PaperSuccessful development of a method for the incorporation of Fmoc-Arg(Pbf)-OH in solid-phase peptide synthesis using <i>N</i>-butylpyrrolidinone (NBP) as solvent
de la Torre, Beatriz G.; Kumar, Ashish; Alhassan, Mahama et al. · 2020 · Green Chemistry · DOI
Full title: Successful development of a method for the incorporation of Fmoc-Arg(Pbf)-OH in solid-phase peptide synthesis using <i>N</i>-butylpyrrolidinone (NBP) as solvent
Authors: de la Torre, Beatriz G.; Kumar, Ashish; Alhassan, Mahama; Bucher, Christoph; Albericio, Fernando; Lopez, John
PaperGreen solvents and Safe Reagents in SPPS taking advantage of induction heating and automation: synthesis and HPLC-free purification of difficult sequences
Pacini, L.; Muthyala, M.; Marder, O. et al. · 2024 · Proceedings of the 37th European Peptide Symposium · DOI
Full title: Green solvents and Safe Reagents in SPPS taking advantage of induction heating and automation: synthesis and HPLC-free purification of difficult sequences
Authors: Pacini, L.; Muthyala, M.; Marder, O.; Aguiar, L.; Zitterbart, R.; Rovero, P.; Papini, A.
Year: 2024
Venue: Proceedings of the 37th European Peptide Symposium
PaperHighlighting multicomponent reactions as an efficient and facile alternative route in the chemical synthesis of organic-based molecules: a tremendous growth in the past 5 years
Mohlala, Reagan Lehlogonolo; Rashamuse, Thompho Jason; Coyanis, Elena Mabel · 2024 · Frontiers in Chemistry · DOI
Full title: Highlighting multicomponent reactions as an efficient and facile alternative route in the chemical synthesis of organic-based molecules: a tremendous growth in the past 5 years
Authors: Mohlala, Reagan Lehlogonolo; Rashamuse, Thompho Jason; Coyanis, Elena Mabel
PaperGreen solvent mixture for ultrasound-assisted solid-phase peptide synthesis: a fast and versatile method and its applications in flow and natural product synthesis
Liao, Jingyuan; Zhang, Renrong; Jia, Xuelei et al. · 2024 · Green Chemistry · DOI
Full title: Green solvent mixture for ultrasound-assisted solid-phase peptide synthesis: a fast and versatile method and its applications in flow and natural product synthesis
PaperTotal Synthesis of Novel Antimicrobial β-Hairpin Capitellacin Via Rapid Flow-Based SPPS Assembly and Regioselective On-Resin Disulfide Cyclisation
Shepperson, Oscar A.; Hanna, Cameron C.; Brimble, Margaret A. et al. · 2022 · International Journal of Peptide Research and Therapeutics · DOI
Full title: Total Synthesis of Novel Antimicrobial β-Hairpin Capitellacin Via Rapid Flow-Based SPPS Assembly and Regioselective On-Resin Disulfide Cyclisation
Authors: Shepperson, Oscar A.; Hanna, Cameron C.; Brimble, Margaret A.; Harris, Paul W. R.; Cameron, Alan J.
Year: 2022
Venue: International Journal of Peptide Research and Therapeutics
PaperInvestigation of bioactive natural compounds for cardiovascular diseases and daqu fermentation, and the exploration of Beauveria bassiana as a biocontrol agent for the mountain pine beetle epidemic
Fernandez, Kleinberg Xiandrell · 2024 · University of Alberta Library · DOI
Full title: Investigation of bioactive natural compounds for cardiovascular diseases and daqu fermentation, and the exploration of Beauveria bassiana as a biocontrol agent for the mountain pine beetle epidemic
PaperDevelopment of synthetic strategies towards libraries of heterocyclic and bicyclic inhibitors of Cdc25A & development of solid phase synthesis of cyclic peptides
Luo, Hao · 2015 · Hannover : Gottfried Wilhelm Leibniz Universität Hannover · DOI
Full title: Development of synthetic strategies towards libraries of heterocyclic and bicyclic inhibitors of Cdc25A & development of solid phase synthesis of cyclic peptides
Authors: Luo, Hao
Year: 2015
Venue: Hannover : Gottfried Wilhelm Leibniz Universität Hannover
PaperScalable and Sustainable DMF-Free Solid-Phase Synthesis of Liraglutide by 1-Tert-Butyl-3-Ethylcarbodiimide-Mediated Couplings and Catch-and-Release Acylation and Purification Strategies
Pacini, Lorenzo; Muthyala, Manoj Kumar; Zitterbart, Robert et al. · 2025 · International Journal of Peptide Research and Therapeutics · DOI
Full title: Scalable and Sustainable DMF-Free Solid-Phase Synthesis of Liraglutide by 1-Tert-Butyl-3-Ethylcarbodiimide-Mediated Couplings and Catch-and-Release Acylation and Purification Strategies
Authors: Pacini, Lorenzo; Muthyala, Manoj Kumar; Zitterbart, Robert; Marder, Oleg; Rovero, Paolo; Papini, Anna Maria
Year: 2025
Venue: International Journal of Peptide Research and Therapeutics
PaperBypassing Osmotic Shock Dilemma in a Polystyrene Resin Using the Green Solvent Cyclopentyl methyl Ether (CPME): A Morphological Perspective
Al Musaimi, Othman; El-Faham, Ayman; Almarhoon, Zainab et al. · 2019 · Polymers · DOI
Full title: Bypassing Osmotic Shock Dilemma in a Polystyrene Resin Using the Green Solvent Cyclopentyl methyl Ether (CPME): A Morphological Perspective
Authors: Al Musaimi, Othman; El-Faham, Ayman; Almarhoon, Zainab; Basso, Alessandra; de la Torre, Beatriz G.; Albericio, Fernando
PaperEfficient generation of recombinant hydrazides for the production of scarce proteins and development of chemical probes for detecting protein sulfenylation
Ekanayake, Oshini · 2020 · University of Delaware · DOI
Full title: Efficient generation of recombinant hydrazides for the production of scarce proteins and development of chemical probes for detecting protein sulfenylation
PaperEfficient Synthesis of Peptides with 4-Methylpiperidine as Fmoc Removal Reagent by Solid Phase Synthesis
García Castañeda, Javier Eduardo; Vergel Galeano, Cristian Francisco; Rivera Monroy, Zuly Jenny et al. · 2017 · Journal of the Mexican Chemical Society · DOI
Full title: Efficient Synthesis of Peptides with 4-Methylpiperidine as Fmoc Removal Reagent by Solid Phase Synthesis
Authors: García Castañeda, Javier Eduardo; Vergel Galeano, Cristian Francisco; Rivera Monroy, Zuly Jenny; Rosas Pérez, Javier Eduardo
PaperApplication of a new green protocol in Solid-Phase Peptide Synthesis: identification of a new green solvent mixture compatible with ETT/TBEC
Vivenzio, G.; Scala, M.; Campiglia, P. et al. · 2024 · Proceedings of the 37th European Peptide Symposium · DOI
Full title: Application of a new green protocol in Solid-Phase Peptide Synthesis: identification of a new green solvent mixture compatible with ETT/TBEC
Authors: Vivenzio, G.; Scala, M.; Campiglia, P.; Sala, M.
Year: 2024
Venue: Proceedings of the 37th European Peptide Symposium
PaperReplacing DMF in solid-phase peptide synthesis: varying the composition of green binary solvent mixtures as a tool to mitigate common side-reactions
Jadhav, Sandip; Martin, Vincent; Egelund, Peter H. G. et al. · 2021 · Green Chemistry · DOI
Full title: Replacing DMF in solid-phase peptide synthesis: varying the composition of green binary solvent mixtures as a tool to mitigate common side-reactions
Authors: Jadhav, Sandip; Martin, Vincent; Egelund, Peter H. G.; Johansson Castro, Henrik; Krüger, Tobias; Richner, Franziska; Thordal Le Quement, Sebastian; Albericio, Fernando; Dettner, Frank; Lechner, Carolin; Schönleber, Ralph; Pedersen, Daniel Sejer
PaperSilylated Tag-Assisted Peptide Synthesis: Continuous One-Pot Elongation for the Production of Difficult Peptides under Environmentally Friendly Conditions
Full title: Silylated Tag-Assisted Peptide Synthesis: Continuous One-Pot Elongation for the Production of Difficult Peptides under Environmentally Friendly Conditions
PaperSolid-Phase Peptide Synthesis of Dipeptide (Histidine-β-Alanine) as a Chelating Agent by Using Trityl Chloride Resin, for Removal of Al<sup>3+</sup>, Cu<sup>2+</sup>, Hg<sup>2+</sup>and Pb<sup>2+</sup>: Experimental and Theoretical Study
Rahimi, Rahmatollah; Khosravi, Maryam; Tehrani, Mohammd H. H. et al. · 2016 · Journal of the Brazilian Chemical Society · DOI
Full title: Solid-Phase Peptide Synthesis of Dipeptide (Histidine-β-Alanine) as a Chelating Agent by Using Trityl Chloride Resin, for Removal of Al<sup>3+</sup>, Cu<sup>2+</sup>, Hg<sup>2+</sup>and Pb<sup>2+</sup>: Experimental and Theoretical Study
PaperA practical method for the synthesis of small peptides using DCC and HOBt as activators in H2O–THF while avoiding the use of protecting groups†
Herrera-Guzmán, Karina; Jaime-Vasconcelos, Miguel Ángel; Torales, Eréndira et al. · 2024 · RSC Advances · DOI
Full title: A practical method for the synthesis of small peptides using DCC and HOBt as activators in H2O–THF while avoiding the use of protecting groups†
Authors: Herrera-Guzmán, Karina; Jaime-Vasconcelos, Miguel Ángel; Torales, Eréndira; Chacón, Itzel; Gaviño, Rubén; García-Ríos, Eréndira; Cárdenas, Jorge; Morales-Serna, José A.
