.J.)
PaperSolid-phase peptide synthesis (SPPS), C-terminal vs. side-chain anchoring: a reality or a myth.
Cherkupally, Prabhakar, Acosta, Gerardo A, Ramesh, Suhas, De la Torre, Beatriz G, Govender, Thavendran, Kruger, Hendrik G, Albericio, Fernando · 2014 · Amino acids · DOI
Full title: Solid-phase peptide synthesis (SPPS), C-terminal vs. side-chain anchoring: a reality or a myth.
Authors: Cherkupally, Prabhakar, Acosta, Gerardo A, Ramesh, Suhas, De la Torre, Beatriz G, Govender, Thavendran, Kruger, Hendrik G, Albericio, Fernando
PaperSynthesis, characterization, conformational analysis of a cyclic conjugated octreotate peptide and biological evaluation of (99m)Tc-HYNIC-His(3)-Octreotate as novel tracer for the imaging of somatostatin receptor-positive tumors.
Full title: Synthesis, characterization, conformational analysis of a cyclic conjugated octreotate peptide and biological evaluation of (99m)Tc-HYNIC-His(3)-Octreotate as novel tracer for the imaging of somatostatin receptor-positive tumors.
Full title: Thirteen decades of peptide synthesis: key developments in solid phase peptide synthesis and amide bond formation utilized in peptide ligation.
PaperTo Rink or Not to Rink Amide Link, that is the Question to Address for More Economical and Environmentally Sound Solid-Phase Peptide Synthesis
T. Kassem, David Sabatino, X. Jia, X. X. Zhu, W. Lubell · 2009 · International Journal of Peptide Research and Therapeutics · DOI
Full title: To Rink or Not to Rink Amide Link, that is the Question to Address for More Economical and Environmentally Sound Solid-Phase Peptide Synthesis
Authors: T. Kassem, David Sabatino, X. Jia, X. X. Zhu, W. Lubell
Year: 2009
Venue: International Journal of Peptide Research and Therapeutics
PaperTc-99m and Fluorescence-Labeled Anti-Flt1 Peptide as a Multimodal Tumor Imaging Agent Targeting Vascular Endothelial Growth Factor-Receptor 1.
Kim, Myoung Hyoun, Kim, Seul-Gi, Kim, Dae-Weung · 2018 · Nuclear medicine and molecular imaging · DOI
Full title: Tc-99m and Fluorescence-Labeled Anti-Flt1 Peptide as a Multimodal Tumor Imaging Agent Targeting Vascular Endothelial Growth Factor-Receptor 1.
Authors: Kim, Myoung Hyoun, Kim, Seul-Gi, Kim, Dae-Weung
PaperAnthranilamide and nitrotyrosine as a donor-acceptor pair in internally quenched fluorescent substrates for endopeptidases: multicolumn peptide synthesis of enzyme substrates for subtilisin Carlsberg and pepsin.
Meldal, M, Breddam, K · 1991 · Analytical biochemistry · DOI
Full title: Anthranilamide and nitrotyrosine as a donor-acceptor pair in internally quenched fluorescent substrates for endopeptidases: multicolumn peptide synthesis of enzyme substrates for subtilisin Carlsberg and pepsin.
PaperTotal synthesis, structure elucidation and expanded bioactivity of icosalide A: effect of lipophilicity and ester to amide substitution on its bioactivity.
Full title: Total synthesis, structure elucidation and expanded bioactivity of icosalide A: effect of lipophilicity and ester to amide substitution on its bioactivity.
PaperGreen solvent mixture for ultrasound-assistant solid-phase peptide synthesis: a fast versatility method and its applications in flow and natural products synthesis
Jingyuan Liao, Renrong Zhang, X. Jia, Meiling Wang, Chaoyi Li, Juntao Wang, R. Tang, Junrong Huang, Hengzhi You, Fener Chen · 2024 · Green Chemistry · DOI
Full title: Green solvent mixture for ultrasound-assistant solid-phase peptide synthesis: a fast versatility method and its applications in flow and natural products synthesis
PaperRetrofitting HPLC Hardware for Affordable and Accessible Flow-Based Peptide Synthesis
Andrew M. White, Darcy Williamson, Caitlin L. Gare, Flynn C. Attard, Abby Kidston, Lara R. Malins · 2025 · Australian journal of chemistry (Print) · DOI
Full title: Retrofitting HPLC Hardware for Affordable and Accessible Flow-Based Peptide Synthesis
Authors: Andrew M. White, Darcy Williamson, Caitlin L. Gare, Flynn C. Attard, Abby Kidston, Lara R. Malins
PaperTick saliva protein Evasin-3 modulates chemotaxis by disrupting CXCL8 interactions with glycosaminoglycans and CXCR2
S. S. Denisov, J. H. Ippel, A. Heinzmann, R. Koenen, A. Ortega-Gómez, O. Soehnlein, T. Hackeng, I. Dijkgraaf · 2019 · Journal of Biological Chemistry · DOI
Full title: Tick saliva protein Evasin-3 modulates chemotaxis by disrupting CXCL8 interactions with glycosaminoglycans and CXCR2
Authors: S. S. Denisov, J. H. Ippel, A. Heinzmann, R. Koenen, A. Ortega-Gómez, O. Soehnlein, T. Hackeng, I. Dijkgraaf
PaperComputational-aided design: minimal peptide sequence to block dengue virus transmission into cells.