PaperScalable and Sustainable DMF-Free Solid-Phase Synthesis of Liraglutide by 1-Tert-Butyl-3-Ethylcarbodiimide-Mediated Couplings and Catch-and-Release Acylation and Purification Strategies
Pacini, Lorenzo; Muthyala, Manoj Kumar; Zitterbart, Robert et al. · 2025 · International Journal of Peptide Research and Therapeutics · DOI
Full title: Scalable and Sustainable DMF-Free Solid-Phase Synthesis of Liraglutide by 1-Tert-Butyl-3-Ethylcarbodiimide-Mediated Couplings and Catch-and-Release Acylation and Purification Strategies
Authors: Pacini, Lorenzo; Muthyala, Manoj Kumar; Zitterbart, Robert; Marder, Oleg; Rovero, Paolo; Papini, Anna Maria
Year: 2025
Venue: International Journal of Peptide Research and Therapeutics
PaperKey Green Chemistry research areas from a pharmaceutical manufacturers’ perspective revisited
Bryan, Marian C.; Dunn, Peter J.; Entwistle, David A. et al. · 2018 · Green Chemistry · DOI
Full title: Key Green Chemistry research areas from a pharmaceutical manufacturers’ perspective revisited
Authors: Bryan, Marian C.; Dunn, Peter J.; Entwistle, David A.; Gallou, Fabrice; Koenig, Stefan G.; Hayler, John; Hickey, Matthew; Hughes, Shaun; Kopach, Michael E.; Moine, Gérard; Richardson, Paul; Roschangar, Frank; Steven, Alan; Weiberth, Franz J.
PaperGreen Solvent Mixtures for Solid-Phase Peptide Synthesis: A Dimethylformamide-Free Highly Efficient Synthesis of Pharmaceutical-Grade Peptides
Ferrazzano, Lucia; Corbisiero, Dario; Martelli, Giulia et al. · 2019 · ACS Sustainable Chemistry & Engineering · DOI
Full title: Green Solvent Mixtures for Solid-Phase Peptide Synthesis: A Dimethylformamide-Free Highly Efficient Synthesis of Pharmaceutical-Grade Peptides
PaperAssessing the correlation of microscopy‐based and volumetry‐based measurements for resin swelling in a range of potential greener solvents for SPPS
Magtaan, Jordan Kevin; Devocelle, Marc; Kelleher, Fintan · 2020 · Journal of Peptide Science · DOI
Full title: Assessing the correlation of microscopy‐based and volumetry‐based measurements for resin swelling in a range of potential greener solvents for SPPS
Authors: Magtaan, Jordan Kevin; Devocelle, Marc; Kelleher, Fintan
PaperScalable and sustainable DMF-free solid-phase synthesis of liraglutideby 1-tert-butyl-3-ethylcarbodiimide-mediated couplings and catch-and-release acylation and purification strategies
Pacini, Lorenzo; Muthyala, Manoj Kumar; Zitterbart, Robert et al. · 2025 · DOI
Full title: Scalable and sustainable DMF-free solid-phase synthesis of liraglutideby 1-tert-butyl-3-ethylcarbodiimide-mediated couplings and catch-and-release acylation and purification strategies
Authors: Pacini, Lorenzo; Muthyala, Manoj Kumar; Zitterbart, Robert; Marder, Oleg; Rovero, Paolo; Papini, Anna Maria
PaperThe Antimicrobial Peptide Capitellacin: Chemical Synthesis of Analogues to Probe the Role of Disulphide Bridges and Their Replacement with Vinyl Sulphides
Shepperson, Oscar A.; Harris, Paul W. R.; Brimble, Margaret A. et al. · 2024 · Antibiotics · DOI
Full title: The Antimicrobial Peptide Capitellacin: Chemical Synthesis of Analogues to Probe the Role of Disulphide Bridges and Their Replacement with Vinyl Sulphides
Authors: Shepperson, Oscar A.; Harris, Paul W. R.; Brimble, Margaret A.; Cameron, Alan J.
PaperBrønsted Acid–Lewis Acid (BA–LA) Induced Final Deprotection/Peptide Resin Cleavage in Fmoc/<i>t-</i>Bu Solid-Phase Peptide Synthesis: HCl/FeCl<sub>3</sub> and AcOH/FeCl<sub>3</sub> as Viable PFAS-Free Alternatives for TFA
Pawlas, Jan; André, Christophe; Rasmussen, Jon H. et al. · 2024 · Organic Letters · DOI
Full title: Brønsted Acid–Lewis Acid (BA–LA) Induced Final Deprotection/Peptide Resin Cleavage in Fmoc/<i>t-</i>Bu Solid-Phase Peptide Synthesis: HCl/FeCl<sub>3</sub> and AcOH/FeCl<sub>3</sub> as Viable PFAS-Free Alternatives for TFA
Authors: Pawlas, Jan; André, Christophe; Rasmussen, Jon H.; Ludemann-Hombourger, Olivier
PaperPeptides conjugated to 2-alkoxy-8-oxo-adenine as potential synthetic vaccines triggering TLR7
Gential, Geoffroy P. P.; Hogervorst, Tim P.; Tondini, Elena et al. · 2019 · Bioorganic & Medicinal Chemistry Letters · DOI
Full title: Peptides conjugated to 2-alkoxy-8-oxo-adenine as potential synthetic vaccines triggering TLR7
Authors: Gential, Geoffroy P. P.; Hogervorst, Tim P.; Tondini, Elena; Graaff, Michel J. van de; Overkleeft, Herman S.; Codée, Jeroen D. C.; Marel, Gijsbert A. van der; Ossendorp, Ferry; Filippov, Dmitri V.
PaperUsing <sup>19</sup>F NMR and two‐level factorial design to explore thiol‐fluoride substitution in hexafluorobenzene and its application in peptide stapling and cyclisation
Dognini, Paolo; Killoran, Patrick M.; Hanson, George S. M. et al. · 2020 · Peptide Science · DOI
Full title: Using <sup>19</sup>F NMR and two‐level factorial design to explore thiol‐fluoride substitution in hexafluorobenzene and its application in peptide stapling and cyclisation
Authors: Dognini, Paolo; Killoran, Patrick M.; Hanson, George S. M.; Halsall, Lewis; Chaudhry, Talhat; Islam, Zasharatul; Giuntini, Francesca; Coxon, Christopher R.
PaperSmall animal PET imaging with the 68Ga-labeled pH (low) insertion peptide-like peptide YJL-4 in a triple-negative breast cancer mouse model
Chen, YueHua; Song, ShuangShuang; Sun, YanQin et al. · 2024 · figshare · DOI
Full title: Small animal PET imaging with the 68Ga-labeled pH (low) insertion peptide-like peptide YJL-4 in a triple-negative breast cancer mouse model
PaperMethodologies for attaching polypyridyl ligands into amino acids and synthesis and biological evaluation of novel light activated peptidomimetic cysteine protease inhibitors caged by RuII(bpy)2
Respondek, Tomasz · 2013 · DigitalCommons - WayneState (Wayne State University)
Full title: Methodologies for attaching polypyridyl ligands into amino acids and synthesis and biological evaluation of novel light activated peptidomimetic cysteine protease inhibitors caged by RuII(bpy)2
Authors: Respondek, Tomasz
Year: 2013
Venue: DigitalCommons - WayneState (Wayne State University)
PaperTargeted Amino Acid Substitutions in a Trichoderma Peptaibol Confer Activity against Fungal Plant Pathogens and Protect Host Tissues from Botrytis cinerea Infection
De Zotti, Marta; Sella, Luca; Bolzonello, Angela et al. · 2020 · International Journal of Molecular Sciences · DOI
Full title: Targeted Amino Acid Substitutions in a Trichoderma Peptaibol Confer Activity against Fungal Plant Pathogens and Protect Host Tissues from Botrytis cinerea Infection
Authors: De Zotti, Marta; Sella, Luca; Bolzonello, Angela; Gabbatore, Laura; Peggion, Cristina; Bortolotto, Alessandro; Elmaghraby, Ibrahim; Tundo, Silvio; Favaron, Francesco
Year: 2020
Venue: International Journal of Molecular Sciences
PaperA Targeted Drug Delivery Strategy for Trypanosomiasis Towards a Diastereoselective Boronate Ester Mediated Intramolecular Diels-Alder Cycloaddition
Gordhan, Heeren M. · 2017 · TigerPrints (Clemson University)
Full title: A Targeted Drug Delivery Strategy for Trypanosomiasis Towards a Diastereoselective Boronate Ester Mediated Intramolecular Diels-Alder Cycloaddition
Authors: Gordhan, Heeren M.