Arumugam, Aathe Cangaree, Agharbaoui, Fatima Ezzahra, Khazali, Ahmad Suhail, Yusof, Rohana, Abd Rahman, Noorsaadah, Ahmad Fuaad, Abdullah Al Hadi · 2022 · Journal of biomolecular structure & dynamics · DOI
Full title: Computational-aided design: minimal peptide sequence to block dengue virus transmission into cells.
Authors: Arumugam, Aathe Cangaree, Agharbaoui, Fatima Ezzahra, Khazali, Ahmad Suhail, Yusof, Rohana, Abd Rahman, Noorsaadah, Ahmad Fuaad, Abdullah Al Hadi
Year: 2022
Venue: Journal of biomolecular structure & dynamics
PaperProtein chemical synthesis by serine and threonine ligation.
Zhang, Yinfeng, Xu, Ci, Lam, Hiu Yung, Lee, Chi Lung, Li, Xuechen · 2013 · Proceedings of the National Academy of Sciences of the United States of America · DOI
Full title: Protein chemical synthesis by serine and threonine ligation.
PaperSolid-phase peptide synthesis using mild base cleavage of N alpha-fluorenylmethyloxycarbonylamino acids, exemplified by a synthesis of dihydrosomatostatin.
Chang, C D, Meienhofer, J · 1978 · International journal of peptide and protein research · DOI
Full title: Solid-phase peptide synthesis using mild base cleavage of N alpha-fluorenylmethyloxycarbonylamino acids, exemplified by a synthesis of dihydrosomatostatin.
Authors: Chang, C D, Meienhofer, J
Year: 1978
Venue: International journal of peptide and protein research
PaperPeptides as potential virus inhibitors. Synthesis and bioassay of five respiratory syncytial virus peptide analogs with antimeasles activity.
T. Lobl, H. Renis, R. Epand, L. Maggiora, M. Wathen · 2009 · International journal of peptide & protein research · DOI
Full title: Peptides as potential virus inhibitors. Synthesis and bioassay of five respiratory syncytial virus peptide analogs with antimeasles activity.
Authors: T. Lobl, H. Renis, R. Epand, L. Maggiora, M. Wathen
Year: 2009
Venue: International journal of peptide & protein research
PaperEfficient solid phase synthesis of mixed Thr(P)-, Ser(P)- and Tyr(P)-containing phosphopeptides by "global" "phosphite-triester" phosphorylation.
J. Perich · 2009 · International journal of peptide & protein research · DOI
Full title: Efficient solid phase synthesis of mixed Thr(P)-, Ser(P)- and Tyr(P)-containing phosphopeptides by "global" "phosphite-triester" phosphorylation.
Authors: J. Perich
Year: 2009
Venue: International journal of peptide & protein research
PaperPressure monitoring of continuous-flow solid-phase peptide synthesis.
Baru, M B, Mustaeva, L G, Vagenina, I V, Gorbunova, E Y, Cherskii, V V · 2001 · The journal of peptide research : official journal of the American Peptide Society · DOI
Full title: Pressure monitoring of continuous-flow solid-phase peptide synthesis.
Authors: Baru, M B, Mustaeva, L G, Vagenina, I V, Gorbunova, E Y, Cherskii, V V
Year: 2001
Venue: The journal of peptide research : official journal of the American Peptide Society
PaperPreparation of a multiple antigen glycopeptide (MAG) carrying the Tn antigen. A possible approach to a synthetic carbohydrate vaccine.
Bay, S, Lo-Man, R, Osinaga, E, Nakada, H, Leclerc, C, Cantacuzène, D · 1997 · The journal of peptide research : official journal of the American Peptide Society · DOI
Full title: Preparation of a multiple antigen glycopeptide (MAG) carrying the Tn antigen. A possible approach to a synthetic carbohydrate vaccine.
Authors: Bay, S, Lo-Man, R, Osinaga, E, Nakada, H, Leclerc, C, Cantacuzène, D
Year: 1997
Venue: The journal of peptide research : official journal of the American Peptide Society
PaperDesign, synthesis, tandem mass spectrometric sequencing and biological activity of NGF mimetics.