Year: 2017
Venue: TigerPrints (Clemson University)
PaperAlternative chemistries for the synthesis of thrombospondin‐1 type 1 repeats
Tiefenbrunn, Theresa K.; Blanco‐Canosa, Juan; Dawson, Philip E. · 2010 · Peptide Science · DOI
Full title: Alternative chemistries for the synthesis of thrombospondin‐1 type 1 repeats
Authors: Tiefenbrunn, Theresa K.; Blanco‐Canosa, Juan; Dawson, Philip E.
PaperSupplementary material from "Phenothiazine-linked Glutamic Acid Dendrons: An Easy Access and a New Class of SARS-CoV2 Main Protease Inhibitors"
Singh, Sameer; Gangopadhyay, Aditi; D, Sriram et al. · 2025 · The Royal Society · DOI
Full title: Supplementary material from "Phenothiazine-linked Glutamic Acid Dendrons: An Easy Access and a New Class of SARS-CoV2 Main Protease Inhibitors"
PaperNew green base for Fmoc removal in solid-phase peptide synthesis: 1,5-diazabicyclo[4.3.0]non-5-ene (DBN), a promising sustainable alternative to piperidine
Scala, Maria Carmina; Vivenzio, Giovanni; Manfra, Michele et al. · 2025 · Taylor & Francis · DOI
Full title: New green base for Fmoc removal in solid-phase peptide synthesis: 1,5-diazabicyclo[4.3.0]non-5-ene (DBN), a promising sustainable alternative to piperidine
Authors: Scala, Maria Carmina; Vivenzio, Giovanni; Manfra, Michele; Sala, Marina; Campiglia, Pietro
Paper[68Ga]FSC-(RGD)3 a trimeric RGD peptide for imaging αvβ3 integrin expression based on a novel siderophore derived chelating scaffold—synthesis and evaluation
Peter A. Knetsch; Chuangyan Zhai; Christine Rangger et al. · 2015 · OpenAlex · DOI
Full title: [68Ga]FSC-(RGD)3 a trimeric RGD peptide for imaging αvβ3 integrin expression based on a novel siderophore derived chelating scaffold—synthesis and evaluation
Authors: Peter A. Knetsch; Chuangyan Zhai; Christine Rangger; Michael Blatzer; Hubertus Haas; Piriya Kaeopookum; Roland Haubner; Clemens Decristoforo
PaperTotal synthesis of argyrin A and analogues thereof
Chen, Chou-Hsiung · 2013 · Nottingham ePrints (University of Nottingham)
Full title: Total synthesis of argyrin A and analogues thereof
Authors: Chen, Chou-Hsiung
Year: 2013
Venue: Nottingham ePrints (University of Nottingham)
PaperAnalogs of a Natural Peptaibol Exert Anticancer Activity in Both Cisplatin- and Doxorubicin-Resistant Cells and in Multicellular Tumor Spheroids
Casagrande, Naike; Borghese, Cinzia; Gabbatore, Laura et al. · 2021 · International Journal of Molecular Sciences · DOI
Full title: Analogs of a Natural Peptaibol Exert Anticancer Activity in Both Cisplatin- and Doxorubicin-Resistant Cells and in Multicellular Tumor Spheroids
PaperSupplementary material from "Macrocylases as synthetic tools for ligand synthesis: enzymatic synthesis of cyclic peptides containing metal-binding amino acids"
Brewster, Richard C.; Labeaga, Irati Colmenero; Soden, Catriona E. et al. · 2021 · The Royal Society · DOI
Full title: Supplementary material from "Macrocylases as synthetic tools for ligand synthesis: enzymatic synthesis of cyclic peptides containing metal-binding amino acids"
Authors: Brewster, Richard C.; Labeaga, Irati Colmenero; Soden, Catriona E.; Jarvis, Amanda G.
PaperSynthesis of U-theraphotoxin-Pv1a_1, an Aedes aegypti larvicidal disulfide bridged peptide from the Colombian tarantula Pamphobeteus verdolaga (Araneae: Theraphosidae)
Estrada-Gómez, Sebastián; Salinas-Restrepo, Cristian; Vargas-Muñoz, Leidy Johana et al. · 2025 · Toxicon: X · DOI
Full title: Synthesis of U-theraphotoxin-Pv1a_1, an Aedes aegypti larvicidal disulfide bridged peptide from the Colombian tarantula Pamphobeteus verdolaga (Araneae: Theraphosidae)
PaperA novel approach to amino acid synthesis: acid-assisted reactions with dimethyl carbonate for efficient <i>O</i>-methylated, <i>N</i>,<i>O</i>-methylated and <i>N</i>-formylated derivatives
Worsawat, Pattamabhorn; Noppawan, Pakin; Supanchaiyamat, Nontipa et al. · 2024 · Green Chemistry · DOI
Full title: A novel approach to amino acid synthesis: acid-assisted reactions with dimethyl carbonate for efficient <i>O</i>-methylated, <i>N</i>,<i>O</i>-methylated and <i>N</i>-formylated derivatives
Authors: Worsawat, Pattamabhorn; Noppawan, Pakin; Supanchaiyamat, Nontipa; Wu, Himmy; McElroy, Con R.; Hunt, Andrew J.
PaperRemoval of acid-labile protecting or anchoring groups in the presence of polyfluorinated alcohol: Application to solid-phase peptide synthesis
Stetsenko, D. A.; Apukhtina, V. S.; Chelobanov, B. P. et al. · 2016 · Russian Journal of Bioorganic Chemistry · DOI
Full title: Removal of acid-labile protecting or anchoring groups in the presence of polyfluorinated alcohol: Application to solid-phase peptide synthesis
Authors: Stetsenko, D. A.; Apukhtina, V. S.; Chelobanov, B. P.; Palladino, P.
PaperSulfur And Selenium In Peptides And Proteins: Part I – Chemoselective Methods For Disulfide Bond Formation, Part Ii – Function Of Selenium In Enzymes.
Ste.Marie, Emma J. · 2020 · ScholarWorks @UVM (University of Vermont)
Full title: Sulfur And Selenium In Peptides And Proteins: Part I – Chemoselective Methods For Disulfide Bond Formation, Part Ii – Function Of Selenium In Enzymes.
Authors: Ste.Marie, Emma J.
Year: 2020
Venue: ScholarWorks @UVM (University of Vermont)
PaperGreening the Solid-Phase Peptide Synthesis Process. 2-MeTHF for the Incorporation of the First Amino Acid and Precipitation of Peptides after Global Deprotection
Al Musaimi, Othman; Jad, Yahya E.; Kumar, Ashish et al. · 2018 · Organic Process Research & Development · DOI
Full title: Greening the Solid-Phase Peptide Synthesis Process. 2-MeTHF for the Incorporation of the First Amino Acid and Precipitation of Peptides after Global Deprotection
Authors: Al Musaimi, Othman; Jad, Yahya E.; Kumar, Ashish; El-Faham, Ayman; Collins, Jonathan M.; Basso, Alessandra; de la Torre, Beatriz G.; Albericio, Fernando
PaperDesign, synthesis, and biological evaluation of a multifunctional neuropeptide-Y conjugate for selective nuclear delivery of radiolanthanides
Chastel, Adrien; Worm, Dennis J.; Alves, Isabel D. et al. · 2020 · EJNMMI Research · DOI
Full title: Design, synthesis, and biological evaluation of a multifunctional neuropeptide-Y conjugate for selective nuclear delivery of radiolanthanides
PaperLinear Peptide Analogues from Jatropha’s Orbitides Promote Migration of Human Neonatal Foreskin Fibroblasts in vitro and Collagen Deposition
Suelem D. Ramalho; Pinto, Meri Emili F.; Andricopulo, Renata K. et al. · 2019 · SciELO journals · DOI
Full title: Linear Peptide Analogues from Jatropha’s Orbitides Promote Migration of Human Neonatal Foreskin Fibroblasts in vitro and Collagen Deposition
Authors: Suelem D. Ramalho; Pinto, Meri Emili F.; Andricopulo, Renata K.; Sanches, Paulo R. S.; Edilberto R. Silveira; Cilli, Eduardo M.; Andricopulo, Adriano D.; Vanderlan S. Bolzani
PaperSynthesis and cellular penetration properties of new phosphonium based cationic amphiphilic peptides† †Electronic supplementary information (ESI) available. See DOI: 10.1039/c8md00113h
Silva Nigenda, Ezequiel; Postma, Tobias M.; Hezwani, Mohammed et al. · 2018 · MedChemComm · DOI
Full title: Synthesis and cellular penetration properties of new phosphonium based cationic amphiphilic peptides† †Electronic supplementary information (ESI) available. See DOI: 10.1039/c8md00113h
Authors: Silva Nigenda, Ezequiel; Postma, Tobias M.; Hezwani, Mohammed; Pirvan, Alin; Gannon, Susan; Smith, Carol-Anne; Riehle, Mathis; Liskamp, Rob M. J.