Estenne-Bouhtou, G, Kullander, K, Karlsson, M, Ebendal, T, Hacksell, U, Luthman, K · 1996 · International journal of peptide and protein research · DOI
Full title: Design, synthesis, tandem mass spectrometric sequencing and biological activity of NGF mimetics.
Authors: Estenne-Bouhtou, G, Kullander, K, Karlsson, M, Ebendal, T, Hacksell, U, Luthman, K
Year: 1996
Venue: International journal of peptide and protein research
Katritzky, Alan R, Khashab, Niveen M, Yoshioka, Megumi, Haase, Danniebelle N, Wilson, Krista R, Johnson, Jodie V, Chung, Alfred, Haskell-Luevano, Carrie · 2007 · Chemical biology & drug design · DOI
Full title: Microwave-assisted solid-phase peptide synthesis utilizing N-Fmoc-protected (alpha-aminoacyl)benzotriazoles.
Authors: Katritzky, Alan R, Khashab, Niveen M, Yoshioka, Megumi, Haase, Danniebelle N, Wilson, Krista R, Johnson, Jodie V, Chung, Alfred, Haskell-Luevano, Carrie
PaperSonophoresis-mediated permeation and retention of peptide dendrimers across human epidermis.
Mutalik, Srinivas, Nayak, Usha Y, Kalra, Rohit, Kumar, Aravind, Kulkarni, Raghavendra V, Parekh, Harendra S · 2012 · Skin research and technology : official journal of International Society for Bioengineering and the Skin (ISBS) [and] International Society for Digital Imaging of Skin (ISDIS) [and] International Society for Skin Imaging (ISSI) · DOI
Full title: Sonophoresis-mediated permeation and retention of peptide dendrimers across human epidermis.
Authors: Mutalik, Srinivas, Nayak, Usha Y, Kalra, Rohit, Kumar, Aravind, Kulkarni, Raghavendra V, Parekh, Harendra S
Year: 2012
Venue: Skin research and technology : official journal of International Society for Bioengineering and the Skin (ISBS) [and] International Society for Digital Imaging of Skin (ISDIS) [and] International Society for Skin Imaging (ISSI)
PaperIn Vivo Molecular Imaging of Somatostatin Receptors in Pancreatic Islet Cells and Neuroendocrine Tumors by Miniaturized Confocal Laser-Scanning Fluorescence Microscopy
Fottner, C., Mettler, Esther, Goetz, M., Schirrmacher, E., Anlauf, M., Strand, D., Schirrmacher, R., Klöppel, G., Delaney, P., Schreckenberger, M., Galle, P. R., Neurath, M. F., Kiesslich, R., Weber, M. M. · 2010 · The Journal of Clinical Endocrinology & Metabolism · DOI
Full title: In Vivo Molecular Imaging of Somatostatin Receptors in Pancreatic Islet Cells and Neuroendocrine Tumors by Miniaturized Confocal Laser-Scanning Fluorescence Microscopy
Authors: Fottner, C., Mettler, Esther, Goetz, M., Schirrmacher, E., Anlauf, M., Strand, D., Schirrmacher, R., Klöppel, G., Delaney, P., Schreckenberger, M., Galle, P. R., Neurath, M. F., Kiesslich, R., Weber, M. M.
Year: 2010
Venue: The Journal of Clinical Endocrinology & Metabolism
PaperIn vivo molecular imaging of somatostatin receptors in pancreatic islet cells and neuroendocrine tumors by miniaturized confocal laser-scanning fluorescence microscopy.
Fottner, C, Mettler, E, Goetz, M, Schirrmacher, E, Anlauf, M, Strand, D, Schirrmacher, R, Klöppel, G, Delaney, P, Schreckenberger, M, Galle, P R, Neurath, M F, Kiesslich, R, Weber, M M · 2010 · Endocrinology · DOI
Full title: In vivo molecular imaging of somatostatin receptors in pancreatic islet cells and neuroendocrine tumors by miniaturized confocal laser-scanning fluorescence microscopy.