PaperSynthetic studies with the brevicidine and laterocidine lipopeptide antibiotics including analogues with enhanced properties and in vivo efficacy†
Al Ayed, Karol; Ballantine, Ross D.; Hoekstra, Michael et al. · 2022 · Chemical Science · DOI
Full title: Synthetic studies with the brevicidine and laterocidine lipopeptide antibiotics including analogues with enhanced properties and in vivo efficacy†
Authors: Al Ayed, Karol; Ballantine, Ross D.; Hoekstra, Michael; Bann, Samantha J.; Wesseling, Charlotte M. J.; Bakker, Alexander T.; Zhong, Zheng; Li, Yong-Xin; Brüchle, Nora C.; van der Stelt, Mario; Cochrane, Stephen A.; Martin, Nathaniel I.
Paper- **DOI:** 10.26262/heal.auth.ir.347860 - **Authors:** Γιαννόπουλος-Δημητρίου, Αλέξανδρος του Δημητρίου - **Year:** 2023 - **Journal:** Aristotle University of Thessaloniki
Γιαννόπουλος-Δημητρίου, Αλέξανδρος του Δημητρίου · 2023 · Aristotle University of Thessaloniki · DOI
Full title: - **DOI:** 10.26262/heal.auth.ir.347860 - **Authors:** Γιαννόπουλος-Δημητρίου, Αλέξανδρος του Δημητρίου - **Year:** 2023 - **Journal:** Aristotle University of Thessaloniki
Authors: Γιαννόπουλος-Δημητρίου, Αλέξανδρος του Δημητρίου
PaperSolid‐Phase Synthesis of the Aged‐Nonapeptide‐Nerve‐Agent Adduct of Butyrylcholinesterase as Reference Materials for Analytical Verification
Bielmann, Andreas; Curty, Christophe; Bochet, Christian G. · 2017 · Helvetica Chimica Acta · DOI
Full title: Solid‐Phase Synthesis of the Aged‐Nonapeptide‐Nerve‐Agent Adduct of Butyrylcholinesterase as Reference Materials for Analytical Verification
Authors: Bielmann, Andreas; Curty, Christophe; Bochet, Christian G.
PaperDesign of PSMA ligands with modifications at the inhibitor part: an approach to reduce the salivary gland uptake of radiolabeled PSMA inhibitors?
Felber, Veronika Barbara; Valentin, Manuel Amando; Hans-Jürgen Wester · 2021 · figshare · DOI
Full title: Design of PSMA ligands with modifications at the inhibitor part: an approach to reduce the salivary gland uptake of radiolabeled PSMA inhibitors?
Authors: Felber, Veronika Barbara; Valentin, Manuel Amando; Hans-Jürgen Wester
PaperPreparation, Radiolabeling with 68Ga/177Lu and Preclinical Evaluation of Novel Angiotensin Peptide Analog: A New Class of Peptides for Breast Cancer Targeting
Full title: Preparation, Radiolabeling with 68Ga/177Lu and Preclinical Evaluation of Novel Angiotensin Peptide Analog: A New Class of Peptides for Breast Cancer Targeting
PaperDesign, synthesis and structure-activity relationship study of wollamide B; a new potential anti TB agent
Asfaw, Henok; Laqua, Katja; Walkowska, Anna Maria et al. · 2017 · PLoS ONE · DOI
Full title: Design, synthesis and structure-activity relationship study of wollamide B; a new potential anti TB agent
Authors: Asfaw, Henok; Laqua, Katja; Walkowska, Anna Maria; Cunningham, Fraser; Martinez-Martinez, Maria Santos; Cuevas-Zurita, Juan Carlos; Ballell-Pages, Lluís; Imming, Peter
PaperNew green base for Fmoc removal in solid-phase peptide synthesis: 1,5-diazabicyclo[4.3.0]non-5-ene (DBN), a promising sustainable alternative to piperidine
Scala, Maria Carmina; Vivenzio, Giovanni; Manfra, Michele et al. · 2025 · Taylor & Francis · DOI
Full title: New green base for Fmoc removal in solid-phase peptide synthesis: 1,5-diazabicyclo[4.3.0]non-5-ene (DBN), a promising sustainable alternative to piperidine
Authors: Scala, Maria Carmina; Vivenzio, Giovanni; Manfra, Michele; Sala, Marina; Campiglia, Pietro
PaperSynthesis, Antitumor and Antibacterial Studies of New Shortened Analogues of (KLAKLAK)2-NH2 and Their Conjugates Containing Unnatural Amino Acids
Jaber, Sirine; Iliev, Ivan; Angelova, Tsvetelina et al. · 2021 · Molecules · DOI
Full title: Synthesis, Antitumor and Antibacterial Studies of New Shortened Analogues of (KLAKLAK)2-NH2 and Their Conjugates Containing Unnatural Amino Acids
PaperAn optimized protocol for the synthesis of peptides containing trans-cyclooctene and bicyclononyne dienophiles as useful multifunctional bioorthogonal probes
La-Venia, Agustina; Dzijak, Rastislav; Rampmaier, Robert et al. · 2021 · Zenodo · DOI
Full title: An optimized protocol for the synthesis of peptides containing trans-cyclooctene and bicyclononyne dienophiles as useful multifunctional bioorthogonal probes
Authors: La-Venia, Agustina; Dzijak, Rastislav; Rampmaier, Robert; Vrabel, Milan
PaperA novel series of dipeptide derivatives containing indole-3-carboxylic acid conjugates as potential antimicrobial agents: the design, solid phase peptide synthesis, in vitro biological evaluation, and molecular docking study†
Tivari, Sunil R.; Kokate, Siddhant V.; Delgado-Alvarado, Enrique et al. · 2023 · RSC Advances · DOI
Full title: A novel series of dipeptide derivatives containing indole-3-carboxylic acid conjugates as potential antimicrobial agents: the design, solid phase peptide synthesis, in vitro biological evaluation, and molecular docking study†
PaperExploring the Chemical Properties and Medicinal Applications of Tetramethylthiocycloheptyne Sulfoximine Used in Strain-Promoted Azide–Alkyne Cycloaddition Reactions
Timmers, Matt; Kipper, Andi; Frey, Raphael et al. · 2023 · Pharmaceuticals · DOI
Full title: Exploring the Chemical Properties and Medicinal Applications of Tetramethylthiocycloheptyne Sulfoximine Used in Strain-Promoted Azide–Alkyne Cycloaddition Reactions
PaperA Novel Amphibian Antimicrobial Peptide, Phylloseptin-PV1, Exhibits Effective Anti-staphylococcal Activity Without Inducing Either Hepatic or Renal Toxicity in Mice
Yue Liu; Daning Shi; Jin Wang et al. · 2020 · OpenAlex · DOI
Full title: A Novel Amphibian Antimicrobial Peptide, Phylloseptin-PV1, Exhibits Effective Anti-staphylococcal Activity Without Inducing Either Hepatic or Renal Toxicity in Mice
Authors: Yue Liu; Daning Shi; Jin Wang; Xiaoling Chen; Mei Zhou; Xinping Xi; Jianming Cheng; Chengbang Ma; Tianbao Chen; Chris Shaw; Lei Wang
PaperCombining Real-Time Monitoring Using Raman Spectroscopy, Rotating-Bed Reactors, and Green Solvents to Improve Sustainability in Solid-Phase Peptide Synthesis
Fournier, Eugenie; Vijeta, Arjun; Babii, Oleg et al. · 2024 · ACS Sustainable Chemistry & Engineering · DOI
Full title: Combining Real-Time Monitoring Using Raman Spectroscopy, Rotating-Bed Reactors, and Green Solvents to Improve Sustainability in Solid-Phase Peptide Synthesis
PaperDipropyleneglycol Dimethylether, New Green Solvent for Solid-Phase Peptide Synthesis: Further Challenges to Improve Sustainability in the Development of Therapeutic Peptides
Vivenzio, Giovanni; Scala, Maria Carmina; Marino, Pasquale et al. · 2023 · Pharmaceutics · DOI
Full title: Dipropyleneglycol Dimethylether, New Green Solvent for Solid-Phase Peptide Synthesis: Further Challenges to Improve Sustainability in the Development of Therapeutic Peptides
Authors: Vivenzio, Giovanni; Scala, Maria Carmina; Marino, Pasquale; Manfra, Michele; Campiglia, Pietro; Sala, Marina
PaperSupplementary material from "Phenothiazine-linked Glutamic Acid Dendrons: An Easy Access and a New Class of SARS-CoV2 Main Protease Inhibitors"
Singh, Sameer; Gangopadhyay, Aditi; D, Sriram et al. · 2025 · The Royal Society · DOI
Full title: Supplementary material from "Phenothiazine-linked Glutamic Acid Dendrons: An Easy Access and a New Class of SARS-CoV2 Main Protease Inhibitors"
Paper1,3,5-Triazine as Branching Connector for the Construction of Novel Antimicrobial Peptide Dendrimers: Synthesis and Biological Characterization
Sheyi, Rotimi; Mhlongo, Jessica T.; Jorba, Marta et al. · 2024 · International Journal of Molecular Sciences · DOI
Full title: 1,3,5-Triazine as Branching Connector for the Construction of Novel Antimicrobial Peptide Dendrimers: Synthesis and Biological Characterization
Authors: Sheyi, Rotimi; Mhlongo, Jessica T.; Jorba, Marta; Fusté, Ester; Sharma, Anamika; Viñas, Miguel; Albericio, Fernando; Espinal, Paula; de la Torre, Beatriz G.