Authors: Fottner, C, Mettler, E, Goetz, M, Schirrmacher, E, Anlauf, M, Strand, D, Schirrmacher, R, Klöppel, G, Delaney, P, Schreckenberger, M, Galle, P R, Neurath, M F, Kiesslich, R, Weber, M M
PaperAbstract 4106: A novel synthetic long peptide vaccine composition targeting multiple PD-L1 T-cell epitopes exhibits anti-tumor efficacy in a syngeneic mouse colorectal cancer model
Kenneth Nansheng Lin, Melvin Toh · 2024 · Cancer Research · DOI
Full title: Abstract 4106: A novel synthetic long peptide vaccine composition targeting multiple PD-L1 T-cell epitopes exhibits anti-tumor efficacy in a syngeneic mouse colorectal cancer model
PaperIn Vivo Molecular Imaging of Somatostatin Receptors in Pancreatic Islet Cells and Neuroendocrine Tumors by Miniaturized Confocal Laser-Scanning Fluorescence Microscopy
Fottner, Christian, Mettler, E., Goetz, Martin, Schirrmacher, E., Anlauf, M., Strand, D., Schirrmacher, R., Klöppel, G., Delaney, P., Schreckenberger, M., Galle, P. R., Neurath, M. F., Kießlich, Ralf, Weber, M. M. · 2010 · Endocrine Reviews · DOI
Full title: In Vivo Molecular Imaging of Somatostatin Receptors in Pancreatic Islet Cells and Neuroendocrine Tumors by Miniaturized Confocal Laser-Scanning Fluorescence Microscopy
Authors: Fottner, Christian, Mettler, E., Goetz, Martin, Schirrmacher, E., Anlauf, M., Strand, D., Schirrmacher, R., Klöppel, G., Delaney, P., Schreckenberger, M., Galle, P. R., Neurath, M. F., Kießlich, Ralf, Weber, M. M.
PaperEnantioselective Synthesis of (2S,3S)‐epi‐Oxetin and Its Incorporation into Conformationally Constrained Pyrrolidinyl PNA with an Oxetane Backbone
Pattarakiat Seankongsuk, Viwat Vchirawongkwin, R. Bates, Panuwat Padungros, T. Vilaivan · 2017 · Asian Journal of Organic Chemistry · DOI
Full title: Enantioselective Synthesis of (2S,3S)‐epi‐Oxetin and Its Incorporation into Conformationally Constrained Pyrrolidinyl PNA with an Oxetane Backbone
Authors: Pattarakiat Seankongsuk, Viwat Vchirawongkwin, R. Bates, Panuwat Padungros, T. Vilaivan
PaperSynthesis, characterization, and evaluation of PS-PPDC resin: a novel flexible cross-linked polymeric support for solid-phase organic synthesis.
Siyad, M A; Vinod Kumar, G S · 2012 · Biopolymers · DOI
Full title: Synthesis, characterization, and evaluation of PS-PPDC resin: a novel flexible cross-linked polymeric support for solid-phase organic synthesis.
PaperChemical synthesis of a polypeptide backbone derived from the primary sequence of the cancer protein NY-ESO-1 enabled by kinetically controlled ligation and pseudoprolines.
Harris, Paul W R, Brimble, Margaret A · 2015 · Biopolymers · DOI
Full title: Chemical synthesis of a polypeptide backbone derived from the primary sequence of the cancer protein NY-ESO-1 enabled by kinetically controlled ligation and pseudoprolines.
PaperDesigning Chimeric Peptides: A Powerful Tool for Enhancing Antibacterial Activity
H. M. Pineda-Castañeda, Kevin Andrey Huertas‐Ortiz, A. Leal‐Castro, Yerly Vargas‐Casanova, C. Parra‐Giraldo, J. García‐Castañeda, Z. Rivera-Monroy · 2020 · Chemistry and Biodiversity · DOI
Full title: Designing Chimeric Peptides: A Powerful Tool for Enhancing Antibacterial Activity
Authors: H. M. Pineda-Castañeda, Kevin Andrey Huertas‐Ortiz, A. Leal‐Castro, Yerly Vargas‐Casanova, C. Parra‐Giraldo, J. García‐Castañeda, Z. Rivera-Monroy
PaperSynthesis of a 6,6-spiroketal amino acid and its incorporation into a peptide turn sequence using solid-phase peptide synthesis.
Kueh, Jui Thiang Brian, Choi, Ka Wai, Williams, Geoffrey M, Moehle, Kerstin, Bacsa, Bernadett, Robinson, John A, Brimble, Margaret A · 2013 · Chemistry (Weinheim an der Bergstrasse, Germany) · DOI
Full title: Synthesis of a 6,6-spiroketal amino acid and its incorporation into a peptide turn sequence using solid-phase peptide synthesis.
Authors: Kueh, Jui Thiang Brian, Choi, Ka Wai, Williams, Geoffrey M, Moehle, Kerstin, Bacsa, Bernadett, Robinson, John A, Brimble, Margaret A
Year: 2013
Venue: Chemistry (Weinheim an der Bergstrasse, Germany)
PaperSynthesis of Peptides Containing a Combination of Free and 2-trans-Cyclooctene Carbamate Protected Lysine Residues.
Doelman, W, Ligthart, N A M, van de Plassche, M A T, de Geus, M A R, Reinalda, L, Isendoorn, M M E, Filippov, D V, van Kasteren, S I · 2024 · Chembiochem : a European journal of chemical biology · DOI
Full title: Synthesis of Peptides Containing a Combination of Free and 2-trans-Cyclooctene Carbamate Protected Lysine Residues.
Authors: Doelman, W, Ligthart, N A M, van de Plassche, M A T, de Geus, M A R, Reinalda, L, Isendoorn, M M E, Filippov, D V, van Kasteren, S I
Year: 2024
Venue: Chembiochem : a European journal of chemical biology
PaperRapid total synthesis of cyclic lipodepsipeptides as a premise to investigate their self-assembly and biological activity.
De Vleeschouwer, Matthias, Sinnaeve, Davy, Van den Begin, Jos, Coenye, Tom, Martins, José C, Madder, Annemieke · 2014 · Chemistry (Weinheim an der Bergstrasse, Germany) · DOI
Full title: Rapid total synthesis of cyclic lipodepsipeptides as a premise to investigate their self-assembly and biological activity.
Authors: De Vleeschouwer, Matthias, Sinnaeve, Davy, Van den Begin, Jos, Coenye, Tom, Martins, José C, Madder, Annemieke
Year: 2014
Venue: Chemistry (Weinheim an der Bergstrasse, Germany)
PaperAn Efficient, Site‐Selective and Spontaneous Peptide Macrocyclisation During in vitro Translation
Liu, Minglong, Yoshisada, Ryoji, Amedi, Avand, Hopstaken, Antonius J. P., Pascha, Mirte N., Haan, Cornelis A. M. de, Geerke, Daan P., Poole, David A., Jongkees, Seino A. K. · 2022 · Chemistry - A European Journal · DOI
Full title: An Efficient, Site‐Selective and Spontaneous Peptide Macrocyclisation During in vitro Translation
Authors: Liu, Minglong, Yoshisada, Ryoji, Amedi, Avand, Hopstaken, Antonius J. P., Pascha, Mirte N., Haan, Cornelis A. M. de, Geerke, Daan P., Poole, David A., Jongkees, Seino A. K.
PaperAn Optimized Protocol for the Synthesis of Peptides Containing trans-Cyclooctene and Bicyclononyne Dienophiles as Useful Multifunctional Bioorthogonal Probes.
La-Venia, Agustina, Dzijak, Rastislav, Rampmaier, Robert, Vrabel, Milan · 2021 · Chemistry (Weinheim an der Bergstrasse, Germany) · DOI
Full title: An Optimized Protocol for the Synthesis of Peptides Containing trans-Cyclooctene and Bicyclononyne Dienophiles as Useful Multifunctional Bioorthogonal Probes.
Authors: La-Venia, Agustina, Dzijak, Rastislav, Rampmaier, Robert, Vrabel, Milan
Year: 2021
Venue: Chemistry (Weinheim an der Bergstrasse, Germany)
PaperSynthesis of BODIPY-Labeled Cholesterylated Glycopeptides by Tandem Click Chemistry for Glycocalyxification of Giant Unilamellar Vesicles (GUVs).
Stuhr-Hansen, Nicolai, Vagianou, Charikleia-Despoina, Blixt, Ola · 2017 · Chemistry (Weinheim an der Bergstrasse, Germany) · DOI
Full title: Synthesis of BODIPY-Labeled Cholesterylated Glycopeptides by Tandem Click Chemistry for Glycocalyxification of Giant Unilamellar Vesicles (GUVs).
Authors: Stuhr-Hansen, Nicolai, Vagianou, Charikleia-Despoina, Blixt, Ola
Year: 2017
Venue: Chemistry (Weinheim an der Bergstrasse, Germany)
PaperSynthesis and Evaluation of Non-Hydrolyzable Phospho-Lysine Peptide Mimics.
Hauser, Anett, Poulou, Eleftheria, Müller, Fabian, Schmieder, Peter, Hackenberger, Christian P R · 2021 · Chemistry (Weinheim an der Bergstrasse, Germany) · DOI
Full title: Synthesis and Evaluation of Non-Hydrolyzable Phospho-Lysine Peptide Mimics.
Authors: Hauser, Anett, Poulou, Eleftheria, Müller, Fabian, Schmieder, Peter, Hackenberger, Christian P R
Year: 2021
Venue: Chemistry (Weinheim an der Bergstrasse, Germany)
PaperRapid Chemical Synthesis of Serine Protease Inhibitor Kazal-type 13 (SPINK13) Glycoform by a Combined Method with Glycan Insertion Strategy and Fast-Flow Fmoc SPPS.
Nomura, Kota, Okamoto, Ryo, Maki, Yuta, Hayashibara, Ayumu, Takao, Toshifumi, Fukuoka, Tomoya, Miyoshi, Eiji, Pentelute, Bradley L, Kajihara, Yasuhiro · 2023 · Chemistry (Weinheim an der Bergstrasse, Germany) · DOI
Full title: Rapid Chemical Synthesis of Serine Protease Inhibitor Kazal-type 13 (SPINK13) Glycoform by a Combined Method with Glycan Insertion Strategy and Fast-Flow Fmoc SPPS.