Year: 2024
Venue: International Journal of Molecular Sciences
PaperSynthesis, Antimalarial Activity and Molecular Dynamics Studies of Pipecolisporin: A Novel Cyclic Hexapeptide with Potent Therapeutic Potential
Kurniaty, Nety; Fakih, Taufik Muhammad; Maharani, Rani et al. · 2025 · Molecules · DOI
Full title: Synthesis, Antimalarial Activity and Molecular Dynamics Studies of Pipecolisporin: A Novel Cyclic Hexapeptide with Potent Therapeutic Potential
PaperNovel Protocol for the Chemical Synthesis of Crustacean Hyperglycemic Hormone Analogues — An Efficient Experimental Tool for Studying Their Functions
Mosco, Alessandro; Zlatev, Vientsislav; Guarnaccia, Corrado et al. · 2012 · PLoS ONE · DOI
Full title: Novel Protocol for the Chemical Synthesis of Crustacean Hyperglycemic Hormone Analogues — An Efficient Experimental Tool for Studying Their Functions
PaperAn Efficient, Site‐Selective and Spontaneous Peptide Macrocyclisation During in vitro Translation
Liu, Minglong; Yoshisada, Ryoji; Amedi, Avand et al. · 2022 · Chemistry - A European Journal · DOI
Full title: An Efficient, Site‐Selective and Spontaneous Peptide Macrocyclisation During in vitro Translation
Authors: Liu, Minglong; Yoshisada, Ryoji; Amedi, Avand; Hopstaken, Antonius J. P.; Pascha, Mirte N.; Haan, Cornelis A. M. de; Geerke, Daan P.; Poole, David A.; Jongkees, Seino A. K.
PaperAqueous Microwave-Assisted Solid-Phase Peptide Synthesis Using Fmoc Strategy. II. Racemization Studies and Water Based Synthesis of Cysteine- Containing Peptides
Hojo, Keiko; Shinozaki, Natsuki; Hara, Asaki et al. · 2013 · Protein & Peptide Letters · DOI
Full title: Aqueous Microwave-Assisted Solid-Phase Peptide Synthesis Using Fmoc Strategy. II. Racemization Studies and Water Based Synthesis of Cysteine- Containing Peptides
PaperSupplementary material from "Macrocylases as synthetic tools for ligand synthesis: enzymatic synthesis of cyclic peptides containing metal-binding amino acids"
Brewster, Richard C.; Labeaga, Irati Colmenero; Soden, Catriona E. et al. · 2021 · The Royal Society · DOI
Full title: Supplementary material from "Macrocylases as synthetic tools for ligand synthesis: enzymatic synthesis of cyclic peptides containing metal-binding amino acids"
Authors: Brewster, Richard C.; Labeaga, Irati Colmenero; Soden, Catriona E.; Jarvis, Amanda G.
PaperNovel luminescent peptide conjugates for assessing protein and other biomolecules location and function
Blackmore, Lorraine · 2013 · Dublin City University Open Access Institutional Repository (Dublin City University)
Full title: Novel luminescent peptide conjugates for assessing protein and other biomolecules location and function
Authors: Blackmore, Lorraine
Year: 2013
Venue: Dublin City University Open Access Institutional Repository (Dublin City University)
PaperA Peptide-Based Nanocarrier for an Enhanced Delivery and Targeting of Flurbiprofen into the Brain for the Treatment of Alzheimer’s Disease: An In Vitro Study
Al-azzawi, Shafq; Masheta, Dhafir; Guildford, Anna et al. · 2020 · Nanomaterials · DOI
Full title: A Peptide-Based Nanocarrier for an Enhanced Delivery and Targeting of Flurbiprofen into the Brain for the Treatment of Alzheimer’s Disease: An In Vitro Study
PaperLinear Peptide Analogues from Jatropha’s Orbitides Promote Migration of Human Neonatal Foreskin Fibroblasts in vitro and Collagen Deposition
Suelem D. Ramalho; Pinto, Meri Emili F.; Andricopulo, Renata K. et al. · 2019 · SciELO journals · DOI
Full title: Linear Peptide Analogues from Jatropha’s Orbitides Promote Migration of Human Neonatal Foreskin Fibroblasts in vitro and Collagen Deposition
Authors: Suelem D. Ramalho; Pinto, Meri Emili F.; Andricopulo, Renata K.; Sanches, Paulo R. S.; Edilberto R. Silveira; Cilli, Eduardo M.; Andricopulo, Adriano D.; Vanderlan S. Bolzani
PaperApplication of a new green protocol in solid-phase peptide synthesis: identification of a new green solvent mixture compatible with TBEC/ETT
Vivenzio, Giovanni; Scala, Maria Carmina; Auriemma, Giulia et al. · 2024 · Taylor & Francis · DOI
Full title: Application of a new green protocol in solid-phase peptide synthesis: identification of a new green solvent mixture compatible with TBEC/ETT
Authors: Vivenzio, Giovanni; Scala, Maria Carmina; Auriemma, Giulia; Sardo, Carla; Campiglia, Pietro; Sala, Marina
PaperApplication of a new green protocol in solid-phase peptide synthesis: identification of a new green solvent mixture compatible with TBEC/ETT
Vivenzio, Giovanni; Scala, Maria Carmina; Auriemma, Giulia et al. · 2024 · Green Chemistry Letters and Reviews · DOI
Full title: Application of a new green protocol in solid-phase peptide synthesis: identification of a new green solvent mixture compatible with TBEC/ETT
Authors: Vivenzio, Giovanni; Scala, Maria Carmina; Auriemma, Giulia; Sardo, Carla; Campiglia, Pietro; Sala, Marina
PaperA Chemical Biology Approach to Understanding Molecular Recognition of Lipid II by Nisin(1–12): Synthesis and NMR Ensemble Analysis of Nisin(1–12) and Analogues
Dickman, Rachael; Danelius, Emma; Mitchell, Serena A. et al. · 2019 · Chemistry (Weinheim an Der Bergstrasse, Germany) · DOI
Full title: A Chemical Biology Approach to Understanding Molecular Recognition of Lipid II by Nisin(1–12): Synthesis and NMR Ensemble Analysis of Nisin(1–12) and Analogues
Authors: Dickman, Rachael; Danelius, Emma; Mitchell, Serena A.; Hansen, D. Flemming; Erdélyi, Máté; Tabor, Alethea B.
Year: 2019
Venue: Chemistry (Weinheim an Der Bergstrasse, Germany)
Paper[68Ga]FSC-(RGD)3 a trimeric RGD peptide for imaging αvβ3 integrin expression based on a novel siderophore derived chelating scaffold—synthesis and evaluation
Peter A. Knetsch; Chuangyan Zhai; Christine Rangger et al. · 2015 · OpenAlex · DOI
Full title: [68Ga]FSC-(RGD)3 a trimeric RGD peptide for imaging αvβ3 integrin expression based on a novel siderophore derived chelating scaffold—synthesis and evaluation
Authors: Peter A. Knetsch; Chuangyan Zhai; Christine Rangger; Michael Blatzer; Hubertus Haas; Piriya Kaeopookum; Roland Haubner; Clemens Decristoforo
PaperChemical Synthesis of Modularly Modified Analogs of E2/NS1 Peptides on a Novel Chemically and Mechanically Stable Terpolymer of 1,6-Hexanediol Diacrylate, N-Vinylpyrrolidone on Styrene Support
Jacob, Sunil; Harry, Nissy Ann; Binoj, K.K. et al. · 2023 · Trends in Sciences · DOI
Full title: Chemical Synthesis of Modularly Modified Analogs of E2/NS1 Peptides on a Novel Chemically and Mechanically Stable Terpolymer of 1,6-Hexanediol Diacrylate, N-Vinylpyrrolidone on Styrene Support
PaperApplication of a new green protocol in solid-phase peptide synthesis: identification of a new green solvent mixture compatible with TBEC/ETT
Vivenzio, Giovanni; Scala, Maria Carmina; Auriemma, Giulia et al. · 2024 · Taylor & Francis · DOI
Full title: Application of a new green protocol in solid-phase peptide synthesis: identification of a new green solvent mixture compatible with TBEC/ETT
Authors: Vivenzio, Giovanni; Scala, Maria Carmina; Auriemma, Giulia; Sardo, Carla; Campiglia, Pietro; Sala, Marina
Paper<i>N</i>‐Butylpyrrolidinone is an equally good solvent as <i>N</i>,<i>N</i>‐dimethylformamide for microwave assisted solid phase peptide synthesis
Öhlander, Andrea; Lüdtke, Carsten; Sahakjan, Artur et al. · 2024 · Journal of Peptide Science · DOI
Full title: <i>N</i>‐Butylpyrrolidinone is an equally good solvent as <i>N</i>,<i>N</i>‐dimethylformamide for microwave assisted solid phase peptide synthesis
Authors: Öhlander, Andrea; Lüdtke, Carsten; Sahakjan, Artur; Johnsson, Richard E.
PaperDesign of PSMA ligands with modifications at the inhibitor part: an approach to reduce the salivary gland uptake of radiolabeled PSMA inhibitors?