PaperSynthesis of Asparagine Derivatives Harboring a Lewis X Type DC-SIGN Ligand and Evaluation of their Impact on Immunomodulation in Multiple Sclerosis.
Doelman, Ward, Marqvorsen, Mikkel H S, Chiodo, Fabrizio, Bruijns, Sven C M, van der Marel, Gijsbert A, van Kooyk, Yvette, van Kasteren, Sander I, Araman, Can · 2021 · Chemistry (Weinheim an der Bergstrasse, Germany) · DOI
Full title: Synthesis of Asparagine Derivatives Harboring a Lewis X Type DC-SIGN Ligand and Evaluation of their Impact on Immunomodulation in Multiple Sclerosis.
Authors: Doelman, Ward, Marqvorsen, Mikkel H S, Chiodo, Fabrizio, Bruijns, Sven C M, van der Marel, Gijsbert A, van Kooyk, Yvette, van Kasteren, Sander I, Araman, Can
Year: 2021
Venue: Chemistry (Weinheim an der Bergstrasse, Germany)
PaperExploring the Chemical Properties and Medicinal Applications of Tetramethylthiocycloheptyne Sulfoximine Used in Strain-Promoted Azide–Alkyne Cycloaddition Reactions
Timmers, Matt; Kipper, Andi; Frey, Raphael et al. · 2023 · Pharmaceuticals · DOI
Full title: Exploring the Chemical Properties and Medicinal Applications of Tetramethylthiocycloheptyne Sulfoximine Used in Strain-Promoted Azide–Alkyne Cycloaddition Reactions
Full title: Chemical Synthesis Of Peptides And Peptide Thioesters
Authors: Sharma, Indrajeet
Year: 2011
Venue: DigitalCommons - WayneState (Wayne State University)
PaperPoly(Arginine) Derived Cancer-Targeting Peptides for the Development of a Cancer-Targeted Gene Therapy Approach in HepG2 Liver Cancer Cells
Joseph, Stesha C. · 2014 · Seton Hall University eRepository (Seton Hall University)
Full title: Poly(Arginine) Derived Cancer-Targeting Peptides for the Development of a Cancer-Targeted Gene Therapy Approach in HepG2 Liver Cancer Cells
Authors: Joseph, Stesha C.
Year: 2014
Venue: Seton Hall University eRepository (Seton Hall University)
PaperVersatility Of N-Peptidyl And N-Glycopeptidyl Nitroindolines For The Formation Of Peptide/Glycopeptide Acids, Amides, And Thioesters
Barrera, Luis A. · 2015 · DigitalCommons@UTEP (The University of Texas at El Paso)
Full title: Versatility Of N-Peptidyl And N-Glycopeptidyl Nitroindolines For The Formation Of Peptide/Glycopeptide Acids, Amides, And Thioesters
Authors: Barrera, Luis A.
Year: 2015
Venue: DigitalCommons@UTEP (The University of Texas at El Paso)
PaperLuminescent Bimetallic Ir III /Au I Peptide Bioconjugates as Potential Theranostic Agents
Luengo, Andrés; Marzo, Isabel; Reback, Matthew L. et al. · 2020 · Chemistry - A European Journal · DOI
Full title: Luminescent Bimetallic Ir III /Au I Peptide Bioconjugates as Potential Theranostic Agents
Authors: Luengo, Andrés; Marzo, Isabel; Reback, Matthew L.; Daubit, Isabelle Marie; Fernández‐Moreira, Vanesa; Metzler‐Nolte, Nils; Gimeno, M. Concepción
PaperSolid-Phase Synthesis of Peptide Hydrazides: Moving Toward Green Chemistry.
Leko, Maria; Filippova, Polina; Rustler, Karin et al. · 2025 · Journal of peptide science : an official publication of the European Peptide Society · DOI
Full title: Solid-Phase Synthesis of Peptide Hydrazides: Moving Toward Green Chemistry.
PaperAqueous microwave-assisted solid-phase peptide synthesis using Fmoc strategy. III: racemization studies and water-based synthesis of histidine-containing peptides.
Hojo, Keiko; Shinozaki, Natsuki; Hidaka, Koushi et al. · 2014 · Amino acids · DOI
Full title: Aqueous microwave-assisted solid-phase peptide synthesis using Fmoc strategy. III: racemization studies and water-based synthesis of histidine-containing peptides.
Authors: Hojo, Keiko; Shinozaki, Natsuki; Hidaka, Koushi; Tsuda, Yuko; Fukumori, Yoshinobu; Ichikawa, Hideki; Wade, John D
PaperApplication of mechanochemistry to green, scalable, and continuous manufacturing of pharmaceutically relevant peptides by twin-screw extrusion.
Daurio, Dominick; Jacobsen, Casey S; Nagapudi, Karthik et al. · 2025 · Journal of pharmaceutical sciences · DOI
Full title: Application of mechanochemistry to green, scalable, and continuous manufacturing of pharmaceutically relevant peptides by twin-screw extrusion.
Authors: Daurio, Dominick; Jacobsen, Casey S; Nagapudi, Karthik; Saw, Robert; Silva Elipe, Maria Victoria; Thiel, Oliver; Balgley, Renata; Chamarthy, Sai Prasanth; Alvarez-Nunez, Fernando
PaperFmoc-Removal with Pyrrolidine Expands the Available Solvent Space in Green Solid-Phase Peptide Synthesis
Egelund, Peter H. G.; Jadhav, Sandip V.; Martin, Vincent et al. · 2021 · ACS Sustainable Chemistry & Engineering · DOI
Full title: Fmoc-Removal with Pyrrolidine Expands the Available Solvent Space in Green Solid-Phase Peptide Synthesis
Authors: Egelund, Peter H. G.; Jadhav, Sandip V.; Martin, Vincent; Johansson, Henrik; Richner, Franziska; Quement, Sebastian T. Le; Dettner, Frank; Lechner, Carolin C.; Schoenleber, Ralph O.; Pedersen, Daniel Sejer
PaperMild, orthogonal solid-phase peptide synthesis: use of N alpha-dithiasuccinoyl (Dts) amino acids and N-(iso-propyldithio)carbonylproline, together with p-alkoxybenzyl ester anchoring linkages.
Albericio, F; Barany, G · 1987 · International journal of peptide and protein research · DOI
Full title: Mild, orthogonal solid-phase peptide synthesis: use of N alpha-dithiasuccinoyl (Dts) amino acids and N-(iso-propyldithio)carbonylproline, together with p-alkoxybenzyl ester anchoring linkages.
Authors: Albericio, F; Barany, G
Year: 1987
Venue: International journal of peptide and protein research
PaperAqueous microwave-assisted solid-phase peptide synthesis using fmoc strategy. II. Racemization studies and water based synthesis of cysteine-containing peptides.
Hojo, Keiko; Shinozaki, Natsuki; Hara, Asaki et al. · 2013 · Protein and peptide letters · DOI
Full title: Aqueous microwave-assisted solid-phase peptide synthesis using fmoc strategy. II. Racemization studies and water based synthesis of cysteine-containing peptides.
ThesisThe self-assembly of redox active peptides: Synthesis and electrochemical capacitive behavior
Piccoli, Julia P. [UNESP]; Santos, Adriano [UNESP]; Santos-Filho, Norival A. [UNESP] et al. · 2018 · Universidade Estadual Paulista (UNESP) · DOI
Full title: The self-assembly of redox active peptides: Synthesis and electrochemical capacitive behavior
Authors: Piccoli, Julia P. [UNESP]; Santos, Adriano [UNESP]; Santos-Filho, Norival A. [UNESP]; Lorenzón, Esteban N. [UNESP]; Cilli, Eduardo M. [UNESP]; Bueno, Paulo R. [UNESP]
ThesisComparative investigation of the cleavage step in the synthesis of model peptide resins: Implications for N-alpha-9-fluorenylmethyloxycarbonyl-solid phase peptide synthesis
Jubilut, Guita Nicolaewsky; Cilli, Eduardo Maffud [UNESP]; Crusca, Edson et al. · 2014 · Universidade Estadual Paulista (UNESP) · DOI
Full title: Comparative investigation of the cleavage step in the synthesis of model peptide resins: Implications for N-alpha-9-fluorenylmethyloxycarbonyl-solid phase peptide synthesis
ThesisCorrelation between the mobility of spin-labeled peptide chains and resin solvation: An approach to optimize the synthesis of aggregating sequences
Cilli, Eduardo Maffud [UNESP]; Marchetto, Reinaldo [UNESP]; Schreier, S. et al. · 2014 · Universidade Estadual Paulista (UNESP) · DOI
Full title: Correlation between the mobility of spin-labeled peptide chains and resin solvation: An approach to optimize the synthesis of aggregating sequences
Authors: Cilli, Eduardo Maffud [UNESP]; Marchetto, Reinaldo [UNESP]; Schreier, S.; Nakaie, C. R.