Felber, Veronika Barbara; Valentin, Manuel Amando; Hans-Jürgen Wester · 2021 · figshare · DOI
Full title: Design of PSMA ligands with modifications at the inhibitor part: an approach to reduce the salivary gland uptake of radiolabeled PSMA inhibitors?
Authors: Felber, Veronika Barbara; Valentin, Manuel Amando; Hans-Jürgen Wester
PaperSelf-assembled proteomimetic (SAP) with antibody-like binding from short PNA–peptide conjugates
Brennecke, Benjamin; Civili, Beatrice; Sabale, Pramod M. et al. · 2025 · Proceedings of the National Academy of Sciences of the United States of America · DOI
Full title: Self-assembled proteomimetic (SAP) with antibody-like binding from short PNA–peptide conjugates
Authors: Brennecke, Benjamin; Civili, Beatrice; Sabale, Pramod M.; Barluenga, Sofia; Meyer, Benjamin; Winssinger, Nicolas
Year: 2025
Venue: Proceedings of the National Academy of Sciences of the United States of America
PaperSynthesis of the transmembrane domain of the spike protein from SARS‐CoV‐2 using solid phase peptide synthesis and determination of its oligomerization state
Grimes, Loyal T.; Reichart, Timothy M. · 2022 · The FASEB Journal · DOI
Full title: Synthesis of the transmembrane domain of the spike protein from SARS‐CoV‐2 using solid phase peptide synthesis and determination of its oligomerization state
PaperDesign, synthesis, and biological evaluation of a multifunctional neuropeptide-Y conjugate for selective nuclear delivery of radiolanthanides
Chastel, Adrien; Worm, Dennis; Alves, Isabel et al. · 2020 · figshare · DOI
Full title: Design, synthesis, and biological evaluation of a multifunctional neuropeptide-Y conjugate for selective nuclear delivery of radiolanthanides
PaperSynthesis of Trifluoromethyl Ketone Containing Amino Acid Building Blocks for the Preparation of Peptide-Based Histone Deacetylase (HDAC) Inhibitors
Olsen, Christian; Moreno-Yruela, Carlos · 2018 · Synthesis · DOI
Full title: Synthesis of Trifluoromethyl Ketone Containing Amino Acid Building Blocks for the Preparation of Peptide-Based Histone Deacetylase (HDAC) Inhibitors
PaperSynthesis of Trypsin-modulating Oostatic Factor (TMOF) and its Analogues by Solid-phase Peptide Synthesis Using DIC/Oxyma as Coupling Reagent
Maharani, Rani; Yanti, Eka Fitri; Melati, M.Devia Irma et al. · 2015 · Procedia Chemistry · DOI
Full title: Synthesis of Trypsin-modulating Oostatic Factor (TMOF) and its Analogues by Solid-phase Peptide Synthesis Using DIC/Oxyma as Coupling Reagent
PaperVenomous gland transcriptome and venom proteomic analysis of the scorpion Androctonus amoreuxi reveal new peptides with anti-SARS-CoV2 activity.
Ghazal A, Clarke D, Abdel-Rahman MA, Ribeiro A, Hijazi K, Collie-Duguid E, Pattinson C, Burgoyne K, Muhammad T, Alfadhel S, Heidari Z, Samir R, Gerges MM, Colamarino RA, Houssen WE. · 2023 · DOI
Full title: Venomous gland transcriptome and venom proteomic analysis of the scorpion Androctonus amoreuxi reveal new peptides with anti-SARS-CoV2 activity.
Authors: Ghazal A, Clarke D, Abdel-Rahman MA, Ribeiro A, Hijazi K, Collie-Duguid E, Pattinson C, Burgoyne K, Muhammad T, Alfadhel S, Heidari Z, Samir R, Gerges MM, Colamarino RA, Houssen WE.
PaperSynthesis of <i>C</i>‐Glycosyl Amino Acid Building Blocks Suitable for the Solid‐Phase Synthesis of Multivalent Glycopeptide Mimics
Reintjens, Niels R. M.; Koemans, Tony S.; Zilverschoon, Nick et al. · 2020 · European Journal of Organic Chemistry · DOI
Full title: Synthesis of <i>C</i>‐Glycosyl Amino Acid Building Blocks Suitable for the Solid‐Phase Synthesis of Multivalent Glycopeptide Mimics
Authors: Reintjens, Niels R. M.; Koemans, Tony S.; Zilverschoon, Nick; Castelli, Riccardo; Cordfunke, Robert A.; Drijfhout, Jan Wouter; Meeuwenoord, Nico J.; Overkleeft, Herman S.; Filippov, Dmitri V.; van der Marel, Gijsbert A.; Codée, Jeroen D. C.
PaperSynthesis, Physicochemical Characterization, In Vitro 2D/3D Human Cell Culture, and In Vitro Aerosol Dispersion Performance of Advanced Spray Dried and Co-Spray Dried Angiotensin (1—7) Peptide and PNA5 with Trehalose as Microparticles/Nanoparticles for Targeted Respiratory Delivery as Dry Powder Inhalers
Alabsi, Wafaa; Acosta, Maria F.; Al-Obeidi, Fahad A. et al. · 2021 · Pharmaceutics · DOI
Full title: Synthesis, Physicochemical Characterization, In Vitro 2D/3D Human Cell Culture, and In Vitro Aerosol Dispersion Performance of Advanced Spray Dried and Co-Spray Dried Angiotensin (1—7) Peptide and PNA5 with Trehalose as Microparticles/Nanoparticles for Targeted Respiratory Delivery as Dry Powder Inhalers
Authors: Alabsi, Wafaa; Acosta, Maria F.; Al-Obeidi, Fahad A.; Hay, Meredith; Polt, Robin; Mansour, Heidi M.
PaperDesign, synthesis, and biological evaluation of a multifunctional neuropeptide-Y conjugate for selective nuclear delivery of radiolanthanides
Chastel, Adrien; Worm, Dennis; Alves, Isabel et al. · 2020 · figshare · DOI
Full title: Design, synthesis, and biological evaluation of a multifunctional neuropeptide-Y conjugate for selective nuclear delivery of radiolanthanides
PaperSide-Chain Unprotected Fmoc-Arg/His/Tyr-OH Couplings and Their Application in Solid-Phase Peptide Synthesis through a Minimal-Protection/Green Chemistry Strategy
Yang, Yi; Hansen, Lena; Ryberg, Per · 2022 · Organic Process Research & Development · DOI
Full title: Side-Chain Unprotected Fmoc-Arg/His/Tyr-OH Couplings and Their Application in Solid-Phase Peptide Synthesis through a Minimal-Protection/Green Chemistry Strategy
PaperNatural Plasmodium falciparum Infection Stimulates Human Antibodies to MSP1 Epitopes Identified in Mice Infection Models upon Non-Natural Modified Peptidomimetic Vaccination
Rodríguez, Zully Johana; Melo, Fredy Leonardo; Torres, Angela et al. · 2023 · Molecules · DOI
Full title: Natural Plasmodium falciparum Infection Stimulates Human Antibodies to MSP1 Epitopes Identified in Mice Infection Models upon Non-Natural Modified Peptidomimetic Vaccination
Authors: Rodríguez, Zully Johana; Melo, Fredy Leonardo; Torres, Angela; Agrawal, Nikhil; Cortés-Vecino, Jesús Alfredo; Lozano, José Manuel
PaperThe Effect of Counterion and Tertiary Amine on the Efficiency of <i>N</i>‐Triazinylammonium Sulfonates in Solution and Solid‐Phase Peptide Synthesis
Kolesinska, Beata; Rozniakowski, Kamil K.; Fraczyk, Justyna et al. · 2015 · European Journal of Organic Chemistry · DOI
Full title: The Effect of Counterion and Tertiary Amine on the Efficiency of <i>N</i>‐Triazinylammonium Sulfonates in Solution and Solid‐Phase Peptide Synthesis
Authors: Kolesinska, Beata; Rozniakowski, Kamil K.; Fraczyk, Justyna; Relich, Inga; Papini, Anna Maria; Kaminski, Zbigniew J.
PaperUltrasonic-Assisted Solid-Phase Peptide Synthesis of DOTA-TATE and DOTA-<i>linker</i>-TATE Derivatives as a Simple and Low-Cost Method for the Facile Synthesis of Chelator–Peptide Conjugates
Raheem, Shvan J.; Schmidt, Benjamin W.; Solomon, Viswas Raja et al. · 2021 · Bioconjugate Chemistry · DOI
Full title: Ultrasonic-Assisted Solid-Phase Peptide Synthesis of DOTA-TATE and DOTA-<i>linker</i>-TATE Derivatives as a Simple and Low-Cost Method for the Facile Synthesis of Chelator–Peptide Conjugates
Authors: Raheem, Shvan J.; Schmidt, Benjamin W.; Solomon, Viswas Raja; Salih, Akam K.; Price, Eric W.
PaperCover Feature: Upscaled Synthesis of α‐ and β‐Peptides in a Continuous‐Flow Reactor Using Propylene Carbonate as an Eco‐Friendly Solvent (Chem. Methods 8/2025)
Varró, Nikolett; Mándityné Huszka, Beáta; Erdei, Eszter et al. · 2025 · Chemistry–Methods · DOI
Full title: Cover Feature: Upscaled Synthesis of α‐ and β‐Peptides in a Continuous‐Flow Reactor Using Propylene Carbonate as an Eco‐Friendly Solvent (Chem. Methods 8/2025)
Authors: Varró, Nikolett; Mándityné Huszka, Beáta; Erdei, Eszter; Mándoki, András; Mándity, István M.