ThesisOne-pot Ligation Strategy for Atypical Ubiquitin Chains Synthesis by Using the Trifluoroacetamidomethyl-protected Isopeptide-linked Ub (Tfacm-isoUb) Unit
Si, Yan-Yan; Liang, Lu-Jun; Tang, Shan et al. · 2018 · Hong Kong University of Science and Technology (HKUST) · DOI
Full title: One-pot Ligation Strategy for Atypical Ubiquitin Chains Synthesis by Using the Trifluoroacetamidomethyl-protected Isopeptide-linked Ub (Tfacm-isoUb) Unit
ThesisGreening the solid-phase peptide synthesis process. 2-MeTHF for the incorporation of the first amino acid and precipitation of peptides after global deprotection
Al Musaimi, Othman; Jad, Yahya E; Kumar, Ashish et al. · 2021 · Imperial College London · DOI
Full title: Greening the solid-phase peptide synthesis process. 2-MeTHF for the incorporation of the first amino acid and precipitation of peptides after global deprotection
Authors: Al Musaimi, Othman; Jad, Yahya E; Kumar, Ashish; El-Faham, Ayman; Collins, Jonathan M; Basso, Alessandra; de la Torre, Beatriz G; Albericio, Fernando
ThesisBypassing osmotic shock dilemma in a polystyrene resin using the green solvent cyclopentyl methyl Ether (CPME): a morphological perspective
Al Musaimi, Othman; El-Faham, Ayman; Almarhoon, Zainab et al. · 2022 · Imperial College London · DOI
Full title: Bypassing osmotic shock dilemma in a polystyrene resin using the green solvent cyclopentyl methyl Ether (CPME): a morphological perspective
Authors: Al Musaimi, Othman; El-Faham, Ayman; Almarhoon, Zainab; Basso, Alessandra; de la Torre, Beatriz G; Albericio, Fernando
ThesisSynthesis of cyclodextrin composites incorporating targeting and drug carrying capabilities : a thesis submitted in partial fulfilment of the requirements for the degree of Doctor of Philosophy in Chemistry, Massey University, Turitea Campus, Palmerston North, New Zealand
White, Rachel Jane · 2010 · Massey University · DOI
Full title: Synthesis of cyclodextrin composites incorporating targeting and drug carrying capabilities : a thesis submitted in partial fulfilment of the requirements for the degree of Doctor of Philosophy in Chemistry, Massey University, Turitea Campus, Palmerston North, New Zealand
ThesisSelective thiazoline peptide cyclisation compatible with mRNA display and efficient synthesis
Liu, Minglong; Morewood, Richard; Yoshisada, Ryoji et al. · 2023 · Utrecht University · DOI
Full title: Selective thiazoline peptide cyclisation compatible with mRNA display and efficient synthesis
Authors: Liu, Minglong; Morewood, Richard; Yoshisada, Ryoji; Pascha, Mirte N; Hopstaken, Antonius J P; Tarcoveanu, Eliza; Poole, David A; de Haan, Cornelis A M; Nitsche, Christoph; Jongkees, Seino A K
Scalable and Sustainable DMF-Free Solid-Phase Synthesis of Liraglutide by 1-Tert-Butyl-3-Ethylcarbodiimide-Mediated Couplings and Catch-and-Release Acylation and Purification Strategies
Pacini, Lorenzo, Muthyala, Manoj Kumar, Zitterbart, Robert, Marder, Oleg, Rovero, Paolo, Papini, Anna Maria · 2025
Full title: Scalable and Sustainable DMF-Free Solid-Phase Synthesis of Liraglutide by 1-Tert-Butyl-3-Ethylcarbodiimide-Mediated Couplings and Catch-and-Release Acylation and Purification Strategies
Authors: Pacini, Lorenzo, Muthyala, Manoj Kumar, Zitterbart, Robert, Marder, Oleg, Rovero, Paolo, Papini, Anna Maria
Stereoselective synthesis of Gly-Gly-type (E)-methylalkene and (Z)-chloroalkene dipeptide isosteres and their application to 14-mer RGG peptidomimetics.
Full title: Stereoselective synthesis of Gly-Gly-type (E)-methylalkene and (Z)-chloroalkene dipeptide isosteres and their application to 14-mer RGG peptidomimetics.
Solid Phase Synthesis of an Insect Pyrokinin Analog Incorporating an Imidazoline Ring as Isosteric Replacement of a <em>trans</em> Peptide Bond
Kaczmarek, Krzysztof; Pacholczyk‐Sienicka, Barbara; Albrecht, Łukasz et al. · 2021
Full title: Solid Phase Synthesis of an Insect Pyrokinin Analog Incorporating an Imidazoline Ring as Isosteric Replacement of a <em>trans</em> Peptide Bond
Authors: Kaczmarek, Krzysztof; Pacholczyk‐Sienicka, Barbara; Albrecht, Łukasz; Zabrocki, Janusz; Nachman, Ronald J.
Development of synthetic strategies towards libraries of heterocyclic and bicyclic inhibitors of Cdc25A & development of solid phase synthesis of cyclic peptides
Luo, Hao · 2015
Full title: Development of synthetic strategies towards libraries of heterocyclic and bicyclic inhibitors of Cdc25A & development of solid phase synthesis of cyclic peptides