PaperSmall animal PET imaging with the 68Ga-labeled pH (low) insertion peptide-like peptide YJL-4 in a triple-negative breast cancer mouse model
Chen, YueHua; Song, ShuangShuang; Sun, YanQin et al. · 2024 · figshare · DOI
Full title: Small animal PET imaging with the 68Ga-labeled pH (low) insertion peptide-like peptide YJL-4 in a triple-negative breast cancer mouse model
PaperStructure-Function Studies of Polymyxin B Lipononapeptides
Gallardo-Godoy, Alejandra; Hansford, Karl A.; Muldoon, Craig et al. · 2019 · Molecules · DOI
Full title: Structure-Function Studies of Polymyxin B Lipononapeptides
Authors: Gallardo-Godoy, Alejandra; Hansford, Karl A.; Muldoon, Craig; Becker, Bernd; Elliott, Alysha G.; Huang, Johnny X.; Pelingon, Ruby; Butler, Mark S.; Blaskovich, Mark A. T.; Cooper, Matthew A.
Full title: A straightforward method to prevent the under-estimated problem of aspartimide formation during chemical ligation-mediated protein synthesis
PaperThe application of anisole in greener solid-phase peptide synthesis protocols – Compatibility with green bases in Fmoc removal and new green binary mixture for coupling
Přibylka, Adam; Pastorek, Milan; Grepl, Martin et al. · 2021 · Tetrahedron · DOI
Full title: The application of anisole in greener solid-phase peptide synthesis protocols – Compatibility with green bases in Fmoc removal and new green binary mixture for coupling
Authors: Přibylka, Adam; Pastorek, Milan; Grepl, Martin; Schütznerová, Eva Přibylka
PaperEnvironmentally Friendly SPPS II: Scope of Green Fmoc Removal Protocol Using NaOH and Its Application for Synthesis of Commercial Drug Triptorelin
Přibylka, Adam; Krchňák, Viktor; Schütznerová, Eva · 2020 · The Journal of Organic Chemistry · DOI
Full title: Environmentally Friendly SPPS II: Scope of Green Fmoc Removal Protocol Using NaOH and Its Application for Synthesis of Commercial Drug Triptorelin
Authors: Přibylka, Adam; Krchňák, Viktor; Schütznerová, Eva
PaperAqueous microwave-assisted solid-phase peptide synthesis using Fmoc strategy. III: Racemization studies and water-based synthesis of histidine-containing peptides
Hojo, Keiko; Shinozaki, Natsuki; Hidaka, Koushi et al. · 2014 · Amino Acids · DOI
Full title: Aqueous microwave-assisted solid-phase peptide synthesis using Fmoc strategy. III: Racemization studies and water-based synthesis of histidine-containing peptides
Authors: Hojo, Keiko; Shinozaki, Natsuki; Hidaka, Koushi; Tsuda, Yuko; Fukumori, Yoshinobu; Ichikawa, Hideki; Wade, John D.
PaperNew green base for Fmoc removal in solid-phase peptide synthesis: 1,5-diazabicyclo[4.3.0]non-5-ene (DBN), a promising sustainable alternative to piperidine
Scala, Maria Carmina; Vivenzio, Giovanni; Manfra, Michele et al. · 2025 · Green Chemistry Letters and Reviews · DOI
Full title: New green base for Fmoc removal in solid-phase peptide synthesis: 1,5-diazabicyclo[4.3.0]non-5-ene (DBN), a promising sustainable alternative to piperidine
Authors: Scala, Maria Carmina; Vivenzio, Giovanni; Manfra, Michele; Sala, Marina; Campiglia, Pietro
PaperI. Synthesis and Bioactivity of Novel Proteasome Inhibiting Syrbactins and II. Peptide Assembly by Ligation of Hydroxyl Amino Acids and Mildly Activated Esters
Bakas, Nicole A. · 2017 · eScholarship (California Digital Library)
Full title: I. Synthesis and Bioactivity of Novel Proteasome Inhibiting Syrbactins and II. Peptide Assembly by Ligation of Hydroxyl Amino Acids and Mildly Activated Esters
Authors: Bakas, Nicole A.
Year: 2017
Venue: eScholarship (California Digital Library)
PaperQuantum Defects as a Toolbox for the Covalent Functionalization of Carbon Nanotubes with Peptides and Proteins
Mann, Florian A.; Herrmann, Niklas; Opazo, Felipe et al. · 2020 · Angewandte Chemie International Edition · DOI
Full title: Quantum Defects as a Toolbox for the Covalent Functionalization of Carbon Nanotubes with Peptides and Proteins
Authors: Mann, Florian A.; Herrmann, Niklas; Opazo, Felipe; Kruss, Sebastian
PaperOptimization of peptide synthesis time and sustainability using novel eco‐friendly binary solvent systems with induction heating on an automated peptide synthesizer
Pacini, Lorenzo; Muthyala, Manoj; Aguiar, Luisa et al. · 2024 · Journal of Peptide Science · DOI
Full title: Optimization of peptide synthesis time and sustainability using novel eco‐friendly binary solvent systems with induction heating on an automated peptide synthesizer
Authors: Pacini, Lorenzo; Muthyala, Manoj; Aguiar, Luisa; Zitterbart, Robert; Rovero, Paolo; Papini, Anna Maria
PaperStructural and functional properties of the Kunitz-type and C-terminal domains of Amblyomin-X supporting its antitumor activity
Morais, K. L. P.; Ciccone, L.; Stura, E. et al. · 2023 · Frontiers in Molecular Biosciences · DOI
Full title: Structural and functional properties of the Kunitz-type and C-terminal domains of Amblyomin-X supporting its antitumor activity
Authors: Morais, K. L. P.; Ciccone, L.; Stura, E.; Alvarez-Flores, M. P.; Mourier, G.; Driessche, M. Vanden; Sciani, J. M.; Iqbal, A.; Kalil, S. P.; Pereira, G. J.; Marques-Porto, R.; Cunegundes, P.; Juliano, L.; Servent, D.; Chudzinski-Tavassi, A. M.
PaperRe-evaluating the stability of COMU in different solvents.
Kumar, Ashish; Jad, Yahya E; de la Torre, Beatriz G et al. · 2017 · Journal of peptide science : an official publication of the European Peptide Society · DOI
Full title: Re-evaluating the stability of COMU in different solvents.
Authors: Kumar, Ashish; Jad, Yahya E; de la Torre, Beatriz G; El-Faham, Ayman; Albericio, Fernando
Year: 2017
Venue: Journal of peptide science : an official publication of the European Peptide Society
PaperSelf-Assembly of a Novel Pentapeptide into Hydrogelated Dendritic Architecture: Synthesis, Properties, Molecular Docking and Prospective Applications
Jitaru, Stefania-Claudia; Enache, Andra-Cristina; Cojocaru, Corneliu et al. · 2024 · Gels · DOI
Full title: Self-Assembly of a Novel Pentapeptide into Hydrogelated Dendritic Architecture: Synthesis, Properties, Molecular Docking and Prospective Applications
Authors: Jitaru, Stefania-Claudia; Enache, Andra-Cristina; Cojocaru, Corneliu; Drochioiu, Gabi; Petre, Brîndușa Alina; Grădinaru, Vasile Robert
PaperExpanding the Structural Biologist's Tool Chest by Chemical and Biocompatible Modification of Peptides: from Characterizing Marine Snail Toxins to OutPHOXIng Tryptophan
Grigoryan, Alexander · 2015 · CUNY Academic Works (City University of New York)
Full title: Expanding the Structural Biologist's Tool Chest by Chemical and Biocompatible Modification of Peptides: from Characterizing Marine Snail Toxins to OutPHOXIng Tryptophan
Authors: Grigoryan, Alexander
Year: 2015
Venue: CUNY Academic Works (City University of New York)
PaperTroubleshooting When Using γ-Valerolactone (GVL) in Green Solid-Phase Peptide Synthesis
Kumar, Ashish; Thompson-Adewumi, Adeniyi; Nandhini, K. P. et al. · 2019 · Organic Process Research & Development · DOI
Full title: Troubleshooting When Using γ-Valerolactone (GVL) in Green Solid-Phase Peptide Synthesis
Authors: Kumar, Ashish; Thompson-Adewumi, Adeniyi; Nandhini, K. P.; Collins, Jonathan M.; Albericio, Fernando; de la Torre, Beatriz G.
Successful development of a method for the incorporation of Fmoc-Arg(Pbf)-OH in solid-phase peptide synthesis using <i>N</i>-butylpyrrolidinone (NBP) as solvent
de la Torre, Beatriz G.; Kumar, Ashish; Alhassan, Mahama et al. · 2020
Full title: Successful development of a method for the incorporation of Fmoc-Arg(Pbf)-OH in solid-phase peptide synthesis using <i>N</i>-butylpyrrolidinone (NBP) as solvent
Authors: de la Torre, Beatriz G.; Kumar, Ashish; Alhassan, Mahama; Bucher, Christoph; Albericio, Fernando; Lopez, John
Green solvents and Safe Reagents in SPPS taking advantage of induction heating and automation: synthesis and HPLC-free purification of difficult sequences
Pacini, L.; Muthyala, M.; Marder, O. et al. · 2024
Full title: Green solvents and Safe Reagents in SPPS taking advantage of induction heating and automation: synthesis and HPLC-free purification of difficult sequences
Authors: Pacini, L.; Muthyala, M.; Marder, O.; Aguiar, L.; Zitterbart, R.; Rovero, P.; Papini, A.
Highlighting multicomponent reactions as an efficient and facile alternative route in the chemical synthesis of organic-based molecules: a tremendous growth in the past 5 years
Full title: Highlighting multicomponent reactions as an efficient and facile alternative route in the chemical synthesis of organic-based molecules: a tremendous growth in the past 5 years
Authors: Mohlala, Reagan Lehlogonolo; Rashamuse, Thompho Jason; Coyanis, Elena Mabel
Green solvent mixture for ultrasound-assisted solid-phase peptide synthesis: a fast and versatile method and its applications in flow and natural product synthesis
Liao, Jingyuan; Zhang, Renrong; Jia, Xuelei et al. · 2024
Full title: Green solvent mixture for ultrasound-assisted solid-phase peptide synthesis: a fast and versatile method and its applications in flow and natural product synthesis
Total Synthesis of Novel Antimicrobial β-Hairpin Capitellacin Via Rapid Flow-Based SPPS Assembly and Regioselective On-Resin Disulfide Cyclisation
Shepperson, Oscar A.; Hanna, Cameron C.; Brimble, Margaret A. et al. · 2022
Full title: Total Synthesis of Novel Antimicrobial β-Hairpin Capitellacin Via Rapid Flow-Based SPPS Assembly and Regioselective On-Resin Disulfide Cyclisation
Authors: Shepperson, Oscar A.; Hanna, Cameron C.; Brimble, Margaret A.; Harris, Paul W. R.; Cameron, Alan J.
Investigation of bioactive natural compounds for cardiovascular diseases and daqu fermentation, and the exploration of Beauveria bassiana as a biocontrol agent for the mountain pine beetle epidemic
Fernandez, Kleinberg Xiandrell · 2024
Full title: Investigation of bioactive natural compounds for cardiovascular diseases and daqu fermentation, and the exploration of Beauveria bassiana as a biocontrol agent for the mountain pine beetle epidemic
Development of synthetic strategies towards libraries of heterocyclic and bicyclic inhibitors of Cdc25A & development of solid phase synthesis of cyclic peptides
Luo, Hao · 2015
Full title: Development of synthetic strategies towards libraries of heterocyclic and bicyclic inhibitors of Cdc25A & development of solid phase synthesis of cyclic peptides
Scalable and Sustainable DMF-Free Solid-Phase Synthesis of Liraglutide by 1-Tert-Butyl-3-Ethylcarbodiimide-Mediated Couplings and Catch-and-Release Acylation and Purification Strategies
Pacini, Lorenzo; Muthyala, Manoj Kumar; Zitterbart, Robert et al. · 2025
Full title: Scalable and Sustainable DMF-Free Solid-Phase Synthesis of Liraglutide by 1-Tert-Butyl-3-Ethylcarbodiimide-Mediated Couplings and Catch-and-Release Acylation and Purification Strategies
Authors: Pacini, Lorenzo; Muthyala, Manoj Kumar; Zitterbart, Robert; Marder, Oleg; Rovero, Paolo; Papini, Anna Maria
Bypassing Osmotic Shock Dilemma in a Polystyrene Resin Using the Green Solvent Cyclopentyl methyl Ether (CPME): A Morphological Perspective
Al Musaimi, Othman; El-Faham, Ayman; Almarhoon, Zainab et al. · 2019
Full title: Bypassing Osmotic Shock Dilemma in a Polystyrene Resin Using the Green Solvent Cyclopentyl methyl Ether (CPME): A Morphological Perspective
Authors: Al Musaimi, Othman; El-Faham, Ayman; Almarhoon, Zainab; Basso, Alessandra; de la Torre, Beatriz G.; Albericio, Fernando
Efficient generation of recombinant hydrazides for the production of scarce proteins and development of chemical probes for detecting protein sulfenylation
Ekanayake, Oshini · 2020
Full title: Efficient generation of recombinant hydrazides for the production of scarce proteins and development of chemical probes for detecting protein sulfenylation
Application of a new green protocol in Solid-Phase Peptide Synthesis: identification of a new green solvent mixture compatible with ETT/TBEC
Vivenzio, G.; Scala, M.; Campiglia, P. et al. · 2024
Full title: Application of a new green protocol in Solid-Phase Peptide Synthesis: identification of a new green solvent mixture compatible with ETT/TBEC
Authors: Vivenzio, G.; Scala, M.; Campiglia, P.; Sala, M.
Replacing DMF in solid-phase peptide synthesis: varying the composition of green binary solvent mixtures as a tool to mitigate common side-reactions
Jadhav, Sandip; Martin, Vincent; Egelund, Peter H. G. et al. · 2021
Full title: Replacing DMF in solid-phase peptide synthesis: varying the composition of green binary solvent mixtures as a tool to mitigate common side-reactions
Authors: Jadhav, Sandip; Martin, Vincent; Egelund, Peter H. G.; Johansson Castro, Henrik; Krüger, Tobias; Richner, Franziska; Thordal Le Quement, Sebastian; Albericio, Fernando; Dettner, Frank; Lechner, Carolin; Schönleber, Ralph; Pedersen, Daniel Sejer
Silylated Tag-Assisted Peptide Synthesis: Continuous One-Pot Elongation for the Production of Difficult Peptides under Environmentally Friendly Conditions
Full title: Silylated Tag-Assisted Peptide Synthesis: Continuous One-Pot Elongation for the Production of Difficult Peptides under Environmentally Friendly Conditions
Solid-Phase Peptide Synthesis of Dipeptide (Histidine-β-Alanine) as a Chelating Agent by Using Trityl Chloride Resin, for Removal of Al<sup>3+</sup>, Cu<sup>2+</sup>, Hg<sup>2+</sup>and Pb<sup>2+</sup>: Experimental and Theoretical Study
Rahimi, Rahmatollah; Khosravi, Maryam; Tehrani, Mohammd H. H. et al. · 2016
Full title: Solid-Phase Peptide Synthesis of Dipeptide (Histidine-β-Alanine) as a Chelating Agent by Using Trityl Chloride Resin, for Removal of Al<sup>3+</sup>, Cu<sup>2+</sup>, Hg<sup>2+</sup>and Pb<sup>2+</sup>: Experimental and Theoretical Study
A practical method for the synthesis of small peptides using DCC and HOBt as activators in H2O–THF while avoiding the use of protecting groups†
Herrera-Guzmán, Karina; Jaime-Vasconcelos, Miguel Ángel; Torales, Eréndira et al. · 2024
Full title: A practical method for the synthesis of small peptides using DCC and HOBt as activators in H2O–THF while avoiding the use of protecting groups†
Authors: Herrera-Guzmán, Karina; Jaime-Vasconcelos, Miguel Ángel; Torales, Eréndira; Chacón, Itzel; Gaviño, Rubén; García-Ríos, Eréndira; Cárdenas, Jorge; Morales-Serna, José A.
Scalable and Sustainable DMF-Free Solid-Phase Synthesis of Liraglutide by 1-Tert-Butyl-3-Ethylcarbodiimide-Mediated Couplings and Catch-and-Release Acylation and Purification Strategies
Pacini, Lorenzo; Muthyala, Manoj Kumar; Zitterbart, Robert et al. · 2025
Full title: Scalable and Sustainable DMF-Free Solid-Phase Synthesis of Liraglutide by 1-Tert-Butyl-3-Ethylcarbodiimide-Mediated Couplings and Catch-and-Release Acylation and Purification Strategies
Authors: Pacini, Lorenzo; Muthyala, Manoj Kumar; Zitterbart, Robert; Marder, Oleg; Rovero, Paolo; Papini, Anna Maria
Key Green Chemistry research areas from a pharmaceutical manufacturers’ perspective revisited
Bryan, Marian C.; Dunn, Peter J.; Entwistle, David A. et al. · 2018
Full title: Key Green Chemistry research areas from a pharmaceutical manufacturers’ perspective revisited
Authors: Bryan, Marian C.; Dunn, Peter J.; Entwistle, David A.; Gallou, Fabrice; Koenig, Stefan G.; Hayler, John; Hickey, Matthew; Hughes, Shaun; Kopach, Michael E.; Moine, Gérard; Richardson, Paul; Roschangar, Frank; Steven, Alan; Weiberth, Franz J.
Green Solvent Mixtures for Solid-Phase Peptide Synthesis: A Dimethylformamide-Free Highly Efficient Synthesis of Pharmaceutical-Grade Peptides
Ferrazzano, Lucia; Corbisiero, Dario; Martelli, Giulia et al. · 2019
Full title: Green Solvent Mixtures for Solid-Phase Peptide Synthesis: A Dimethylformamide-Free Highly Efficient Synthesis of Pharmaceutical-Grade Peptides